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5-{[(2-fluorophenyl)methyl]amino}-N-(furan-2-ylmethyl)-N,1-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-{4-[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-4-oxobutyl}piperidin-2-one
(1R,7S)-6-(4-hydroxypiperidine-1-carbonyl)-3-[(3-methoxyphenyl)methyl]-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
(1-{2-[(3,4-dimethoxyphenyl)methyl]-1,3-benzoxazole-6-carbonyl}piperidin-2-yl)methanol
1-ethyl-N-[2-(1H-indol-3-yl)ethyl]-N-(pyridin-3-ylmethyl)-1H-pyrazole-3-carboxamide
8-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-N,2-dipropyl-2,8-diazaspiro[4.5]decane-3-carboxamide
2-{[5-(1-ethyl-1H-pyrazol-4-yl)-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
N-(1-{3-[3-(3-methylbutanoyl)piperidine-1-carbonyl]phenyl}-1H-pyrazol-4-yl)-2-(3-methylphenyl)acetamide
N-cyclopentyl-N-({3-[(4-fluorophenyl)methoxy]phenyl}methyl)-2H-1,3-benzodioxole-5-carboxamide
1-(4-ethyl-5-methylthiophene-3-carbonyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-(2-methoxyethyl)-1-methyl-N-[(5-methylthiophen-2-yl)methyl]piperidine-2-carboxamide
1-[3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]cyclopentan-1-ol
methyl 1-[(3R,5S)-5-[4-(4-fluorophenyl)piperazine-1-carbonyl]-1-[(4-methoxy-2,5-dimethylphenyl)methyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
3-{[(4-fluorophenyl)methyl]sulfanyl}-N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]propanamide
6-{4-[(dimethylamino)methyl]phenyl}naphthalen-2-ol
N-(2-fluoroethyl)-3-{[(3-methoxyphenyl)methyl](methyl)sulfamoyl}benzamide
N-(2-hydroxyethyl)-N-(1,3-thiazol-2-ylmethyl)-[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carboxamide
1-(6-{4-[(3-methylphenyl)methyl]piperazin-1-yl}pyrimidin-4-yl)piperidin-4-ol
2-(adamantan-1-ylsulfanyl)-N-methyl-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]acetamide
(1s,4s)-4-(4-phenyl-1,4-diazepane-1-carbonyl)cyclohexan-1-ol
1-{3-[3-(5-methylfuran-2-yl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]propyl}piperidin-2-one
4-[6-(2,4-dichlorophenyl)pyrimidin-4-yl]morpholine
4-methoxy-N-(2-{4-[(4-phenylpiperidin-1-yl)methyl]phenoxy}propyl)benzamide
1-{3-[(2,3-dihydro-1,4-benzodioxin-6-yl)amino]piperidin-1-yl}-2-(pyridin-2-ylsulfanyl)ethan-1-one
1-[2-methyl-4-(2-methylphenyl)piperazin-1-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
3-[1-(6-ethyl-2-oxo-1,2-dihydropyridin-4-yl)-N-(2-phenylethyl)formamido]propanamide
N,1,3-trimethyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
4-[5-(2-{5-[2-(methylsulfanyl)ethyl]-4-phenyl-1H-imidazol-1-yl}ethyl)-1H-1,2,4-triazol-3-yl]pyridine
1-(2H-1,3-benzodioxole-5-carbonyl)-3-(naphthalene-1-carbonyl)piperidine
N-cyclopentyl-N-{[4-methoxy-3-(propan-2-yloxy)phenyl]methyl}-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
(3-{2-[1-(4,6-dimethylpyrimidin-2-yl)piperidin-4-yl]-1H-imidazol-1-yl}propyl)dimethylamine
2-[6-(5-chloro-2-methoxypyridin-4-yl)pyridin-3-yl]acetic acid
4-(2-{1-[4-(1H-1,2,4-triazol-3-yl)benzoyl]piperidin-2-yl}ethyl)morpholine
2-(3-hydroxyphenyl)-1-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-7H-pyrrolo[2,3-d]pyrimidin-4-amine
1-ethyl-4-[2-(2-methylphenyl)pyrrolidine-1-carbonyl]-1,2-dihydropyridin-2-one
2-amino-5-methyl-6-(1-methyl-1H-pyrazol-4-yl)-4-(2-phenylpyrimidin-5-yl)pyridine-3-carbonitrile
2-(1-ethyl-1H-pyrazol-4-yl)-6-fluoro-N-methyl-N-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]quinoline-4-carboxamide
N-cyclobutyl-1-[1-(propan-2-yl)piperidin-4-yl]piperidine-3-carboxamide
3,5-dichloro-N,4-dimethyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]benzamide
(1-{2-amino-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperidin-4-yl)(phenyl)methanol
(2S,3R)-2-amino-1-[2,4-bis(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-3-hydroxybutan-1-one
1-[(3-fluorophenyl)methyl]-4-[2-(1H-pyrazol-1-yl)benzoyl]piperazine
2-{2-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-2,7-diazaspiro[4.5]decan-6-one
(3aS,6aS)-N-[4-(2-methylphenyl)phenyl]-octahydropyrrolo[2,3-c]pyrrole-1-carboxamide
N-[5-(4-cyclohexylpiperazine-1-carbonyl)-7-oxo-4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl]-3-fluorobenzamide
{[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}[2-(pyridin-2-yl)ethyl]amine
N-[2-(3-oxopiperazine-1-carbonyl)phenyl]-2,5-dihydro-1H-pyrrole-2-carboxamide
N,N-dimethyl-2-(5-methyl-1,2-oxazole-4-sulfonamidomethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
N-{2-methyl-4-[3-(1,2-oxazinan-2-yl)propanamido]phenyl}pentanamide