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2-[(3,5-difluorophenyl)methyl]-N-ethyl-3-oxo-2,8-diazaspiro[4.5]decane-8-carboxamide
{[1-benzyl-2-(2-methylpropanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amine
2-{[ethyl(pyridin-4-ylmethyl)amino]methyl}-4-phenylphenol
1-[3-(methylsulfanyl)propyl]-N-[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
1-{4-[(3-acetylphenyl)methyl]-1,8-dioxa-4,11-diazaspiro[5.6]dodecan-11-yl}-2-methoxyethan-1-one
3-[(2-{1-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]piperidin-4-yl}-1H-imidazol-1-yl)methyl]pyridine
N-(2-ethyl-3-methyl-1-benzofuran-7-yl)-4-(1,3-thiazol-2-yl)piperazine-1-carboxamide
2-(2-{1-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperidin-3-yl}-1H-imidazol-1-yl)acetamide
1-{2-[2-(2,1,3-benzoxadiazol-4-yl)-1H-imidazol-1-yl]ethyl}imidazolidin-2-one
N-[(3S)-1-[7-acetyl-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]pyrrolidin-3-yl]acetamide
1-(carbamoylmethyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-propylpiperidine-4-carboxamide
(2S,4R)-1-(naphthalen-2-ylmethyl)-N-(propan-2-yl)-4-({[2-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
(2R,3R,6R)-3-(4-fluorophenyl)-5-(5-methylpyrazine-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
6-{6-[(pyridin-3-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridin-3-amine
N-[(2-fluorophenyl)methyl]-2-[3-(hydroxymethyl)-3-(prop-2-en-1-yl)piperidin-1-yl]acetamide
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carboxamide
3-[1-(but-3-enoyl)piperidin-3-yl]-N-[(2-fluorophenyl)methyl]propanamide
methyl (2S,4R)-4-(5-chloro-3-phenyl-1H-indole-2-amido)-1-[(4-fluorophenyl)methyl]pyrrolidine-2-carboxylate
1-[cyclopropyl(1-methyl-1H-imidazol-2-yl)methyl]-4-[3-(1H-pyrazol-1-yl)phenyl]-1H-1,2,3-triazole
(1S,3R)-N1-[(2-chloro-6-fluorophenyl)methyl]-1,N2,N2,3,3-pentamethylcyclopentane-1,3-dicarboxamide
1-[(1R,2R)-2-hydroxycyclohexyl]-3-(2-methoxy-6-methylphenyl)-1-propylurea
1-{3-[({1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}amino)methyl]phenyl}ethan-1-one
N-({2,4-dimethyl-5-[(4-methylpiperazin-1-yl)methyl]phenyl}methyl)-1-(methoxymethyl)-N-methylcyclopropan-1-amine
2-[2-(azepan-1-ylmethyl)-4-(pyrimidin-2-yl)phenoxy]-N-[(4-fluorophenyl)methyl]acetamide
ethyl 1-{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}-4-(oxan-2-ylmethyl)piperidine-4-carboxylate
N-{[7-(5-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-4-(thiophen-2-yl)butanamide
N,7-dimethyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}pyrazolo[1,5-a]pyrimidine-6-carboxamide
4-ethoxy-N-{[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methyl}pyrimidin-2-amine
1'-{[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl}spiro[indene-1,4'-piperidine]
4-[1-(2,2-diphenylethyl)piperidin-3-yl]morpholine
2,3-dimethyl-N-(1,2-oxazol-3-ylmethyl)-1H-indole-7-carboxamide
4-[2-ethoxy-5-(trifluoromethyl)phenyl]-4H-1,2,4-triazole
7-methyl-2-{[1-(propan-2-yl)-1H-1,3-benzodiazol-2-yl]methyl}-2,7-diazaspiro[4.5]decan-6-one
N-{[5-methyl-7-(pyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}cyclopropanecarboxamide
4-{3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl}-6-methylpyrimidin-2-amine
N-[(3R,4S)-1-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]-4-propylpyrrolidin-3-yl]-2-hydroxyacetamide
N-ethyl-N-(2-methylprop-2-en-1-yl)-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
2-(2H-1,3-benzodioxol-5-yl)-1-[4-(4H-1,2,4-triazol-4-yl)piperidin-1-yl]ethan-1-one
N-{[4-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-4-(1H-pyrazol-3-yl)benzamide
4-(4-fluoropiperidine-1-carbonyl)-1-(pyridin-4-ylmethyl)pyrrolidin-2-one
9-{4-[(2-hydroxyethyl)sulfanyl]benzoyl}-1-oxa-9-azaspiro[5.5]undecan-5-ol
(4S)-4-(methoxymethyl)-1-[1-(4-methoxyphenyl)piperidin-4-yl]-3,3-dimethylpiperidin-4-ol
5-(1-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-4-phenyl-1H-imidazol-5-yl)pyrimidin-2-amine
4-{2-oxo-2-[2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepan-4-yl]ethyl}-3,4-dihydro-2H-1,4-benzoxazin-3-one
[(4-methanesulfonylphenyl)methyl](methyl)[(3-phenyl-1,2-oxazol-5-yl)methyl]amine
4-(2H-1,3-benzodioxole-5-carbonyl)-5-methyl-1-(4-methylphenyl)piperazin-2-one
2-(2,3-dihydro-1H-inden-1-yl)-N-[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]acetamide
4-[4-(2-chlorophenyl)piperidin-4-yl]-N-ethylpyrimidin-2-amine
(1R,7S)-N-methyl-N-(1,2-oxazol-5-ylmethyl)-4-oxo-3-[4-(propan-2-yl)phenyl]-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-N-methyl-N-[2-(pyridin-2-yl)ethyl]piperidin-3-amine