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2-[5-(3-chloro-2,6-difluorophenyl)-4-phenyl-1H-imidazol-1-yl]-2-methylpropane-1,3-diol
5-[4-(2-methylphenyl)-1,4-diazepane-1-carbonyl]pyrazin-2-ol
3-({2-[1-(4-methyl-1H-imidazole-2-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
3-[(3R,4S)-1-(4-methylphthalazin-1-yl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
1-({4-[3-(azepan-1-yl)-2-hydroxypropoxy]-3-methoxyphenyl}methyl)piperidin-4-ol
1-{3-[(4-fluorophenyl)amino]piperidin-1-yl}-3-(2-methyl-1H-1,3-benzodiazol-1-yl)propan-1-one
4-phenoxy-1-[3-(1H-pyrazol-1-yl)butanoyl]piperidine-4-carboxylic acid
N-{[4-(3-fluorophenyl)oxan-4-yl]methyl}-4-(pyridin-4-yl)pyrimidin-2-amine
4-{[3-(2,4-dimethoxyphenyl)-1H-pyrazol-4-yl]methyl}thiomorpholine
5-[4-(3-benzyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-1-methyl-1H-pyrrol-3-amine
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-1-[(3,4-dimethoxyphenyl)methyl]-N5-[(4-fluorophenyl)methyl]piperidine-3,5-dicarboxamide
3-(2H-1,3-benzodioxol-5-yl)-5-[1-(methylsulfanyl)propan-2-yl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
3-[2-fluoro-5-(4H-1,2,4-triazol-4-yl)phenyl]-1-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}urea
1'-(2H-1,3-benzodioxol-5-ylmethyl)-5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-(1-{1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-2-phenylethyl)-N,1,3-trimethyl-1H-pyrazole-5-carboxamide
methyl({[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}){[2-(pyrrolidin-1-yl)pyrimidin-5-yl]methyl}amine
N-(3-fluorophenyl)-3-{2-[1-(propan-2-yl)-1H-imidazol-2-yl]-1H-imidazol-1-yl}propanamide
3-(4,5,6,7-tetrahydro-2H-indazol-3-yl)-N-{1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl}propanamide
3-{[1-(3-methylpyridin-4-yl)-3-phenyl-1H-1,2,4-triazol-5-yl]methyl}phenol
1-[(4-fluorophenyl)methyl]-5-{thieno[3,2-d]pyrimidin-4-yl}-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazole
2-{5-[2-(1H-imidazol-2-yl)phenyl]-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-1-yl}ethan-1-ol
N-(2H-1,3-benzodioxol-5-ylmethyl)-1-cyclopentyl-4-oxo-5-(piperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
N,4-dimethyl-5-{4-[(3-methylphenyl)sulfanyl]piperidine-1-carbonyl}-1,3-thiazol-2-amine
4-{[3-(naphthalene-2-carbonyl)piperidin-1-yl]methyl}-1H-pyrazole-3-carboxylic acid
[(3-chloro-4-methoxyphenyl)methyl](methyl)[2-(oxan-2-yl)ethyl]amine
N-(2-hydroxyethyl)-N-[(2-methoxyphenyl)methyl]-2-[(prop-2-en-1-yl)amino]benzamide
4-{4-[(2-methylphenyl)sulfanyl]piperidine-1-carbonyl}pyridine
5-[3-(4-methoxyphenyl)-1H-pyrazol-5-yl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
2-amino-N-{2-[(4-chlorophenyl)sulfanyl]ethyl}-3-ethyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
(2S,4R)-N-[2-(2-fluorophenyl)ethyl]-4-{[(4-phenylphenyl)methyl]amino}-1-(propan-2-yl)pyrrolidine-2-carboxamide
7-chloro-2-methyl-4-(thiophen-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-{4-[(4-fluoro-3-methoxyphenyl)methyl]-1-[(5-methylfuran-2-yl)methyl]piperazin-2-yl}ethan-1-ol
3-cyclopropyl-N-[2-(2-oxopiperidin-1-yl)ethyl]-1H-pyrazole-5-carboxamide
1-cyclopropyl-3-[2-(4-methoxypiperidin-1-yl)-2-oxoethyl]-3-[3-(trifluoromethyl)phenyl]pyrrolidine-2,5-dione
(2R,6R)-4-(oxan-4-yl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
N-methyl-3-{methyl[(2E)-2-methyl-3-phenylprop-2-en-1-yl]amino}butanamide
1-phenyl-N-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}-1H-1,2,3-triazole-5-carboxamide
ethyl(methyl)[({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)sulfamoyl]amine
2-cyclobutyl-N-[(3R,4S)-4-cyclopropyl-1-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]pyrrolidin-3-yl]acetamide
(2S)-2-amino-3-hydroxy-1-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
5-(1-methoxypropan-2-yl)-3-[4-(trifluoromethyl)phenyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
4-({4-methyl-5-[1-(1H-pyrrole-3-carbonyl)piperidin-3-yl]-4H-1,2,4-triazol-3-yl}methyl)morpholine
(3R,4R)-3-cyclopropyl-1-[6-(methoxymethyl)pyrimidin-4-yl]-4-methylpyrrolidin-3-ol
1-{1-oxa-8-azaspiro[4.5]decan-8-yl}-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propan-1-one
N-{2-[4-(4-fluorophenyl)-5-{[(2-methylphenyl)methyl]sulfanyl}-4H-1,2,4-triazol-3-yl]ethyl}-2,3-dimethoxybenzamide
4-(1-ethyl-1H-imidazol-5-yl)-3-methyl-1-(4-methylphenyl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
5-(3-methylbut-2-en-1-yl)-1'-(2-methylpyrimidine-5-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
(3aS,6aS)-5-(1-ethylpiperidin-4-yl)-1-oxo-2-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-(2,3-dihydro-1H-inden-1-yl)-N-[2-(pyridin-2-ylsulfanyl)ethyl]acetamide
4-[(2S,4R)-1-[(4-methoxynaphthalen-1-yl)methyl]-4-[(1-methyl-1H-imidazol-2-yl)sulfanyl]pyrrolidine-2-carbonyl]morpholine