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4-[(4-methylphenyl)sulfanyl]-1-{[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carbonyl}piperidine
5-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-1-(2-phenylethyl)-N-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-[(1-ethyl-1H-imidazol-2-yl)methyl]-1-methyl-3-[1-(1-phenylethyl)-1H-pyrazol-5-yl]urea
3-[N-benzyl-1-(3-ethyl-1H-pyrazol-4-yl)formamido]propanamide
3-{[(cyclopropylmethyl)amino]methyl}-3-hydroxy-1-[(3-methylphenyl)methyl]piperidin-2-one
2-methyl-N-(1-{7-[(2,4,6-trimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)propanamide
1-{2-[1-(2-acetylbenzoyl)piperidin-4-yl]ethyl}pyrrolidin-2-one
1-{1-[(4-fluorophenyl)methyl]piperidin-4-yl}-3-(pyrrolidine-1-carbonyl)piperidine
4-methoxy-3-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}benzamide
N-ethyl-4,6-dimethyl-N-(oxan-4-ylmethyl)-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
6-phenyl-3-{1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}imidazo[2,1-b][1,3]thiazole
3-(hydroxymethyl)-1-[1-methyl-3-(trimethyl-1H-pyrazol-4-yl)-1H-pyrazole-5-carbonyl]piperidin-3-ol
ethyl 4-{1-[(2E)-2-methylbut-2-en-1-yl]piperidin-3-yl}piperazine-1-carboxylate
N-[4-({methyl[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-3-yl)methyl]amino}methyl)phenyl]acetamide
1-(3-{3-cyclobutyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}phenyl)-5-methyl-1H-1,2,3,4-tetrazole
N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-2-(phenylamino)pyrimidine-5-carboxamide
5-(3-methoxyphenyl)-N-methyl-N-(pyrimidin-4-ylmethyl)-1,2,4-triazin-3-amine
1-(1H-1,3-benzodiazol-2-ylmethyl)-N-[3-(1H-pyrazol-1-yl)phenyl]piperidine-3-carboxamide
1-[2-(3-methyl-1H-pyrazol-1-yl)ethyl]-4-(2-methylphenoxy)piperidine
(3R,4R)-4-(hydroxymethyl)-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidin-3-ol
methyl 3-{[1-(3,4-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]carbamoyl}propanoate
N-[(1R,3S)-3-{[3-(4H-1,2,4-triazol-4-yl)propyl]carbamoyl}cyclopentyl]morpholine-4-carboxamide
2-(6-methoxy-3-methyl-1-benzofuran-2-carbonyl)-2-azaspiro[4.4]nonane
4-(4-chlorophenoxy)-N-[1-(pyrazin-2-yl)propan-2-yl]piperidine-4-carboxamide
(1S,5R)-3-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-methyl-4-[3-(2-phenylazetidine-1-carbonyl)phenyl]butan-2-ol
6-methyl-1-[3-(pyridin-3-yl)propyl]-4-(trifluoromethyl)-1,2-dihydropyridin-2-one
N-benzyl-3-[(3-hydroxypiperidin-1-yl)methyl]-N-methylimidazo[1,2-a]pyridine-2-carboxamide
1-[(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(pyridin-3-yl)ethan-1-one
5-methyl-1-{2-[4-(5-methyl-1,2,4-oxadiazol-3-yl)piperidin-1-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[2-(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]-2,3-dihydro-1,4-benzodioxine-6-carboxamide
4-(6-methoxyquinolin-3-yl)-N-(pyridin-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
3-(5-{3,9-diazaspiro[5.5]undecan-3-ylmethyl}thiophen-2-yl)prop-2-yn-1-ol
N-methyl-1-[(3-methylquinoxalin-2-yl)methyl]piperidine-2-carboxamide
6-{[3-(3-oxopiperazin-1-yl)propyl]amino}-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
5-(2-fluorophenyl)-N-[2-(piperazin-1-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}(2-methoxyethyl){[4-(1H-pyrazol-1-yl)phenyl]methyl}amine
5-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]-1-[(2-methoxyphenyl)methyl]piperidin-2-one
N-[(3S)-1-benzylpyrrolidin-3-yl]-3-(1H-imidazol-2-yl)-N-methylbenzamide
3-[3-(dimethylamino)propyl]-8-[(4-methoxyphenyl)methyl]-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-{[1-(3-phenylprop-2-yn-1-yl)piperidin-3-yl]methyl}thiophene-2-carboxamide
1-[4-(2H-1,3-benzodioxol-5-yl)pyrimidin-2-yl]-N-[(5-chlorothiophen-2-yl)methyl]-5-cyclopropyl-1H-pyrazole-4-carboxamide
9-methoxy-7-(6-methoxypyridin-2-yl)-4-(naphthalene-2-sulfonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-{[(4-fluorophenyl)methyl]amino}-N-methyl-N-[3-(oxolan-2-yl)propyl]benzamide
(4aR,8aR)-4-(8-fluoroquinoline-2-carbonyl)-octahydro-2H-1,4-benzoxazine
2-propyl-8-(4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
3-(1-benzofuran-2-yl)-4-({8-methoxy-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}methyl)-1H-pyrazole
2-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
ethyl 1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-3-[(2-methylphenyl)methyl]piperidine-3-carboxylate
3-{2-[2-hydroxy-3-(piperidin-1-yl)propoxy]phenyl}-N-methylbenzamide