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9-(4-oxo-4-phenylbutyl)-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N2-[3-(3,4-dimethoxyphenyl)propyl]-5-fluoro-N4,N4-dimethylpyrimidine-2,4-diamine
N,N-diethyl-1-[(1s,4s)-4-[2-(3-methoxyphenyl)acetamido]cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
1-[7-(2-methylphenyl)-9-(oxolan-3-yloxy)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(pyridin-2-ylsulfanyl)ethan-1-one
2-(5-acetylthiophen-3-yl)-N-[(4-methylphenyl)methyl]acetamide
[(3R,4R)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-(quinoline-6-carbonyl)pyrrolidin-3-yl]methanol
N-{1-[1-(4-chloro-3-fluorobenzoyl)piperidin-4-yl]-1H-pyrazol-5-yl}oxolane-3-carboxamide
[(3S,5R)-1-(3-fluoro-4-methoxybenzoyl)-5-{[(2-methoxyethyl)(methyl)amino]methyl}piperidin-3-yl]methanol
N-[1-(1H-1,3-benzodiazol-2-yl)ethyl]-2-(pyrrolidin-1-yl)-6-(thiophen-2-yl)pyridine-3-carboxamide
1-[4-(pyrrolidin-1-yl)butanoyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-phenyl-4-{[1,2,4]triazolo[1,5-a]pyrimidine-2-carbonyl}morpholine
2-(1-{[1-(9H-purin-6-yl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)propan-2-ol
4-(2,6-dimethylpyridin-3-yl)-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}pyrimidin-2-amine
4-[4-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]-8-methyl-7-(pyrrolidin-1-yl)-1,2,3,4-tetrahydroquinolin-2-one
N-[2-(5-chloro-1H-1,3-benzodiazol-2-yl)ethyl]-2-cyclopropyl-6-methyl-4-oxo-1-(thiophen-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
4,4,4-trifluoro-1-[7-(2-phenylethyl)-2,7-diazaspiro[4.5]decan-2-yl]butan-1-one
4-[(1-acetylpiperidin-4-yl)oxy]-3-methoxy-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]benzamide
2-[1-(6-methoxy-3-methyl-1-benzofuran-2-carbonyl)pyrrolidin-2-yl]-1-methyl-1H-1,3-benzodiazole
N-methyl-N-[2-(1H-pyrazol-4-yl)ethyl]-7-(pyridine-3-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]-4-ethyl-1,4-diazepan-5-one
1-{[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-N,N-diethylpiperidine-3-carboxamide
1-[1-(2-phenylethyl)-5-(2,2,3,3-tetramethylcyclopropanecarbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]-1,4-diazepan-5-one
({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)(methyl)[4-(morpholin-4-yl)butyl]amine
2-[(3,4-difluorophenyl)methyl]-8-ethyl-2,8-diazaspiro[4.5]decan-3-one
4-(3-fluorophenoxy)-1-(oxolane-3-carbonyl)piperidine-4-carboxylic acid
1-ethyl-N-[1-(3-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-methyl-1H-pyrazole-5-carboxamide
3-fluoro-5-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine
3-(3-fluoro-4-methoxybenzoyl)-1-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}piperidine
3-{1-[(2,3-difluorophenyl)methyl]piperidin-4-yl}-N-(prop-2-en-1-yl)pyrrolidine-1-carboxamide
8-cyclopropanecarbonyl-2-[(1-methyl-1H-imidazol-2-yl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-[benzyl(methyl)amino]-3-(2-methoxy-5-{[methyl(pyrazin-2-ylmethyl)amino]methyl}phenoxy)propan-2-ol
1-{2-[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-oxoethyl}pyrrolidin-2-one
2-amino-4-(3-propoxypiperidin-1-yl)quinazoline-6-carboxylic acid
2-(4-ethylpiperazin-1-yl)-N-methyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)acetamide
1-{2-[(7-hydroxy-3,7-dimethyloctyl)amino]ethyl}cyclopentan-1-ol
(4aS,8aR)-2-[5-(3-fluoro-4-methoxyphenyl)-1,2,4-triazin-3-yl]-decahydroisoquinoline
3-[3-(2-methylpiperidin-1-yl)azetidin-1-yl]-6-phenylpyridazine
2-(3,4-difluorobenzoyl)-1-(2,3-dimethoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole
N-[(1S,2R)-2-[(2,3-dihydro-1H-inden-2-yl)amino]cyclobutyl]-2-(ethylamino)-4-methyl-1,3-thiazole-5-carboxamide
1-(2-methylpropyl)-6-(pyridin-3-ylmethoxy)-4-(1,3-thiazole-4-carbonyl)-1,4-diazepan-2-one
methyl 3-{3-[4-(2-methylphenyl)piperazin-1-yl]piperidin-1-yl}propanoate
methyl 8-[(3,5-dimethoxyphenyl)methyl]-2-oxo-1-(prop-2-en-1-yloxy)-1,8-diazaspiro[4.5]decane-4-carboxylate
2-methyl-3-({methyl[2-(oxan-2-yl)ethyl]carbamoyl}amino)benzamide
4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]-1-[3-(5-methylfuran-2-yl)butyl]piperidine
5-[1-(1-methyl-1H-pyrrole-2-carbonyl)pyrrolidin-2-yl]-3-phenyl-1,2,4-oxadiazole
1-[3-(2-oxopyrrolidin-1-yl)benzoyl]-4-{[2-(trifluoromethyl)phenyl]methyl}-1,4-diazepan-5-one
2-cyclopropyl-8-[2-(3,4-dimethyl-6-oxo-1,6-dihydropyridazin-1-yl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
3-(3,4-dimethoxyphenyl)-1-[3-hydroxy-3-(hydroxymethyl)piperidin-1-yl]propan-1-one
1-(2,3-dihydro-1H-inden-2-yl)-N-methylpiperidin-3-amine
4,4,4-trifluoro-1-{3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}butan-1-one