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2-(2,3-dihydro-1H-inden-5-yloxy)-2-methyl-1-[4-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]propan-1-one
1-(2-cyclopropylphenyl)-3-[2-(propane-2-sulfonyl)ethyl]urea
N-cyclohexyl-4-[({[(2-fluorophenyl)methyl]carbamoyl}methyl)amino]piperidine-1-carboxamide
[(2-cyclohexylpyrimidin-5-yl)methyl](methyl)[3-(oxolan-2-yl)propyl]amine
5-(3-ethyl-1,2,4-oxadiazol-5-yl)-1-[2-(4-methoxyphenyl)ethyl]piperidin-2-one
5-(2-ethyl-1,2,3,4-tetrahydroisoquinoline-3-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonitrile
3-(2-{2-azabicyclo[2.2.1]heptan-2-yl}-2-oxoethyl)-1-cyclopropyl-3-[3-(trifluoromethyl)phenyl]pyrrolidine-2,5-dione
9-(3-ethyl-1H-pyrazole-5-carbonyl)-2-[3-(1H-imidazol-1-yl)propyl]-2,9-diazaspiro[5.5]undecan-3-one
4-{dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}-2-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]morpholine
1-methyl-3-[4-(4-methyl-4H-1,2,4-triazol-3-yl)phenyl]-1-[1-(4-methylpyridin-2-yl)propan-2-yl]urea
(3S,4S)-4-propyl-1-[3-(pyrazin-2-yl)propanoyl]pyrrolidine-3-carboxylic acid
3-[2-(dimethylamino)ethyl]-8-[2-methyl-5-(propan-2-yl)furan-3-carbonyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-chloro-N-(2-{imidazo[1,2-a]pyrimidin-2-ylformamido}ethyl)benzamide
1-{1-[3-(4-methylphenoxy)azetidine-1-carbonyl]cyclohexyl}pyrrolidine
N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2-methyl-1,3-thiazole-4-carboxamide
N-ethyl-2-{4-[3-(pyridin-3-yl)-1H-pyrazol-1-yl]phenyl}acetamide
1-[4-(2H-1,3-benzodioxol-5-yl)pyrimidin-2-yl]-5-cyclopropyl-N-[2-(pyridin-2-yl)ethyl]-1H-pyrazole-4-carboxamide
N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetamide
2-(5-{[4-(thiophene-2-carbonyl)piperazin-1-yl]methyl}-1,2,4-oxadiazol-3-yl)pyrazine
N-[(4,6-dimethylpyridin-3-yl)methyl]-3-(3-hydroxy-3-methylbutyl)benzamide
3-[5-(1H-imidazol-2-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]-1-(pyrrolidin-1-yl)propan-1-one
4-(1-{[3-(6-methoxynaphthalen-2-yl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)pyridine
(3R,9aR)-8-(2,5-dimethylbenzenesulfonyl)-3-(2-methylpropyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
5-(1-ethyl-5-methyl-1H-pyrazol-4-yl)-1-(2-methylpropyl)-4-phenyl-1H-imidazole
3,5,7-trimethyl-2-{4-[(2-methyl-1H-imidazol-1-yl)methyl]piperidine-1-carbonyl}-1H-indole
{[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)methylamine
4-(3-hydroxy-3-methylbutyl)-N-[(4-methoxyphenyl)methyl]-N-methylbenzamide
5-[(9aS)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepine-2-carbonyl]-4-chloro-1-ethyl-1H-pyrazole
3-({4-[3-(1H-pyrazol-1-yl)benzoyl]piperazin-1-yl}methyl)benzonitrile
2-(4-{[3-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}-1-(3-methylbut-2-en-1-yl)piperazin-2-yl)ethan-1-ol
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-N-methyl-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetamide
3-[(2R,3R,6R)-5-[(4-methylphenyl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
11-(cyclohexylamino)-4-{[3-(trifluoromethyl)phenyl]methyl}-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
N-[(2-ethoxypyridin-3-yl)methyl]-6-methyl-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
N-[(3S,4R)-1-[(3-cyanophenyl)methyl]-4-(4-methylphenyl)pyrrolidin-3-yl]acetamide
2-{4-[2-chloro-5-(trifluoromethoxy)phenyl]-1H-pyrazol-1-yl}ethan-1-ol
N-(oxan-4-yl)-2-(3-phenylpropyl)-1,3-benzoxazole-5-carboxamide
4-(2-hydroxyethyl)-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-(1-cyclopropylethyl)-9-methoxy-7-(quinolin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-(naphthalen-2-yloxy)-1-[4-(thian-4-yl)piperazin-1-yl]propan-1-one
(3R,5S)-5-[4-(4-chlorophenoxy)piperidine-1-carbonyl]pyrrolidin-3-ol
(2S)-1-(6-fluoro-2-methylquinoline-4-carbonyl)pyrrolidine-2-carboxamide
1-{5-[2-(3-methoxyphenyl)piperidine-1-carbonyl]-2-methylphenyl}imidazolidin-2-one
3-[(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1H-indazole
1-(3-{[4-(methoxymethyl)piperidin-1-yl]methyl}phenoxy)-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
N-cyclopropyl-3-({3-methyl-2-oxo-1-oxa-3,7-diazaspiro[4.4]nonan-7-yl}sulfonyl)benzamide
4-{5-[3-(3-methoxyphenyl)-1H-pyrazol-5-yl]-3-methyl-1H-1,2,4-triazol-1-yl}-1-methylpiperidine
4-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-methyl-5-propylpyrimidine
(4aR,7aS)-N,N-dimethyl-6,6-dioxo-4-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
N-(2-hydroxyethyl)-5-(1H-indole-2-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide