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4-(4-cyclopentyl-1H-1,2,3-triazol-1-yl)-1-(2-fluorobenzenesulfonyl)piperidine
methyl N-{4-[2-(dimethylamino)ethoxy]-1-(4-fluorophenyl)-1H-indazol-3-yl}carbamate
8-(1-ethyl-2-oxo-1,2-dihydropyridine-4-carbonyl)-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-(4-{2-azabicyclo[2.2.1]heptane-2-carbonyl}piperidin-1-yl)-7-methoxy-4-methylquinazoline
N-ethyl-1-[(E)-2-phenylethenesulfonyl]-N-(pyridin-4-ylmethyl)piperidin-3-amine
N-tert-butyl-2-{3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl}acetamide
N-{[5-(2-acetylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3,5-difluorobenzamide
2-{5H,6H,7H,8H-imidazo[1,5-a]pyrazin-7-yl}pyridine-3-carbonitrile
2-[(4-fluorophenyl)methyl]-4-[(2E)-2-methylbut-2-en-1-yl]morpholine
1-cyclopentyl-5-{4-[(3-fluorophenyl)methyl]piperazine-1-carbonyl}-4-oxo-N-(prop-2-en-1-yl)-1,4-dihydropyridine-3-carboxamide
N-(3-cyclopentylpropyl)-3-[5-(3-phenylpropyl)-1,3,4-oxadiazol-2-yl]propanamide
3-[5-(1H-imidazol-4-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]-1-(4-methylpiperazin-1-yl)propan-1-one
1-cyclopropanecarbonyl-4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidine-1-carbonyl]piperidine
9-[(3-fluoro-4-methylphenyl)methyl]-2-(3-methoxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
3-(4-phenoxybutyl)-1,3-diazinane-2,4-dione
1-{4-[3-(4-fluorophenyl)pyrrolidine-1-carbonyl]-3,5-dimethyl-1H-pyrrol-2-yl}ethan-1-one
5-cyclopropanecarbonyl-1'-(2,5-dimethylbenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-chloro-N-{[1-(dimethylamino)cyclohexyl]methyl}-6-fluorobenzamide
3-(1H-imidazol-4-ylmethyl)-4-[5-(pyrrolidin-1-ylmethyl)furan-2-carbonyl]piperazin-2-one
N-methyl-N-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}-1H-pyrazole-4-carboxamide
2-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
2-[5-(1-ethyl-1H-indol-6-yl)-4-phenyl-1H-imidazol-1-yl]acetamide
N-[1-(2-chlorophenyl)cyclopropyl]-1-(2-methoxyacetyl)piperidine-4-carboxamide
(1-{[6-chloro-2-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}piperidin-3-yl)methanol
2-amino-N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-N-methyl-6-(2-methylpropyl)pyrimidine-4-carboxamide
4-(piperidin-4-yl)-8-thia-4,6-diazatricyclo[7.5.0.02,7]tetradeca-1(9),2(7),5-trien-3-one
3-cyano-5-fluoro-N-(1-hydroxybutan-2-yl)-N-(pyridin-3-ylmethyl)benzamide
4-[(1E)-1-(furan-2-yl)prop-1-en-2-yl]-1-methyl-3-(pyridin-3-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
4-(1,2,3,6-tetrahydropyridin-1-yl)-7-(thiophene-2-carbonyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-2-amine
N-[2-hydroxy-2-(4-hydroxyphenyl)ethyl]-3-(piperidine-1-carbonyl)pyrazine-2-carboxamide
1-(cyclohexylmethyl)-3-hydroxy-3-({[2-(3-methylpyridin-2-yl)ethyl]amino}methyl)piperidin-2-one
1-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)-3-(2-oxo-2,3-dihydro-1,3-benzoxazol-6-yl)urea
(3ar,6ar)-N-benzyl-N-(1,3-thiazol-2-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
1,3,6-trimethyl-5-{4-[1-(piperidin-1-yl)ethyl]phenyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
methyl 4-{[4-(1,3-benzoxazol-2-yl)phenyl]carbamoyl}piperidine-1-carboxylate
N-[(4-fluorophenyl)methyl]-N-(3-hydroxypropyl)-2,8-dimethylquinoline-4-carboxamide
2-[(4-chlorophenyl)methyl]-8-(pyrimidin-2-yl)-2,8-diazaspiro[4.5]decan-3-one
2-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-7-fluoro-3-methyl-1H-indole
(4aS,8aR)-1-(2-aminoethyl)-6-(5-fluoro-2-methoxybenzoyl)-decahydro-1,6-naphthyridin-2-one
1-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-4-(pyridin-3-yl)piperidin-4-ol
1-[2-(dimethylamino)-2-(4-methylphenyl)acetyl]piperidine-4-carboxylic acid
1,3-dimethyl-N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
(2S,4R)-N,N-diethyl-4-(2-hydroxyacetamido)-1-(4-methoxybenzoyl)pyrrolidine-2-carboxamide
1-(4-benzyl-6-hydroxy-1,4-diazepan-1-yl)-4-phenylbutane-1,2-dione
N-[1-(3-cyanopyridin-2-yl)piperidin-4-yl]-2-(2,3-dihydro-1H-inden-1-yl)acetamide
5-[4-(3-phenylpropyl)-1,4-diazepane-1-carbonyl]piperidin-2-one
(1R,3S)-3-(2-aminoethoxy)-7-(2-fluoro-4-methylbenzoyl)-7-azaspiro[3.5]nonan-1-ol
N-(4-ethyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)-3-(4H-1,2,4-triazol-3-yl)piperidine-1-carboxamide
N-(4-methoxyphenyl)-1-[5-(4-methoxyphenyl)furan-2-carbonyl]piperidin-3-amine
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N,2-dimethyl-6-(propan-2-yl)pyrimidin-4-amine