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N-(3-{3-[4-(2-methylphenyl)piperazin-1-yl]piperidine-1-carbonyl}phenyl)acetamide
N-[2-(3,4-dimethoxyphenyl)ethyl]-1-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]-N-methylpiperidin-3-amine
N-{3-[({5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}carbamoyl)methoxy]phenyl}propanamide
1-(4-benzylpiperidin-1-yl)-3-{1-[(1R,2S,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]piperidin-4-yl}propan-1-one
N-[2-({2-[(4-methoxyphenyl)methyl]-1,3-benzoxazol-6-yl}formamido)ethyl]acetamide
3-{1-[(2-hydroxy-4-methoxyphenyl)methyl]piperidin-3-yl}-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
3-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraene
N-(3-carbamoylphenyl)-4-(1-hydroxy-3-phenylpropyl)piperidine-1-carboxamide
2-{4-[1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)pyrrolidin-3-yl]piperidin-1-yl}pyrimidine
5-chloro-N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-3-phenyl-1H-indole-2-carboxamide
3-{2-[methyl(2-phenylethyl)amino]ethyl}-8-(oxan-3-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
{2-oxo-2-[4-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]ethyl}urea
N-({5-methyl-2-[2-(3-phenoxypropanamido)phenyl]-1,3-oxazol-4-yl}methyl)cyclopropanecarboxamide
1-methyl-3-(propan-2-yl)-8-{[4-(pyrrolidin-1-yl)phenyl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[(1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidin-4-yl)formamido]acetamide
1-{[2-(4-methoxyphenyl)-7-methylquinolin-3-yl]methyl}-2-methyl-1,4-diazepan-5-one
N-[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]-3-[(1H-pyrazol-3-ylmethyl)sulfamoyl]benzamide
4-[1-(3,5-dimethylphenyl)-3-phenyl-1H-1,2,4-triazol-5-yl]-1-methylpyrrolidin-2-one
2-(1-{1-[4-(1H-indol-3-yl)butan-2-yl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)propan-2-amine
(2R,3S,6R)-5-cyclopropanecarbonyl-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-(1,4-diazepane-1-carbonyl)-N-methyl-N-(2-phenylethyl)-2,3-dihydro-1H-inden-2-amine
(2S)-N2-ethyl-N1-[2-(4-fluorophenoxy)pyridin-3-yl]pyrrolidine-1,2-dicarboxamide
4-(4-acetamido-1H-pyrazol-1-yl)-N-[3-(1H-imidazol-1-yl)-1-phenylpropyl]benzamide
2,6-dimethyl-4-[4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]quinoline
ethyl 4-[2-(pyrrolidin-1-yl)-5,6,7,8-tetrahydroquinazoline-4-amido]piperidine-1-carboxylate
5-(4-methoxyphenyl)-N-[(5-methyl-1,2-oxazol-3-yl)methyl]furan-2-carboxamide
2-(1,5-dimethyl-1H-pyrazol-4-yl)-7-(3-methoxyphenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-methyl-4-(1-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}ethyl)piperazine
N-[1-(2,5-dimethylphenyl)ethyl]-2-(2,5-dioxoimidazolidin-1-yl)acetamide
N-[2-(3,5-dimethoxyphenyl)ethyl]-6-ethyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-(cyclohexylmethyl)-N-methyl-5-({[1-(morpholin-4-yl)cyclopentyl]methyl}amino)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
ethyl 2-{[(1-cycloheptyl-5-oxopyrrolidin-3-yl)carbamoyl]amino}acetate
3-ethyl-1-[1-(4-methoxyphenyl)cyclopropanecarbonyl]piperidine-3-carboxylic acid
{5-[(7-{[4-(benzyloxy)piperidin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)methyl]furan-2-yl}methanol
methyl 4-{[4-(2-{[2-(dimethylamino)ethyl]carbamoyl}ethyl)piperidin-1-yl]methyl}benzoate
(1-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}-4-{[2-(trifluoromethyl)phenyl]methyl}piperidin-4-yl)methanol
[(4-methoxy-2-methylphenyl)methyl](methyl)(oxan-2-ylmethyl)amine
3-{2-[4-(2-chlorophenyl)piperazin-1-yl]-2-oxoethyl}-4-(pyridin-2-ylmethyl)piperazin-2-one
1-ethyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]piperidine-4-carboxamide
(2R,3R,6R)-5-(3-fluoropyridine-4-carbonyl)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
3-(3-methoxyphenyl)-N-(thiolan-3-yl)-1H-pyrazole-5-carboxamide
3-ethyl-3-methyl-4-[2-(thiophen-2-yl)acetyl]piperazin-2-one
1-[1'-(1H-pyrazole-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
3-{1-[4-(2-oxopyrrolidin-1-yl)benzoyl]piperidin-4-yl}benzonitrile
N-(furan-2-ylmethyl)-7-(propan-2-yl)-N-(thiophen-2-ylmethyl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
N-(oxolan-2-ylmethyl)-3-(1H-pyrazol-1-ylmethyl)benzamide
1-[(3-fluorophenyl)methyl]-4-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]piperazin-2-one
3-chloro-4-[(1-methanesulfonylpiperidin-4-yl)oxy]-N-[2-(pyridin-2-yl)ethyl]benzamide
1-(1-{2-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-5-methoxybenzoyl}piperidin-4-yl)propan-1-ol
(3S,4S)-4-(3-methoxyphenyl)-1-[(6-methylpyridin-2-yl)methyl]piperidin-3-ol