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2-[2-(2,3-dihydro-1,4-benzodioxin-6-yl)-1H-1,3-benzodiazol-1-yl]ethan-1-ol
[2-(1H-imidazol-4-yl)ethyl]({[2-(naphthalen-2-yl)pyrimidin-5-yl]methyl})amine
6-methoxy-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-{[5-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-4-(thiophen-2-yl)butanamide
N-cyclopropyl-N-[(2-methoxyphenyl)methyl]-4-(4-methylpiperazin-1-yl)pentanamide
ethyl 1-[(1-ethyl-1H-imidazol-2-yl)methyl]-3-[(3-methoxyphenyl)methyl]piperidine-3-carboxylate
2-[5-(3-methoxyphenoxymethyl)-1H-pyrazole-3-carbonyl]-1,2-oxazolidine
3-(4H-1,2,4-triazol-4-yl)-5,6,7,8-tetrahydronaphthalen-2-ol
4-[(3-fluorophenyl)methyl]-1-{[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]methyl}-1,4-diazepan-5-one
N-[1-(2-phenylethyl)piperidin-3-yl]oxane-4-carboxamide
N-[1-(2,4-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-oxo-2,3-dihydro-1H-imidazole-4-carboxamide
2-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)-7-(2-phenylethyl)-2,7-diazaspiro[4.5]decane
2-{6-[4-(diethylsulfamoyl)phenyl]pyridin-3-yl}acetic acid
1-{1-[(5-chlorothiophen-2-yl)methyl]piperidin-4-yl}-N-(2-methoxyethyl)piperidine-3-carboxamide
N-(4-butylphenyl)-4-(pyridin-3-yl)piperazine-1-carboxamide
3-[3-ethyl-4-(4-fluorophenyl)-1-methyl-1H-pyrazol-5-yl]-1-[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]urea
8-methoxy-N-[3-(methylsulfanyl)propyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
(1S,2R)-N1-[2-(1H-1,2,3-benzotriazol-1-yl)ethyl]-N2-tert-butylcyclohexane-1,2-dicarboxamide
(2S,4S)-1-cyclobutanecarbonyl-N-ethyl-4-(6-methyl-4-oxo-4H-pyran-2-amido)pyrrolidine-2-carboxamide
3-{2-[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]-2-oxoethyl}-1,3-diazinane-2,4-dione
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[2-(N-methylmethanesulfonamido)ethyl]benzamide
1-[(2-fluorophenyl)methyl]-3-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine
1-[(3R,4R)-4-amino-3-hydroxypiperidin-1-yl]-3-(3-methoxy-4-methylphenyl)propan-1-one
N-[(3-chlorophenyl)methyl]-3-[1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)piperidin-4-yl]propanamide
1'-[(5-methylthiophen-2-yl)methyl]-5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
methyl({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)[1-(1,3-thiazol-2-yl)ethyl]amine
methyl 2-(2-{1-[(4-chloro-3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methylacetamido)acetate
3-(3-fluorophenyl)-4-(3-phenyl-1H-pyrazole-4-carbonyl)piperazin-2-one
N-(3,4-dimethylphenyl)-1-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}piperidin-3-amine
3-[2-(3-fluorophenyl)acetyl]-9-methoxy-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
6-[(3S,4R)-3,4-dihydroxy-4-methylpiperidin-1-yl]pyrazine-2-carboxamide
1-{2-[3-(3-methylthiophene-2-carbonyl)piperidin-1-yl]-2-oxoethyl}azepan-2-one
(1S,5R)-6-methyl-3-(naphthalene-2-sulfonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-methyl-5-{4-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]phenyl}-2H-1,2,3,4-tetrazole
(1S,5R)-N6-(3-chloro-2-methylphenyl)-N3,N3-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3,6-dicarboxamide
9-(butane-1-sulfonyl)-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N4-[3-(pyridin-2-yl)propyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-N-[1-(pyridin-4-yl)propan-2-yl]acetamide
4-{[(4aR,8aS)-6-cyclopropanecarbonyl-decahydro-1,6-naphthyridin-1-yl]methyl}-N-methyl-N-phenylaniline
1-[4-(3-methylpyridin-2-yl)piperazin-1-yl]-2-(2,4,7-trimethyl-1H-indol-3-yl)ethan-1-one
2-[3-(cyclopropylmethyl)-5-{[3-(trifluoromethyl)phenyl]methyl}-1H-1,2,4-triazol-1-yl]ethan-1-ol
ethyl 1-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidine-4-carboxylate
(1R,9S)-5-amino-13-methyl-3-(thiophen-3-yl)-6,13-diazatricyclo[7.3.1.02,7]trideca-2,4,6-triene-4-carbonitrile
N-[(2R,3R)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-6-methylpyridine-3-carboxamide
3-({[(1-ethyl-5-oxopyrrolidin-3-yl)methyl](methyl)amino}methyl)-7-(methylsulfanyl)-1,2-dihydroquinolin-2-one
{[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[1-(1,3-thiazol-2-yl)ethyl]amine
(1S,6R)-3-{3-[4-(3-chlorophenyl)piperazin-1-yl]propyl}-3,9-diazabicyclo[4.2.1]nonan-4-one
N-methyl-2-(2-oxo-1,3-oxazolidin-3-yl)-N-{2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}acetamide
2-{5-[(propan-2-ylsulfanyl)methyl]-3-(thiophen-2-ylmethyl)-1H-1,2,4-triazol-1-yl}ethan-1-ol
N-[(3-fluorophenyl)methyl]-3-(piperidine-1-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine