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2-({3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}methyl)benzonitrile
7-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-4-(4-methoxybenzenesulfonyl)-9-(oxolan-2-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-1-[3-(1H-pyrazol-1-yl)benzoyl]piperidine
2-(3-methyl-5-{2H,3H-thieno[3,4-b][1,4]dioxin-5-yl}-1H-1,2,4-triazol-1-yl)pyridine
N-ethyl-1-[(3-methoxyphenyl)methyl]-5-[3-(5-methylfuran-2-yl)butyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2,3-dimethyl-7-[2-methyl-3-(1H-1,2,4-triazol-1-yl)propanoyl]-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
N-[2-(quinolin-8-yloxy)ethyl]-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl](methyl){2-[2-(prop-2-en-1-yl)phenoxy]ethyl}amine
1-[3-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]-2-[1-(propan-2-yl)piperidin-4-yl]ethan-1-one
(3S,4S)-4-[4-(2-methoxyphenyl)piperazin-1-yl]-1-(pyridine-2-carbonyl)pyrrolidin-3-ol
9-(3-phenyl-1,2,4-oxadiazol-5-yl)-1-oxa-9-azaspiro[5.5]undecan-5-ol
N-butyl-2-(methylamino)-N-[(5-methylthiophen-2-yl)methyl]pyrimidine-5-carboxamide
9-(2-aminopyridine-4-carbonyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
4-[(4-methyl-5-{1-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]piperidin-3-yl}-4H-1,2,4-triazol-3-yl)methyl]morpholine
N-[(5-{[(3-methylphenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)methyl]thiophene-2-carboxamide
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-6-methylpyridazin-3-amine
2-(3-{4-[1-(pyrrolidin-1-yl)ethyl]phenyl}phenoxy)acetamide
1-(4-chloro-1H-indole-2-carbonyl)-N,N-dimethylazepan-4-amine
1-[2-(3-benzyl-1H-1,2,4-triazol-5-yl)phenyl]-1,3-diazinane-2,4-dione
3-[2-(3-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamido]propanamide
6-[(1R,2R,6S,7S)-10-oxa-4-azatricyclo[5.2.1.02,6]decane-4-sulfonyl]-1,2,3,4-tetrahydroquinolin-2-one
({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)(methyl)[(2E)-2-methylbut-2-en-1-yl]amine
2-{2-[4-(4-fluorophenyl)-1,4-diazepan-1-yl]-2-oxoethyl}-1,2-dihydrophthalazin-1-one
2-{[3-(2-methoxyethyl)piperidin-1-yl]methyl}-3-methyl-1H-indole
1-{[(oxolan-2-ylmethyl)[(2E)-3-phenylprop-2-en-1-yl]carbamoyl]methyl}piperidine-4-carboxamide
3-{[1-(methoxymethyl)cyclobutyl]formamido}-N-phenylpropanamide
6-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]pyridine-2-carbonitrile
2-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]oxy}-4-methoxy-N-(2-methoxyethyl)benzamide
2-[4-(1-methylpiperidin-4-yl)piperidin-1-yl]-5-[(methylsulfanyl)methyl]pyridine
N-[1-(1,3-benzothiazol-2-yl)piperidin-3-yl]-4-methyl-1H-imidazole-5-carboxamide
1-[(3R,4R)-4-hydroxy-4-(2-methoxyethyl)-3-methylpiperidin-1-yl]-2-(methylsulfanyl)ethan-1-one
2-[1-(3-methylbut-2-en-1-yl)-4-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperazin-2-yl]ethan-1-ol
(3S,4R)-4-(2-methoxyphenyl)-1-[4-(2-methyl-1H-imidazol-1-yl)butanoyl]pyrrolidine-3-carboxylic acid
1-(4-{[methyl(quinoxalin-2-ylmethyl)amino]methyl}thiophen-2-yl)ethan-1-one
N-(2-{7-[(3-fluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-4-methoxybenzamide
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-ethyl-N-{2-[(4-methylphenyl)sulfanyl]ethyl}acetamide
N-[1-(2-methoxyphenyl)ethyl]-N-methyl-2-(4-oxo-3,4-dihydroquinazolin-3-yl)acetamide
6-(2-chlorophenyl)-N-(1-hydroxypropan-2-yl)-N,7-dimethyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
N-{[2-(4-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-2-methylpyrimidine-5-carboxamide
2-[2-(4-chlorophenyl)morpholin-4-yl]-1,3-thiazole-4-carboxamide
N-{[4-(cyclobutylmethoxy)phenyl]methyl}-N-cyclopropyl-3,4-difluorobenzene-1-sulfonamide
5-methyl-4-(1-methyl-1H-1,2,4-triazol-5-yl)-N-[(4-phenyloxan-4-yl)methyl]pyrimidin-2-amine
ethyl 3-benzyl-1-cyclopentylpiperidine-3-carboxylate
(2S,4S)-4-amino-1-(1,6-dimethyl-1H-indole-2-carbonyl)-N-ethylpyrrolidine-2-carboxamide
1-phenyl-4-(7-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)butane-1,4-dione
{[1-(3-fluorophenyl)-3-(5-methylfuran-2-yl)-1H-pyrazol-4-yl]methyl}[3-(4-methyl-1,3-thiazol-5-yl)propyl]amine
1-[2-({[5-(methoxymethyl)furan-2-yl]methyl}amino)ethyl]-N-(2-phenylethyl)-1H-1,2,3-triazole-4-carboxamide
(2S,4R)-4-amino-N-methyl-1-(6-methyl-2-phenylpyrimidin-4-yl)pyrrolidine-2-carboxamide
4-ethyl-3-{1-[2-(2-phenyl-1H-imidazol-1-yl)acetyl]piperidin-3-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
2-[5-(2,4-difluorophenyl)-1H-indazol-1-yl]-N-(2-ethyl-2H-1,2,3-triazol-4-yl)acetamide