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1-cyclopentyl-N-[2-(4-methyl-1H-pyrazol-1-yl)ethyl]-5-oxopyrrolidine-3-carboxamide
4-[(4-fluoro-3-methylphenyl)methyl]-1-(2-methylphenyl)piperazin-2-one
N-(1H-1,3-benzodiazol-2-ylmethyl)-5-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
1-[1-(2H-1,3-benzodioxole-5-carbonyl)piperidin-4-yl]-5-fluoro-2-[(2-methoxyphenyl)methyl]-1H-1,3-benzodiazole
5-[4-(1H-imidazol-1-yl)phenyl]-3-methyl-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazole
methyl 3-[(3S,4R)-1-[(2-hydroxyphenyl)methyl]-4-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-3-yl]propanoate
N-methyl-1-(oxolan-2-ylmethyl)-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
N-ethyl-3-methyl-N-[(2E)-3-phenylprop-2-en-1-yl]pyridine-2-carboxamide
2-chloro-N-({1-[4-(2-oxopyrrolidin-1-yl)butanoyl]piperidin-3-yl}methyl)benzamide
2-{1H-pyrrolo[2,3-b]pyridin-4-yl}benzamide
N-(3-methylpentyl)-1-[4-(1H-pyrazol-1-yl)phenyl]piperidin-4-amine
N-[2-(dimethylamino)ethyl]-N-(thiophen-3-ylmethyl)furan-2-carboxamide
2-(naphthalen-1-yl)-N-{2-[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}acetamide
ethyl 3-[5-(1-methyl-1H-1,3-benzodiazol-2-yl)-4-phenyl-1H-imidazol-1-yl]propanoate
2-methyl-4-{3-[3-(pyrrolidin-1-yl)pyrrolidine-1-carbonyl]phenyl}butan-2-ol
4-benzyl-3-{1-[2-(1H-pyrrol-1-yl)acetyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
5-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2-methyl-1,3-benzoxazole
3-({[(1-benzyl-1H-pyrazol-4-yl)methyl]amino}methyl)pyrrolidin-3-ol
2-(1H-1,3-benzodiazol-1-yl)-N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]acetamide
1-(cyclopropanesulfonyl)-4-[(2,6-dimethylpyridin-3-yl)oxy]piperidine-4-carboxylic acid
2-{2-[(3-methoxyphenyl)methyl]morpholin-4-yl}-N-(5-methyl-1,2-oxazol-3-yl)acetamide
N-{2-[({3-methyl-1-[2-(thiomorpholin-4-yl)ethyl]-1H-pyrazol-4-yl}methyl)amino]ethyl}acetamide
2-{[(6-hydroxypyrimidin-4-yl)methyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
N-[(3S,4S)-4-methoxy-1-(propan-2-yl)pyrrolidin-3-yl]-5,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
4-{[2-(3-methoxyphenyl)pyrrolidin-1-yl]methyl}-5-methyl-2-(5-methylthiophen-2-yl)-1,3-oxazole
9-[(2,3-difluorophenyl)methyl]-2-[2-(dimethylamino)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
7-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-4-(furan-2-carbonyl)-9-(oxolan-2-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-(4-ethylpiperazin-1-yl)-3-(2-methoxy-4-{[methyl(pyridin-3-ylmethyl)amino]methyl}phenoxy)propan-2-ol
1-[1-(2-methoxyacetyl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
N-(2-methoxyethyl)-3-({1-[(2R)-pyrrolidine-2-carbonyl]piperidin-4-yl}oxy)benzamide
N-{[4-(2-phenylethyl)-4H-1,2,4-triazol-3-yl]methyl}-2,8-diazaspiro[4.5]decane-3-carboxamide
8-{3-azaspiro[5.5]undecan-9-yl}-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
N-(2-{[1-(ethylsulfanyl)propan-2-yl]amino}ethyl)-2,2,2-trifluoroacetamide
N-({3-[4-(1H-pyrazol-1-yl)phenyl]phenyl}methyl)acetamide
N-[3-methoxy-4-(3-methylbutanamido)phenyl]-1H-imidazole-2-carboxamide
1-{2-[2-(3-ethoxy-4-hydroxyphenyl)-1H-imidazol-1-yl]ethyl}imidazolidin-2-one
2-[3-(2-fluorophenoxy)azetidine-1-carbonyl]pyridin-3-ol
N-[(4-chlorophenyl)(phenyl)methyl]-3-(2-ethyl-5-oxopyrrolidin-2-yl)propanamide
4-[(2-methoxyphenyl)methyl]-N-(1-methyl-1H-indazol-6-yl)piperazine-1-carboxamide
N-cyclopropyl-3-(3-hydroxy-3-methylbutyl)-N-(1,3-thiazol-2-ylmethyl)benzamide
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-2H-1,3-benzodioxole-5-carboxamide
dimethyl(3-{2-[1-(2-methylbenzoyl)piperidin-4-yl]-1H-imidazol-1-yl}propyl)amine
2-methyl-N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-1,3-benzoxazole-6-carboxamide
2-({6-[(dimethylamino)methyl]-1,4-oxazepan-4-yl}methyl)-4-methoxyphenol
(4aR,6R,8aS)-2-(1,3-benzothiazol-2-yl)-8a-(methoxymethyl)-6-(morpholin-4-yl)-decahydroisoquinoline
(3aS,6aS)-2-methyl-5-(1,3-thiazol-4-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-{2-[2-(3-methoxyphenyl)ethyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}-N,N-bis(prop-2-en-1-yl)piperidine-3-carboxamide
N-[1-(thiophen-3-yl)propan-2-yl]thieno[2,3-d]pyrimidin-4-amine
4-hydroxy-2-phenyl-N-[2-(4H-1,2,4-triazol-4-yl)ethyl]pyrimidine-5-carboxamide
N-(furan-2-ylmethyl)-5-methyl-6-[4-(propan-2-yl)piperazine-1-carbonyl]thieno[2,3-d]pyrimidin-4-amine