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5-(2,6-dimethylphenoxymethyl)-N-ethyl-N-[2-(pyrrolidin-1-yl)ethyl]-1,2-oxazole-3-carboxamide
N-{[2-(morpholin-4-yl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]-1,3-thiazole-5-carboxamide
3-{2-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl}phenol
4-[3-(1H-imidazol-2-yl)piperidin-1-yl]-6-(morpholin-4-yl)pyrimidin-2-amine
N-{[1-(hydroxymethyl)cyclobutyl]methyl}-6-(3-methoxyphenyl)-N-methylimidazo[2,1-b][1,3]thiazole-3-carboxamide
6-(2-aminoethyl)-N-cyclopropyl-2-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]pyrimidin-4-amine
9-(cyclopropylmethyl)-1-methyl-4-[(2-methylpyrimidin-5-yl)methyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
2-(4-{1-[4-(furan-2-yl)pyrimidin-2-yl]-5-(methoxymethyl)-1H-pyrazole-4-carbonyl}piperazin-1-yl)phenol
6-[(3S,7S)-3-(hydroxymethyl)-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-trien-5-yl]pyridine-3-carbonitrile
5-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]-N-methyl-N-(1,2-oxazol-3-ylmethyl)pyridin-2-amine
({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)(methyl)[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]amine
1-(2-methoxyethyl)-4-[4-(4-methoxyphenyl)-1H-imidazol-2-yl]pyrrolidin-2-one
N-({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)-4-(1H-pyrazol-3-yl)benzamide
1-[(4-fluorophenyl)methyl]-3-(3-phenyl-1,2,4-thiadiazol-5-yl)urea
1-{2,3-dimethyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}piperidine-3-carboxamide
2-{9-[(2,4-difluorophenyl)methyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}acetic acid
N-[1-(4-tert-butylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-acetamidoacetamide
2-(4-{[4-(2-amino-6-oxo-1,6-dihydropyrimidin-4-yl)piperazin-1-yl]methyl}phenoxy)acetic acid
1-[(4aR,8aS)-1-(thiophene-2-carbonyl)-decahydro-1,6-naphthyridin-6-yl]-2-phenoxyethan-1-one
2-cyclobutyl-1-[1-(2-methyl-1,3-thiazole-4-carbonyl)piperidin-4-yl]-5-(trifluoromethyl)-1H-1,3-benzodiazole
(1R,5R)-6-(1-benzofuran-5-ylmethyl)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
4-(5-{7-[ethoxy(phenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl}furan-2-yl)-2-methylbut-3-yn-2-ol
N-[3-(1H-imidazol-1-yl)-1-phenylpropyl]-1-[(4-methoxyphenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
6-methyl-2-{2-methyl-2,7-diazaspiro[4.5]decan-7-yl}pyridine-3-carbonitrile
(but-2-yn-1-yl)({[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-1H-pyrazol-4-yl]methyl})(furan-2-ylmethyl)amine
N-benzyl-1-(2-ethylpyrimidine-5-carbonyl)-N-methylpiperidin-4-amine
2-(adamantan-1-yl)-5-[2-(aminomethyl)morpholine-4-carbonyl]pyrimidin-4-ol
N-[2-(2-ethoxyphenyl)ethyl]-2-(1-methylpiperidin-2-yl)acetamide
8-cyclopropanecarbonyl-2-[(2-methyl-1,3-oxazol-4-yl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-2-{tricyclo[9.4.0.03,8]pentadeca-1(11),3(8),4,6,12,14-hexaen-2-yl}acetamide
5-cyclopropanecarbonyl-1'-(3,4-dimethylbenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-(2-{[(2-aminopyrimidin-4-yl)amino]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl)ethan-1-one
2-benzyl-N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-1,3-benzoxazole-5-carboxamide
6-methyl-N-(propan-2-yl)-5-[5-(pyridazin-4-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridine-2-carboxamide
2-[(3R,4S)-3-[(6-cyanopyridin-2-yl)amino]-4-cyclopropylpyrrolidin-1-yl]-N,N-dimethylacetamide
1,5-dimethyl-N-({1-[(4-methylpiperazin-1-yl)methyl]cyclopropyl}methyl)-1H-pyrazole-4-carboxamide
(1S,6R)-9-(1-ethyl-3,5-dimethyl-1H-pyrazole-4-carbonyl)-3-methyl-3,9-diazabicyclo[4.2.1]nonan-4-one
4-cyclopropyl-6-[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]pyrimidine
1-(1-ethylpiperidin-4-yl)-4-[4-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]piperazine
4-benzyl-3-ethyl-1-(4-ethylbenzoyl)-1,4-diazepan-5-one
7-methyl-2-{2-[3-(1H-1,2,3,4-tetrazol-1-yl)phenoxy]acetyl}-2,7-diazaspiro[4.5]decan-6-one
(3R,4S)-1-{6-chloroimidazo[1,2-a]pyridine-2-carbonyl}-4-(5-methylfuran-2-yl)pyrrolidin-3-amine
4-fluoro-N-(2-{7-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)benzamide
2-[4-(3-cyanopyridin-2-yl)-1H-pyrazol-1-yl]-N-(1-cyclohexyl-1H-pyrazol-5-yl)acetamide
2-(4-chloro-2-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]methyl}phenoxy)acetic acid
N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-2-methyl-1H-1,3-benzodiazole-5-carboxamide
(2S)-2-amino-1-{4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-cyclohexylethan-1-one
N-[(3R,7S,8aS)-3-[(1S)-1-hydroxyethyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-methoxybenzamide
N-[(1R,3S)-3-(cyclooctylcarbamoyl)cyclopentyl]-3-hydroxybenzamide
N-(1-{7-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)pyridine-3-carboxamide