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[(3R,4R)-1-(2,5-difluorobenzoyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
N-[(5-chloro-1-benzothiophen-3-yl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxamide
1-[2-({[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}amino)ethyl]piperidin-4-ol
N-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
N-(2-methyl-2H-1,2,3-triazol-4-yl)-2-[3-(pyrimidin-5-yl)-1H-indazol-1-yl]acetamide
(4aR,7aS)-1-cyclobutanecarbonyl-4-[(2-ethoxyphenyl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-{[2-(3-methoxyphenyl)-1,3-thiazol-5-yl]methyl}-4-(5-methyl-1,2,4-oxadiazol-3-yl)piperidine
1,3,5-trimethyl-7-[4-(1-methyl-1H-1,2,4-triazol-5-yl)pyrimidin-2-yl]-3,7-diazabicyclo[3.3.1]nonane
6-({3-cyclopentyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}methyl)-2-(methylsulfanyl)pyridine-3-carbonitrile
N-[(2R,4R,6S)-2-phenyl-6-[2-(pyridin-2-yl)pyrimidin-5-yl]oxan-4-yl]acetamide
(2S,4R)-4-{[(4-methoxy-2,3-dimethylphenyl)methyl]amino}-N-(2-methoxyethyl)-1-(propan-2-yl)pyrrolidine-2-carboxamide
N-[2-(cyclohex-1-en-1-yl)ethyl]-2-[1-(naphthalen-1-ylmethyl)-3-oxopiperazin-2-yl]acetamide
4-(3,4-dimethylphenyl)-6-methoxypyrimidine
(4-{[2-(butylsulfanyl)pyrimidin-5-yl]methyl}-1-methylpiperazin-2-yl)methanol
N-ethyl-2-(1-ethyl-1H-pyrazol-4-yl)-7,8-dimethyl-N-(propan-2-yl)quinoline-4-carboxamide
N-[(4-fluorophenyl)methyl]-2-methyl-N-(pyridin-2-ylmethyl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
1-{[4-(hydroxymethyl)oxan-4-yl]methyl}-3-[2-(4-methoxyphenyl)phenyl]-1-methylurea
1-{4-[(3-methylphenyl)methyl]piperazin-1-yl}-3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]propan-1-one
(3S,4S)-1-{[4-(4-fluorophenyl)-1,3-thiazol-2-yl]methyl}-4-(morpholin-4-yl)pyrrolidin-3-ol
1-oxo-N-{2-[(2S)-pyrrolidin-2-yl]ethyl}-1,2-dihydroisoquinoline-4-carboxamide
1-benzyl-4-{3,5-dimethyl-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyrazine-7-carbonyl}-1H-pyrazole
N-propyl-2-(2,6,6-trimethyl-4-oxo-1-propyl-4,5,6,7-tetrahydro-1H-indol-3-yl)acetamide
5-{[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}pyrimidine
7-[2-(4,6,7-trimethyl-1-benzofuran-3-yl)acetyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
5-[4-(3-methyl-1,2-oxazole-5-carbonyl)piperazin-1-yl]-6-phenyl-2,3-dihydropyridazin-3-one
(3aS,6aS)-2-(dimethylsulfamoyl)-5-(furan-3-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(1S,5R)-3-benzyl-6-(1-ethyl-3,5-dimethyl-1H-pyrazole-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-4-[(3-methyl-1H-1,2,4-triazol-5-yl)methyl]-1,4-diazepan-6-ol
N-[1-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
methyl 6-[1-(4-chlorophenyl)cyclobutanecarbonyl]-2-(ethylsulfamoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-[9-methoxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl]cyclopropane-1-carboxamide
(2S,4R)-1-[(4-hydroxyphenyl)methyl]-4-[(4-methoxyphenyl)sulfanyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
9-(2-hydroxy-4-methylbenzoyl)-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
4-methyl-2-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}phenol
N-[(7R,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-(4-methoxy-3-methylphenyl)acetamide
3-(5-{2-[2-(1-benzofuran-2-yl)-1H-imidazol-1-yl]ethyl}-1H-1,2,4-triazol-3-yl)pyridine
N-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]cyclopropanamine
4-({methyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amino}methyl)-N-(2-oxo-2,3-dihydro-1H-indol-5-yl)benzamide
N-ethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-6-{methyl[(1-methylpyrrolidin-2-yl)methyl]amino}pyridine-3-carboxamide
(2-methoxyethyl)({1-[1-(3-methylthiophene-2-carbonyl)piperidin-4-yl]-2-phenylethyl})(pyridin-2-ylmethyl)amine
1-[1-(4-methyl-1,3-thiazol-2-yl)piperidin-4-yl]-3-phenylpropan-1-ol
N-(2-chloro-6-methylphenyl)-2-cyclopropyl-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
3-cyclopropyl-5-[3-(thiophen-2-yl)propyl]-1H-1,2,4-triazole
2-cyclopropyl-N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]-1,3-benzoxazole-6-carboxamide
2-[(6-methoxypyridin-3-yl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
[(4-fluoro-2-methoxyphenyl)methyl]({1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl})amine
(3R,4R)-1-[6-(4-fluorophenyl)pyridazin-3-yl]-3,4-dimethylpyrrolidin-3-ol
3-{2-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-oxoethyl}imidazolidine-2,4-dione
(2S,4R)-4-[2-(5-chloro-6-methyl-1-benzofuran-3-yl)acetamido]-N,1-dimethylpyrrolidine-2-carboxamide
3-(3-hydroxyquinoxalin-2-yl)-N-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}propanamide