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3-{1-[1-(4-chlorophenyl)cyclobutanecarbonyl]piperidin-3-yl}-1-(pyrrolidin-1-yl)propan-1-one
{2-[4-amino-6-(benzylamino)-1,3,5-triazin-2-yl]phenyl}methanol
(4aS,8aR)-1-(2-aminoethyl)-6-(1H-indol-2-ylmethyl)-decahydro-1,6-naphthyridin-2-one
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-2-ethoxypyridine-3-carboxamide
N-(2-ethyl-2H-1,2,3-triazol-4-yl)-2-[5-(thiophen-2-yl)-1H-indazol-1-yl]acetamide
2-{2-[1-(5-chlorothiophene-2-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}acetamide
3-(3,5-dimethylbenzoyl)-9-methoxy-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
2-[(2-amino-5-ethylpyrimidin-4-yl)(methyl)amino]-N-butylacetamide
4-({3-[2-(4-{4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzoyl}piperazin-1-yl)ethoxy]phenyl}methyl)morpholine
5-[5-(methoxymethyl)furan-2-carbonyl]-2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
1-(2,6-difluoro-4-methoxybenzoyl)-4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
1-[5-(propan-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonyl]piperidine-3-carboxamide
3-{3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}-N-methylpropanamide
4-[(3S,4R)-3-cyclopropyl-4-(dimethylamino)pyrrolidine-1-carbonyl]-1-ethyl-1,2-dihydropyridin-2-one
N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-1-(2-phenylethyl)-1H-1,2,3-triazole-4-carboxamide
4-{4-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]piperazin-1-yl}-2-(methylsulfanyl)pyrimidine
4-({[2-(2-ethoxyphenoxy)ethyl](methyl)amino}methyl)-N-methylbenzene-1-sulfonamide
1-{3-[7-(3,6-dimethylpyrazin-2-yl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl]phenyl}imidazolidin-2-one
1-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-2-[2-(1-methyl-1H-imidazol-2-yl)ethyl]piperidine
1-(5-ethyl-1,3,4-oxadiazol-2-yl)-4-(furan-2-carbonyl)piperazine
1-[4-(methylsulfanyl)butan-2-yl]-4-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperazine
3-(2-methyl-1H-indol-1-yl)-N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}propanamide
3-{[4-benzyl-3-(2-hydroxyethyl)piperazin-1-yl]methyl}phenol
2-(2-amino-5,6,7,8-tetrahydroquinazoline-4-carbonyl)-7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decan-6-one
3-methyl-4-{1-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carbonyl]pyrrolidin-2-yl}-1,2,5-oxadiazole
dimethyl(2-{2-[1-(pyridin-2-yl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)amine
4-{1-[1-(6-methoxypyrimidin-4-yl)piperidin-4-yl]piperidine-3-carbonyl}morpholine
1-methyl-5-[4-(2-phenoxyacetyl)piperazine-1-carbonyl]-1H-pyrrole-3-carbonitrile
[1-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)-4-(2-phenoxyethyl)piperidin-4-yl]methanol
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-1-methyl-1H-indole-6-carboxamide
6-[(diethylamino)methyl]-N-[1-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
N-[2-(propan-2-ylsulfanyl)ethyl]-4-(pyrrolidin-1-ylmethyl)benzamide
N-[(1-cyclopentylpiperidin-4-yl)methyl]-2-(propan-2-yl)-N-(pyridin-3-ylmethyl)-1,3-thiazole-4-carboxamide
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-1-(pyridine-4-carbonyl)piperidin-4-amine
2-[(1S,5R)-3-[(2-fluoro-4-methoxyphenyl)methyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
4-[3-(2-chloro-4-fluorophenyl)phenyl]-4H-1,2,4-triazole
N-[(5-chloro-2-ethoxyphenyl)methyl]-N-methyl-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
2-[(2-fluorophenyl)methyl]-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}-1,3-benzoxazole-6-carboxamide
ethyl 1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-3-[(2E)-3-phenylprop-2-en-1-yl]piperidine-3-carboxylate
2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1-(5,6,7,8-tetrahydronaphthalen-1-yl)-1H-imidazole
2-methoxy-N-({5-[(1-methyl-1H-indol-4-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)acetamide
5-(2-methylphenyl)pyrazin-2-amine
N5-[(3-fluorophenyl)methyl]-N3-methyl-N3-(2-methylpropyl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
dimethyl(2-{2-[1-(pyrrolidine-1-sulfonyl)piperidin-4-yl]-1H-imidazol-1-yl}ethyl)amine
1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidine
N-[1-(methoxymethyl)cyclopentyl]-2,3-dihydro-1H-indene-1-carboxamide
4-{1-cyclohexyl-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl}-6-(2-methylpropyl)-1,2-dihydropyrimidin-2-one
2-(2-butylpyrimidin-4-yl)pyridine-4-carboxylic acid
1-benzyl-N-methyl-N-({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)piperidin-4-amine
dimethyl(1-{1-[4-methyl-2-(pyridin-3-yl)pyrimidine-5-carbonyl]piperidin-4-yl}ethyl)amine