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3-[5-oxo-2-(thiophen-3-ylmethyl)pyrrolidin-2-yl]-N-[2-(1,2,3,4-tetrahydroquinolin-1-yl)ethyl]propanamide
6-methyl-4-{4-[1-(morpholin-4-yl)ethyl]piperidine-1-carbonyl}-1,2-dihydroquinolin-2-one
N-(2-hydroxypropyl)-2-[methyl(2-phenylethyl)amino]-2,3-dihydro-1H-indene-2-carboxamide
2-(5-fluoro-2-methoxyphenyl)-2-[4-(3-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]acetic acid
(2E)-N-[(3-methyl-7-{2-[(4S,6R)-6-methyl-2-sulfanylidene-1,3-diazinan-4-yl]acetyl}-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-3-(thiophen-2-yl)prop-2-enamide
(2-{2-[1-(3-methoxypyrazin-2-yl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)dimethylamine
6-methoxy-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
3,4-bis(2-methoxyphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
4-hydroxy-N-(3-hydroxy-3-phenylpropyl)-N-methyl-2-(3-methylphenyl)pyrimidine-5-carboxamide
4-{[2-(2,3-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1-[(3-methylphenyl)methyl]piperazin-2-one
2-({6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)-1-(2-methoxyphenyl)ethan-1-ol
2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazole-4-carboxylic acid
6-methoxy-4-[(4-phenylphenyl)methyl]-1-(pyridin-3-ylmethyl)-1,4-diazepan-2-one
8-(3-carbamoylpyridin-2-yl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-cyclopropyl-4-methoxy-2-{[1-(oxolan-3-ylmethyl)piperidin-4-yl]oxy}benzamide
N-{1-[1-(4-aminopyrimidin-2-yl)piperidin-4-yl]-1H-pyrazol-5-yl}-4-methoxybenzamide
3-(2-methylphenyl)-3-{2-oxo-2-[4-(propan-2-yl)piperazin-1-yl]ethyl}-1-(pyridin-3-ylmethyl)pyrrolidine-2,5-dione
2-[1-(cyclohexylmethyl)-3-oxopiperazin-2-yl]-N-methyl-N-(1,2-oxazol-3-ylmethyl)acetamide
N,N-dimethyl-3-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrazin-2-amine
2-methoxy-2-phenyl-N-{1-[1-(pyridine-3-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}acetamide
4-[1-(2-fluorophenyl)-1H-pyrazol-4-yl]-N-(thiolan-3-yl)pyrimidin-2-amine
2-{4-[6-amino-5-cyano-4-(4-hydroxyphenyl)pyridin-2-yl]-3,5-dimethyl-1H-pyrazol-1-yl}acetic acid
(5S,9aS,9bS)-2-(2,3-dihydro-1H-inden-2-yl)-5-[5-(hydroxymethyl)furan-2-yl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-{[4-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]methyl}-4-(5-methylpyridin-2-yl)piperidin-4-ol
N-[(3S,4R)-4-(4-methylphenyl)-1-(morpholine-4-sulfonyl)pyrrolidin-3-yl]acetamide
6-methoxy-3-methyl-N-(oxan-3-yl)-1-benzofuran-2-carboxamide
3-(2-{[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl](prop-2-en-1-yl)amino}ethyl)-2,3-dihydro-1,3-benzoxazol-2-one
6-{4-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperazin-1-yl}-9H-purine
2-[2-(2-methoxyethyl)piperidine-1-carbonyl]-N-(thiophen-2-ylmethyl)aniline
4-(1H-indol-2-ylmethyl)-9-methoxy-7-(quinolin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-3,4-dihydro-2H-1-benzopyran-3-amine
3-[(4-methylpiperazin-1-yl)sulfonyl]-5-(pyridin-4-yl)benzoic acid
N-butyl-4-{3-[(pyridin-3-ylmethyl)carbamoyl]piperidin-1-yl}piperidine-1-carboxamide
6-(morpholin-4-yl)-N4-(prop-2-en-1-yl)pyrimidine-2,4-diamine
5-benzyl-4-[1-(3,4-dimethoxybenzenesulfonyl)piperidin-4-yl]-2-methylpyrimidine
5-{3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
2-methyl-5-{[2-(1-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]methyl}-[1,2,4]triazolo[1,5-a]pyrimidin-7-ol
3-[2-(1H-imidazol-4-yl)-1H-imidazol-1-yl]piperidin-2-one
1-(6-hydroxy-1,4-oxazepan-4-yl)-2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethan-1-one
1-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-4-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperazine
N-[2-(cyclohex-1-en-1-yl)ethyl]-1-[3-(morpholin-4-yl)propyl]-6-oxopiperidine-3-carboxamide
1-methyl-2-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine
3-[5-(3-acetamidobenzoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanoic acid
methyl (2S)-2-{[4-(4-acetamido-1H-pyrazol-1-yl)phenyl]formamido}-2-phenylacetate
1-[(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)pyrrolidin-1-yl]-2-(2H-1,2,3,4-tetrazol-2-yl)ethan-1-one
2-({[1-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)ethyl]amino}methyl)-5,8-dimethylquinolin-4-ol
N-methyl-N-[1-(2-phenylethyl)piperidin-3-yl]-3-(prop-2-en-1-yloxy)benzamide
N-cyclopentyl-N-{[3-methoxy-4-(oxan-2-ylmethoxy)phenyl]methyl}thiophene-2-carboxamide
2-(5-methyl-2-phenyl-1H-imidazole-4-carbonyl)-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
3-(prop-2-en-1-yl)-1-[4-(1H-pyrazol-1-yl)butanoyl]piperidine-3-carboxylic acid