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4-methyl-3-(2-{2-[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]-1H-imidazol-1-yl}ethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[3-(4-methyl-1,3-thiazol-2-yl)propyl]-4-(piperidin-1-ylmethyl)benzamide
(4aR,7aS)-1-{2-[(6-methylpyridin-3-yl)oxy]acetyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(4aR,8aR)-2-cyclobutanecarbonyl-7-{[2-(difluoromethoxy)phenyl]methyl}-decahydro-2,7-naphthyridin-4a-ol
7-{[5-(4-chlorophenyl)furan-2-yl]methyl}-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
(2S,4S)-N-ethyl-1-methyl-4-[4-(piperidin-1-ylmethyl)benzamido]pyrrolidine-2-carboxamide
2-methyl-N-{[3-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-5-yl]methyl}quinoline-4-carboxamide
3-[3-(3-chlorophenyl)pyrrolidin-1-yl]-5-(5-methylfuran-2-yl)-1,2,4-triazine
5-({3-[4-(trifluoromethyl)phenyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}methyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-1-(2-methylphenyl)piperazin-2-one
N-[(3R)-4-hydroxy-3-methylbutyl]-5-{[(6-methylpyridin-3-yl)oxy]methyl}-1,2-oxazole-3-carboxamide
1-{2-[1-(2H-1,3-benzodioxol-5-yl)-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazol-5-yl]ethyl}-1H-1,2,3,4-tetrazole
N,N,5-trimethyl-2-{[1-(4-methyl-1,4-diazepan-1-yl)hex-5-en-2-yl]oxy}pyrimidin-4-amine
3-cyclopropyl-5-(3,3,3-trifluoropropyl)-1H-1,2,4-triazole
N-methyl-N-[1-(3-phenylpropyl)piperidin-3-yl]-1H-indole-2-carboxamide
5-[(3aR,6aS)-octahydropyrrolo[3,4-c]pyrrole-2-carbonyl]-N,N,4-trimethylpyrimidin-2-amine
N-{[1-(dimethylamino)cyclohexyl]methyl}-5-(pyrrolidin-2-yl)thiophene-2-carboxamide
3-(4-cyclohexylphenyl)-1-methyl-4-{octahydropyrrolo[1,2-a]piperazin-2-ylmethyl}-1H-pyrazole
[(3R,4S)-1-[(6-methoxynaphthalen-2-yl)methyl]-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
2-{2-[2-(4-fluorophenyl)azetidin-1-yl]-2-oxoethyl}-4-methyl-1,2-dihydrophthalazin-1-one
(1R,5R)-6-(3-methylbut-2-en-1-yl)-3-[6-(4H-1,2,4-triazol-4-yl)pyridine-3-carbonyl]-3,6-diazabicyclo[3.2.2]nonane
2-[(1R,5R)-3-benzoyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-1-(2,3-dihydro-1H-indol-1-yl)ethan-1-one
3-[(4-fluorophenyl)methyl]-5-methyl-5-{1-[3-(2-oxoimidazolidin-1-yl)benzoyl]piperidin-4-yl}imidazolidine-2,4-dione
methyl (2S,4S)-4-(2,4-dimethoxybenzamido)-1-{[3-(trifluoromethyl)phenyl]methyl}pyrrolidine-2-carboxylate
3-(4-ethyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)-1-{2-[(4-methylpyridin-2-yl)amino]ethyl}urea
2-hydroxy-4-methoxy-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]benzamide
N-cyclopentyl-5-[(4-hydroxypiperidin-1-yl)methyl]-N-propyl-1,2-oxazole-3-carboxamide
8-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one
2-(2-{1-[2-(methylsulfanyl)pyridine-3-carbonyl]piperidin-3-yl}-1H-imidazol-1-yl)acetamide
2-(4-{[({2-[(dimethylamino)methyl]phenyl}methyl)(methyl)amino]methyl}-3-methyl-1H-pyrazol-1-yl)ethan-1-ol
4-[3-cyclopropyl-1-(3,4-dimethylphenyl)-1H-1,2,4-triazol-5-yl]pyrimidine
ethyl 4-[(4-chlorophenyl)methyl]-1-(2-oxo-2-phenylacetyl)piperidine-4-carboxylate
4-(7-{[3-(dimethylamino)pyrrolidin-1-yl]sulfonyl}-1,2,3,4-tetrahydroisoquinolin-2-yl)-4-oxobutanamide
4-{[3-(2-fluorophenoxymethyl)piperidin-1-yl]methyl}pyridine
8-{5-[3-ethyl-4-(propan-2-yl)piperazine-1-carbonyl]pyridin-2-yl}-1,4-dioxa-8-azaspiro[4.5]decane
1-cyclohexyl-6-hydroxy-4-[(5-methylfuran-2-yl)methyl]-1,4-diazepan-2-one
1-(4-phenyl-1,2,3,6-tetrahydropyridin-1-yl)-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethan-1-one
1-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]-3-(4H-1,2,4-triazol-3-yl)piperidine
1-[4-({2-[4-(1H-pyrazol-1-ylmethyl)phenyl]-1H-imidazol-1-yl}methyl)piperidin-1-yl]ethan-1-one
2-{2-[(2,6-dichlorophenyl)methyl]pyrimidin-4-yl}pyridine-4-carboxylic acid
N3-butyl-N5-cyclopentyl-N3-methyl-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
1-[(2-fluorophenyl)methyl]-4-[3-(furan-2-yl)-1H-pyrazol-1-yl]piperidine-4-carboxylic acid
1-(furan-2-ylmethyl)-N-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}piperidine-4-carboxamide
1-[6-amino-2-(butylsulfanyl)pyrimidin-4-yl]-N-ethylpyrrolidine-3-carboxamide
1-[3-(1H-pyrazol-1-yl)propyl]-3-[3-(trifluoromethyl)benzoyl]piperidine
N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
2-[({6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)methyl]-3,4-dihydroquinazolin-4-one
[1-benzyl-5-(methoxymethyl)-1H-1,2,4-triazol-3-yl](phenyl)methanol
{1-[1-(diphenylmethyl)-1H-1,2,3-triazole-4-carbonyl]piperidin-3-yl}methanol
2-(5-chloro-1H-1,3-benzodiazol-2-yl)-N-[(1-propyl-1H-imidazol-2-yl)methyl]acetamide