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4-(2-methoxyethyl)-N-[3-(3-methylphenyl)phenyl]piperazine-1-carboxamide
N-benzyl-1-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]piperidine-4-carboxamide
ethyl 4-[(2-chlorophenyl)methyl]-1-[(4-methylthiophen-2-yl)sulfonyl]piperidine-4-carboxylate
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-(6-ethylpyrimidin-4-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
3-{[(2,2-dimethyloxan-4-yl)amino]methyl}-1-{[3-(trifluoromethyl)phenyl]methyl}-1H,2H,6H,7H,8H-cyclopenta[g]quinolin-2-one
2-(1-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-2-yl)-1H-1,3-benzodiazole
1-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}-4-phenylpiperidine-4-carbonitrile
N-(1,3-dimethyl-1H-pyrazol-5-yl)-2-[3,5-dimethyl-4-(quinolin-6-yl)-1H-pyrazol-1-yl]acetamide
N-[(1-methanesulfonylpiperidin-3-yl)methyl]-3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
methyl({[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}){[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}amine
2-[4-(1-benzothiophen-3-yl)-2-(morpholin-4-ylmethyl)phenoxy]-N-[(3-methyl-1,2-oxazol-5-yl)methyl]acetamide
2-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}-6-methylpyridine-3-carboxylic acid
7-fluoro-4-(2-methylpyrrolidine-1-carbonyl)-2-(1-propyl-1H-pyrazol-4-yl)quinoline
2-(2-phenylethyl)-9-[2-(pyrrolidin-1-yl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
2-[(3-methoxyphenyl)amino]-N-methyl-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]butanamide
{4-[(3,4-dimethylphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}(pyridin-3-yl)methanol
dimethyl[1-(2-methylphenyl)-2-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)ethyl]amine
N4-{[1-(morpholin-4-yl)cyclopentyl]methyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
2-{1-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]pyrrolidin-3-yl}benzoic acid
3-(3-hydroxy-1,2-oxazol-5-yl)-1-[(1R,3S)-1-hydroxy-3-methoxy-7-azaspiro[3.5]nonan-7-yl]propan-1-one
8-{3-[(3-fluorophenyl)methoxy]benzoyl}-2,8-diazaspiro[4.5]decan-3-one
1-{4-[1-methyl-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]phenyl}pyrrolidin-2-one
1-(2-methoxyacetyl)-N-{[4-methyl-2-(propan-2-yl)-1,3-thiazol-5-yl]methyl}piperidine-3-carboxamide
1-[2-({7-cyclopropanecarbonyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}amino)ethyl]-4,6-dimethyl-1,2-dihydropyrimidin-2-one
(2S,4R)-1-[(4-chlorophenyl)methyl]-N-cycloheptyl-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidine-2-carboxamide
1-{1-[2-(methylsulfanyl)benzoyl]piperidin-3-yl}-2-phenylethan-1-one
1-methyl-N-[2-(phenylsulfanyl)ethyl]-3-(trimethyl-1H-pyrazol-4-yl)-1H-pyrazole-5-carboxamide
(1-benzofuran-2-ylmethyl)({[1-(2-methoxyethyl)piperidin-4-yl]methyl})(pyridin-4-ylmethyl)amine
5-[3-(methoxymethyl)piperidine-1-carbonyl]-2-(pyridin-4-yl)pyridine
2-{5-[1-(pyridin-2-yl)piperidin-3-yl]-3-(pyridin-3-yl)-1H-1,2,4-triazol-1-yl}ethan-1-ol
(2S)-1-[2-(2-fluorophenyl)acetyl]-N-[3-(1H-pyrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
2-({4-[(4-chlorophenyl)methyl]-4-(hydroxymethyl)piperidin-1-yl}methyl)-6-methoxyphenol
N'-cyclopentyl-N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]butanediamide
N-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4-sulfamoylbenzamide
2-{[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
N-[(2S)-1-hydroxy-3-methylbutan-2-yl]-5-[(4-hydroxypiperidin-1-yl)methyl]-1,2-oxazole-3-carboxamide
2,3,6-trimethyl-N-[2-(N-methylmethanesulfonamido)ethyl]quinoline-4-carboxamide
(2S,4R)-N,N-diethyl-1-(naphthalen-1-ylmethyl)-4-[(1-propylpiperidin-4-yl)amino]pyrrolidine-2-carboxamide
3-hydroxy-3-({[(4-methoxyphenyl)methyl]amino}methyl)-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-8-(6-methylpyridin-2-yl)-1,8-diazaspiro[4.5]decane
(4aR,8aR)-1-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-6-(3-methoxybenzoyl)-decahydro-1,6-naphthyridine
(2S,4S,5R)-5-(2,3-difluorophenyl)-4-[(2-methoxyethyl)(methyl)carbamoyl]-1-methylpyrrolidine-2-carboxylic acid
2-[4-(2-methylphenyl)-3-oxopiperazine-1-carbonyl]benzonitrile
1-[(3-methylphenyl)methyl]-4-{[6-(pyrrolidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}piperazine
4-[1-(4-fluorophenyl)-3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]-1-(prop-2-en-1-yl)pyrrolidin-2-one
1-{[2-methanesulfonyl-1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-4-(2-methoxyphenyl)-2-methylpiperazine
2-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-6-(2-methylpropyl)pyrimidine-4-carboxamide
4-(dimethylamino)-1-{4-[(3-fluorophenyl)methyl]piperazin-1-yl}butan-1-one
methyl (2S)-1-{[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidine-2-carboxylate
4-(1-benzofuran-2-ylmethyl)-1-methyl-9-(prop-2-en-1-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one