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N-[(3-fluoro-4-methylphenyl)methyl]-4-{[1-(3-methoxypropanoyl)piperidin-4-yl]oxy}benzamide
N-{imidazo[1,2-a]pyridin-3-ylmethyl}-N,2,3,6-tetramethylquinoline-4-carboxamide
2-(1-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-2-carbonyl}pyrrolidin-2-yl)-6-methyl-1H-1,3-benzodiazole
4-[(5-fluoro-2-methylphenyl)methyl]-3-propylmorpholine
2-{[4-(2,3-dichlorophenyl)-1H-1,2,3-triazol-1-yl]methyl}-5-methylpyrazine
4-{4-[(dimethylamino)methyl]phenyl}-5-propylthiophene-2-carboxylic acid
1-(1-{5H,6H-benzo[h]quinazolin-2-yl}-5-methyl-1H-pyrazole-4-carbonyl)azepane
1-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-3-(1-propyl-1H-1,2,3-triazol-4-yl)urea
N-(2-{4-phenyl-5-[2-(1H-pyrazol-1-yl)ethyl]-1H-imidazol-1-yl}ethyl)acetamide
N3-cycloheptyl-1-cyclopropyl-N5-[1-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
1-{2-[3-(oxolan-3-yl)-1-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}pyrrolidin-2-one
N-(3,5-dimethoxyphenyl)-3-(methanesulfonylmethyl)piperidine-1-carboxamide
7-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}-2,7-diazaspiro[4.4]nonane-1,3-dione
N-[2-(methylamino)ethyl]-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-4-carboxamide
methyl 4-{[1-(cyclohexylmethyl)-5-oxopyrrolidin-3-yl]carbamoyl}butanoate
1-(3-fluorophenyl)-4-(5-methyl-4-phenyl-1H-imidazol-2-yl)pyrrolidin-2-one
N-[3-(morpholin-4-yl)propyl]-2-(trifluoromethyl)pyrimidin-4-amine
{[3-(2-fluorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}(methyl)[(3-methyl-1H-indol-2-yl)methyl]amine
N-{[4-methyl-2-(propan-2-yl)-1,3-thiazol-5-yl]methyl}-3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carboxamide
(4aS,7aR)-1-[(2,6-difluorophenyl)methyl]-4-(2-methylpropyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-(3-methylpiperidin-1-yl)-3-[2-(pyridin-4-ylsulfanyl)acetamido]benzamide
1-cyclohexyl-4-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one
1-[4-({methyl[3-(1-methyl-1H-imidazol-2-yl)propyl]amino}methyl)thiophen-2-yl]ethan-1-one
N-benzyl-2-(ethylamino)-N-(1,3-thiazol-2-ylmethyl)pyrimidine-5-carboxamide
1-[4-(2-fluorophenyl)pyrimidin-2-yl]-5-(methoxymethyl)-N-(pyridin-3-ylmethyl)-1H-pyrazole-4-carboxamide
(1S,5R)-3-methyl-6-[4-(4H-1,2,4-triazol-4-yl)benzoyl]-3,6-diazabicyclo[3.2.2]nonane
methyl 4-{[3-(2,3-dihydro-1H-inden-2-yl)-1-(2-methylpropyl)-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-8-yl]methyl}benzoate
1-{5-[5-(3-methoxyphenyl)-1,2,4-oxadiazol-3-yl]-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridin-2-yl}ethan-1-one
2-cyclopentyl-7-[(4-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
5-{4-[(2-methylphenyl)sulfanyl]piperidine-1-carbonyl}-2-(pyridin-4-yl)pyrimidin-4-ol
N-({1-[(1-ethyl-1H-pyrazol-4-yl)methyl]pyrrolidin-3-yl}methyl)-4-methylpyridine-3-carboxamide
N-(3-methylbutyl)-1-(2-methylpropyl)-5-[4-(6-methylpyridin-2-yl)piperazine-1-carbonyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
2-{4-[5-(4-fluorophenyl)-1,2,4-triazin-3-yl]piperazin-1-yl}ethan-1-ol
N-ethyl-2-[1-(propan-2-yl)-1H-pyrazol-4-yl]-N-(pyridin-3-ylmethyl)quinoline-4-carboxamide
4-(2-chloro-3-methylbenzoyl)-3-(2-hydroxyethyl)piperazin-2-one
1-{3-[2-(3,4-difluorophenyl)ethyl]piperidin-1-yl}-3-(pyrazin-2-yl)propan-1-one
methyl 5-{2,7-diazaspiro[4.5]decan-7-ylmethyl}-2-hydroxybenzoate
(3R,4S)-1-[(2-ethyl-1,3-thiazol-4-yl)methyl]-3,4-dimethylpiperidin-4-ol
N-(3-ethoxypropyl)-2-{3-oxo-1-[(3-phenoxyphenyl)methyl]piperazin-2-yl}acetamide
N-[4-methoxy-3-(methylcarbamoyl)phenyl]thiomorpholine-4-carboxamide
1-{3-[2-(2-methylphenyl)ethyl]piperidin-1-yl}ethan-1-one
N2,N2,N4-trimethyl-N4-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine
(3S,4R)-1-[(5-acetylthiophen-3-yl)methyl]-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
5-(4-fluorophenyl)-N-{[3-(trifluoromethoxy)phenyl]methyl}-1,2,4-triazin-3-amine
1-(5,6-dimethyl-1H-1,3-benzodiazol-7-yl)-5-oxopyrrolidine-3-carboxylic acid
N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-3-(4H-1,2,4-triazol-4-yl)benzamide
4-(1-{[5-(2-methylpropyl)thiophen-2-yl]methyl}azetidin-3-yl)morpholine
N-[2-(5-methylfuran-2-yl)-2-(morpholin-4-yl)ethyl]-1,3-benzothiazole-6-carboxamide
4-{2-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-oxoethyl}piperazin-2-one
N-(1-benzofuran-2-ylmethyl)-1-(2-fluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-amine