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1-{2-[(1R,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-oxoethyl}-1,4-dihydroquinolin-4-one
(3S,4R)-4-(2,3-dimethoxyphenyl)-1-(2-methylpyrimidin-4-yl)pyrrolidine-3-carboxylic acid
2-[1-(2,2-dimethylpropyl)-3-oxopiperazin-2-yl]-N-({5-methylimidazo[1,2-a]pyridin-2-yl}methyl)acetamide
N-(3,5-dimethylphenyl)-6-(1-methyl-1H-pyrazole-5-carbonyl)-6-azaspiro[2.5]octane-1-carboxamide
N-(1-hydroxy-3-methylbutan-2-yl)-6-[4-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
(1R,7S)-3-[(3,4-dimethylphenyl)methyl]-N-methyl-4-oxo-N-(propan-2-yl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
3-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}benzonitrile
1-methyl-6-(quinolin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-{5-[1-(2H-1,3-benzodioxol-5-yl)propan-2-yl]-1-methyl-1H,4H-pyrazolo[3,4-d]imidazol-3-yl}pyridine
[(3R,5S)-1-{[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl}-5-(morpholin-4-ylmethyl)piperidin-3-yl]methanol
[(4-chloro-1-methyl-1H-indazol-3-yl)methyl][(dimethyl-1,2-oxazol-4-yl)methyl]methylamine
N-[(2,5-dimethylphenyl)methyl]azepane-4-carboxamide
N-methyl-N-({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)-3,4-dihydro-2H-1-benzopyran-2-carboxamide
methyl 1-{2-[1-cyclopropyl-2,5-dioxo-3-(4-phenylphenyl)pyrrolidin-3-yl]acetyl}piperidine-2-carboxylate
4-methoxy-6-{6-[(2-methoxyethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}pyrimidin-2-amine
1,3-dimethyl-N-{[8-(thiophen-2-ylmethyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}-1H-pyrazole-5-carboxamide
2-[(5-methylpyrazin-2-yl)methyl]-9-(pyridine-4-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
6-methyl-4-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]-1-[2-(methylsulfanyl)phenyl]piperazin-2-one
4-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
5-({4-phenyl-5-[2-(1H-pyrazol-1-ylmethyl)phenyl]-1H-imidazol-1-yl}methyl)-1H-1,2,3,4-tetrazole
N-(2-ethoxyphenyl)-3,9-diazaspiro[5.6]dodecane-9-carboxamide
4-(8-methylquinolin-5-yl)thiophene-2-carboxamide
1-(2-fluorophenyl)-4-{[5-(oxolan-2-yl)thiophen-2-yl]methyl}piperazine
1-(3-{[2-(3,4-dimethoxyphenyl)ethyl](methyl)amino}piperidin-1-yl)-3-phenylprop-2-yn-1-one
N-[2-(2-methoxyphenyl)ethyl]-6-(quinolin-4-ylmethyl)-6-azaspiro[2.5]octane-1-carboxamide
2-methoxy-4-[(1E)-3-{4-[2-(methylsulfanyl)pyrimidin-4-yl]piperazin-1-yl}prop-1-en-1-yl]phenol
2-(1H-imidazol-2-yl)-N-[(5-methylthiophen-2-yl)methyl]-N-(pyridin-2-ylmethyl)benzamide
1-{[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-(2-methoxyethyl)piperidine
2-[1-(cyclohexylmethyl)-4-[(3-methyl-1H-pyrazol-5-yl)methyl]piperazin-2-yl]ethan-1-ol
3-(azocan-1-yl)-1-[3-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]propan-1-one
N-[(7S,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2,3,4,9-tetrahydro-1H-carbazole-6-carboxamide
3-(2-ethyl-1H-imidazol-1-yl)-1-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]propan-1-one
5-(2-chlorophenyl)-N-[(3S,4S)-4-methoxy-1-(propan-2-yl)pyrrolidin-3-yl]furan-2-carboxamide
4-cyclopropyl-4-methyl-1-[(2-methyl-1,3-thiazol-4-yl)methyl]pyrrolidin-2-one
N,2,2,6,6-pentamethyl-N-{[3-(pyrazin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-amine
1-(2,5-dimethylfuran-3-carbonyl)-4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
2-{1-[(2-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]acetamide
1-methyl-5-{1-[4-(trifluoromethyl)phenyl]-1H-1,2,4-triazol-5-yl}-1,2-dihydropyridin-2-one
1-(2-methyl-1-benzofuran-7-carbonyl)-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
9-methoxy-3-[3-(5-methylfuran-2-yl)butyl]-7-oxo-N-(1,3-thiazol-2-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
1-(2-fluorophenyl)-4-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carbonyl]piperazine
N-[1-(furan-2-ylmethyl)-1H-pyrazol-5-yl]-10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine-5-carboxamide
(3S,4R)-1-{2-[4-(hydroxymethyl)phenyl]acetyl}-4-phenylpyrrolidine-3-carboxylic acid
1-[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidin-1-yl]-2-(4-ethylpiperazin-1-yl)ethan-1-one
N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-{[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidin-3-amine
3-({[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}amino)-N-(2-methoxyphenyl)propanamide
1-(2-methoxyphenyl)-3-[2-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)propyl]urea
4-methoxy-N-(2-methoxyethyl)-2-({1-[(5-methylthiophen-2-yl)methyl]piperidin-4-yl}oxy)benzamide
3-(1,1-dioxo-1λ6-thiolan-3-yl)-3-ethyl-1-[3-(furan-2-yl)phenyl]urea