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4-[(4-chloro-3-fluorophenyl)methyl]-3-[2-(1,2-oxazolidin-2-yl)-2-oxoethyl]piperazin-2-one
9-[2-(4-fluorophenyl)acetyl]-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[(4-hydroxy-6-methylpyrimidin-2-yl)methyl]-2-(piperidin-1-yl)-2,3-dihydro-1H-indene-2-carboxamide
N,4-dimethyl-4-({[4-(trifluoromethoxy)phenyl]carbamoyl}amino)pentanamide
1-{1-[(2,3-dimethyl-1H-indol-7-yl)methyl]piperidin-4-yl}pyrrolidin-2-one
1-(2-methoxyethyl)-4-[1-(2-methoxyphenyl)-1H-pyrazole-4-carbonyl]piperazine
N-benzyl-3-(2-ethylphenoxy)azetidine-1-sulfonamide
2-{3-[3-(4-ethyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]pyrazolo[1,5-a]pyrimidin-6-yl}ethan-1-ol
4-[(dipropylamino)methyl]-N-(1-methoxybutan-2-yl)benzamide
4-(1-tert-butyl-3,5-dimethyl-1H-pyrazol-4-yl)-5,7-dimethoxy-1,2,3,4-tetrahydroquinolin-2-one
ethyl 1-[({1-[(3-fluorophenyl)methyl]-1H-pyrazol-5-yl}carbamoyl)methyl]-1H-imidazole-2-carboxylate
3-(1H-1,3-benzodiazol-2-yl)-N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}propanamide
(2S)-2-hydroxy-1-{4-[2-methyl-6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-1-yl}propan-1-one
1-[(3-hydroxyphenyl)methyl]-N-[4-(pyridin-3-yloxy)phenyl]piperidine-4-carboxamide
N-{[2-(4-acetylpiperazin-1-yl)pyridin-3-yl]methyl}-3-fluoro-4-methoxybenzamide
N-cyclopropyl-2-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridine-4-carboxamide
1-(4-hydroxy-2,3-dimethylphenyl)-5-oxopyrrolidine-3-carboxylic acid
N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1H-pyrrolo[2,3-b]pyridin-6-amine
1-[4-(3,6-dimethylpyrazin-2-yl)piperazin-1-yl]-2-[2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethan-1-one
N-{3-[ethyl(methyl)amino]-2-methylpropyl}-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-{[2-(dimethylamino)pyridin-3-yl]methyl}-2-propyl-1,3-thiazole-4-carboxamide
N-(1-methyl-2-oxopyrrolidin-3-yl)-2-[4-(trifluoromethyl)phenyl]-1,3-thiazole-4-carboxamide
2-(1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}piperidin-4-yl)-1,2,3,4-tetrahydroisoquinoline
2-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-N,N-dimethylpyrimidin-4-amine
4-[5-(ethylsulfanyl)thiophene-2-carbonyl]-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
2-(4-{[4-(methoxymethyl)piperidin-1-yl]methyl}phenyl)-6-(2-methylpropyl)-3,4-dihydropyrimidin-4-one
6-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)pyrrolidine-1-carbonyl]-1,3-benzothiazole
3-{[1-(2-phenylethyl)piperidin-4-yl]oxy}-N-[2-(1H-pyrazol-1-yl)ethyl]benzamide
N-{1-[1-(cyclohex-3-en-1-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-4-phenylbutanamide
1-(4-methyl-1,3-oxazole-5-carbonyl)-N-(6-phenoxypyridin-3-yl)piperidine-4-carboxamide
N-ethyl-5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-N-(2-methylprop-2-en-1-yl)-1,2-oxazole-3-carboxamide
3-[4-(4-methylpyrimidin-2-yl)piperazin-1-yl]propanamide
{[1-benzyl-2-(2-methoxyethanesulfonyl)-1H-imidazol-5-yl]methyl}(ethyl)[(1-methyl-1H-pyrazol-4-yl)methyl]amine
3-{[4-(3-chlorophenyl)-5-{[methyl({[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl})amino]methyl}-4H-1,2,4-triazol-3-yl]sulfanyl}propan-1-ol
5-(2,6-difluorophenoxymethyl)-N-[(2,4-difluorophenyl)methyl]-1,2-oxazole-3-carboxamide
4-(quinolin-4-yl)-1H-pyrrolo[2,3-b]pyridin-6-amine
N-(2-{7-[(4-methylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-phenoxyacetamide
(2-{2-[1-(1-benzofuran-5-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)dimethylamine
2-(dimethylamino)-2-(4-fluorophenyl)-N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]acetamide
N-ethyl-2-{[2-(1H-imidazol-1-yl)ethyl](methyl)amino}pyridine-3-carboxamide
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-(4-hydroxybutyl)acetamide
N-methyl-2-{3-oxo-2-azaspiro[4.4]nonan-2-yl}-N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
2-cyclopropyl-4-phenyl-9-(pyrazin-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)oxan-4-amine
3-[4-(cyclobutylamino)-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-7-carbonyl]pyridin-2-ol
4-[4-({3-cyclopropyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}methyl)phenyl]-2-methylbutan-2-ol
(4-{5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}morpholin-2-yl)methanamine
3-[4-(1,3-benzoxazol-2-yl)phenyl]-1-(1,4-oxazepan-6-ylmethyl)urea
N-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}acetamide
N-{[2,5-dimethoxy-4-(methylsulfanyl)phenyl]methyl}-N-(pyridin-4-ylmethyl)cyclopropanamine