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5-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazole-5-carbonyl}-3-(propan-2-yl)-1H-pyrazole
(4aS,7aR)-1-[2-(2-methylphenyl)acetyl]-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-{[1-(pyridin-2-ylmethyl)piperidin-3-yl]methyl}-1H-1,3-benzodiazole-2-carboxamide
1-[cyclohexyl(methyl)amino]-3-(4-{[4-(2-hydroxyethyl)piperidin-1-yl]methyl}-2-methoxyphenoxy)propan-2-ol
6-[2-(furan-2-yl)azepane-1-carbonyl]-1,3-benzothiazole
2-[4-(2-oxoimidazolidin-1-yl)phenyl]-N-{2-[2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethyl}acetamide
N-cyclopentyl-2-(methylamino)-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)acetamide
6-(4-methanesulfonylphenyl)pyridin-2-ol
3-(prop-2-en-1-yl)-1-[3-(trimethyl-1H-pyrazol-4-yl)propanoyl]piperidine-3-carboxylic acid
4-(3-methylbutyl)-3-{2-oxo-2-[4-(pyrimidin-2-yl)-1,4-diazepan-1-yl]ethyl}piperazin-2-one
2-butyl-N-[(5-methylpyrazin-2-yl)methyl]-1,3-benzoxazole-5-carboxamide
1-(3-{[(propan-2-yl)amino]methyl}phenoxy)-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
5-{4-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]piperazin-1-yl}-2-methyl-2,3-dihydropyridazin-3-one
2-[3-(2-ethylphenoxy)azetidine-1-carbonyl]-1-methylazepane
N,N-dimethyl-2-({2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]acetamido}methyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)-N-[2-(4-methylmorpholin-2-yl)ethyl]acetamide
N-(2-methoxy-5-methylphenyl)-2-[2-(4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]acetamide
N-{[3-(benzyloxy)phenyl]methyl}-2-(morpholin-2-yl)acetamide
[(3R,4R)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-(pyridine-2-carbonyl)pyrrolidin-3-yl]methanol
N-[3-({[3-(2-methoxyphenoxy)propyl](methyl)carbamoyl}amino)phenyl]-N-methylacetamide
6-methoxy-4-[2-(4-methylphenoxy)acetyl]-1-(pyridin-3-ylmethyl)-1,4-diazepan-2-one
4-[(2,6-difluorophenyl)methyl]-7-(2-methylphenyl)-9-(oxolan-3-yloxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-{1-[5-(4-methyl-1H-imidazol-5-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}phenol
N-({7-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-2,5-dimethylfuran-3-carboxamide
3-(2,5-dioxoimidazolidin-4-yl)-N-[2-(4-phenylpyrimidin-2-yl)ethyl]propanamide
4-[2-(butylsulfanyl)pyrimidin-5-yl]-3-methyl-4H,5H,6H,7H-[1,2]thiazolo[5,4-b]pyridin-6-one
N-(1-{4-[4-(3-chlorophenyl)piperazine-1-carbonyl]phenyl}-1H-pyrazol-4-yl)-2-methoxyacetamide
3-(2-butyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-(3-hydroxy-2,2-dimethylpropyl)propanamide
N-(3-hydroxypropyl)-2-(morpholin-4-yl)-6-{8-thiatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-yl}pyridine-3-carboxamide
4-methyl-2-{4-oxo-3H,4H-pyrido[2,3-d]pyrimidin-3-yl}pentanamide
methyl 1-{3-[3-(azetidin-1-ylmethyl)phenoxy]-2-hydroxypropyl}piperidine-4-carboxylate
3-phenyl-4-{1-phenyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-1H-pyrazole
1-{4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-3-(1,2-oxazinan-2-yl)propan-1-one
N-{1-[7-(9H-fluoren-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]-2-methylpropyl}propanamide
(4R)-4-{7-[(4-phenylpiperazin-1-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl}-1,3-thiazolidin-2-one
2-(2-chlorophenyl)-N-{[2-(4-methyl-1,4-diazepan-1-yl)pyridin-3-yl]methyl}acetamide
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-5-methyl-1H-indazole-3-carboxamide
4-{1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-1-(2-methoxyphenyl)-2,2-dimethylpiperazine
(1S,5R)-N-benzyl-7-oxo-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
(3S,4S)-1-{[2-(3,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine-3,4-diol
1-{[3-(2,4-dimethoxyphenyl)-1H-pyrazol-4-yl]methyl}-4-(2-fluorophenoxy)piperidine
1-[(2-fluorophenyl)methyl]-N-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperidin-3-amine
2-[3-(2-ethyl-1H-imidazol-1-yl)propanamido]-N-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
1-(4-{5-[(4-acetylpiperazin-1-yl)methyl]-2-methoxyphenoxy}piperidin-1-yl)-2-(thiophen-3-yl)ethan-1-one
N-cyclopropyl-1-[(3-methoxyphenyl)methyl]-5-[(4-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-(cyclopentylmethyl)-4-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-ylmethyl}-1H-imidazole
1-(2-methylpropyl)-2-{[3-(morpholin-4-yl)azetidin-1-yl]methyl}-1H-1,3-benzodiazole
N-cyclopropyl-3-{[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]sulfamoyl}benzamide
2-{4-[4-methyl-6-(methylamino)pyrimidin-2-yl]-1-[(4-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
1-(cyclohexylmethyl)-N-methyl-6-oxo-N-[(3-propyl-1,2,4-oxadiazol-5-yl)methyl]piperidine-3-carboxamide