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4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-[2-(4-methyl-1,3-thiazol-2-yl)ethyl]benzamide
N-(2-{1-[2-(dimethylamino)ethyl]-5-oxopyrrolidin-2-yl}ethyl)-8-fluoro-4-oxo-1,4-dihydroquinoline-3-carboxamide
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-3-[(2-methylprop-2-en-1-yl)oxy]benzamide
N-[2-(dimethylamino)ethyl]-1-(1-{[4-(2-methylphenyl)phenyl]methyl}piperidin-4-yl)-1H-1,2,3-triazole-4-carboxamide
5-[5-(oxan-2-yl)furan-2-yl]-4-phenyl-1H-imidazole
4-{4-[(4-tert-butyl-1H-1,2,3-triazol-1-yl)methyl]piperidin-1-yl}-2,5-dimethylpyrimidine
N-methyl-2-(morpholine-4-carbonyl)-N-phenyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
(3S,4R)-1-(1-tert-butyl-1H-pyrrole-3-carbonyl)-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
9-(3-methoxypropanoyl)-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-[4-(2,5-difluorophenyl)-1H-pyrazol-5-yl]-1-(3-methylbut-2-en-1-yl)piperidine
3-(3-cyclopropyl-1H-1,2,4-triazol-5-yl)-2-methyl-1,8-naphthyridine
8-{2-[(3-amino-1H-1,2,4-triazol-5-yl)sulfanyl]acetyl}-2-butyl-2,8-diazaspiro[5.5]undecan-3-one
4-[3-(1-benzyl-1H-imidazol-2-yl)piperidin-1-yl]-3-methylpyridine
2-{4-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperazin-1-yl}-1,3-benzothiazole
(2R,6R)-10-methoxy-4-[(6-methylpyridin-2-yl)methyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
4-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]-8-thia-4,6-diazatricyclo[7.5.0.02,7]tetradeca-1(9),2(7),5-trien-3-one
2-(2,4-difluorophenyl)-2-[4-(morpholin-4-yl)piperidin-1-yl]acetic acid
2-methanesulfonyl-1-(3-methoxypropyl)-5-{[1-(propan-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1H-imidazole
N-{2-[4-(hydroxymethyl)piperidin-1-yl]-5,6,7,8-tetrahydroquinazolin-5-yl}pyridine-2-carboxamide
3-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-1-[3-(piperidin-1-ylmethyl)phenyl]urea
3-[1-(1-benzylpiperidin-4-yl)-1H-pyrazol-5-yl]-1-(2-methoxyphenyl)urea
N-(6-fluoropyridin-3-yl)-4-(pyridin-3-ylmethoxy)piperidine-1-carboxamide
3-[2-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]pyridine
2-{[(benzylcarbamoyl)amino]methyl}-N,N-dimethyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
3-(1H-1,3-benzodiazol-1-yl)-5-(morpholine-4-sulfonyl)benzoic acid
2-(3-fluorophenyl)-N-(4-{4-[methyl(1,2-oxazol-3-ylmethyl)amino]piperidin-1-yl}phenyl)acetamide
(1R,5S,6S)-3-cyclopentyl-N-methyl-N-[2-(1H-pyrazol-4-yl)ethyl]-3-azabicyclo[3.1.0]hexane-6-carboxamide
2-(3-fluoropyridin-4-yl)-4-(trifluoromethyl)-5,6,7,8-tetrahydroquinazoline
5-[(5-cyclopropyl-1,2-oxazol-3-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
4-ethyl-3-{1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
9-[2-(4-ethylphenyl)acetyl]-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-amino-4-phenyl-N-[2-(propylsulfanyl)ethyl]pyrimidine-5-carboxamide
N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-1-(methoxymethyl)cyclobutane-1-carboxamide
N-{[2-(2-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}pyrrolidine-2-carboxamide
5-methoxy-N-methyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1H-indole-2-carboxamide
N-[(3S,5S)-5-(ethylcarbamoyl)-1-methylpyrrolidin-3-yl]-6-(3-fluorophenyl)pyridine-3-carboxamide
2-(4-{1-methyl-1H-pyrazolo[1,5-a]imidazole-7-carbonyl}piperazin-1-yl)pyridine-3-carbonitrile
N,N-dimethyl-3-(3-{5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-6-yl}phenyl)propanamide
2-(4-phenylpiperidin-1-yl)-N-[2-(pyridin-3-yl)ethyl]acetamide
N-[2-(dimethylamino)-2-(thiophen-2-yl)ethyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
N-[(2-phenyl-1,3-oxazol-4-yl)methyl]-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1-[(2R)-oxolane-2-carbonyl]piperidine
4-fluoro-N-{[1-(6-methylpyridine-2-carbonyl)piperidin-3-yl]methyl}benzamide
2-(4-fluorophenyl)-1-{1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperidine
(1R,2R)-2-[5-(1H-imidazol-1-ylmethyl)-3-[(phenylsulfanyl)methyl]-1H-1,2,4-triazol-1-yl]cyclohexan-1-ol
N-[(3R,4R)-1-[2-(2H-1,3-benzodioxol-5-yl)acetyl]-3-hydroxypiperidin-4-yl]pyrazine-2-carboxamide
N-{[5-(2-acetylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(pyridin-2-ylsulfanyl)acetamide
5-{3-[4-(naphthalen-2-yl)-1H-1,2,3-triazol-1-yl]propyl}-1,3,4-thiadiazol-2-amine
N,N-dimethyl-2-{[5-(4-phenylazepane-1-carbonyl)pyridin-2-yl]amino}acetamide
N-[3-fluoro-5-(trifluoromethyl)phenyl]-2-(morpholin-3-yl)acetamide