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1-methyl-4-{2-[2-(methylsulfanyl)phenyl]pyridine-4-carbonyl}piperazine
N-[(1-ethylpyrrolidin-2-yl)methyl]-1-[2-(2-methoxyphenyl)ethyl]-2,6-dimethyl-4-oxo-1,4-dihydropyridine-3-carboxamide
N-(6-methylpyridin-3-yl)-1-[1-(1H-pyrazol-1-ylmethyl)cyclopropanecarbonyl]piperazine-2-carboxamide
N-(3-{[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]amino}propyl)pyridin-3-amine
ethyl 4-(5-methyl-2-phenyl-1H-imidazole-4-amido)piperidine-1-carboxylate
1-{7-[(3,4-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-3-(pyridin-4-yl)propan-1-one
4-{[2-(benzylamino)pyrimidin-5-yl]methyl}-1-phenylpiperazin-2-one
N-[2-(3-chlorophenoxy)ethyl]-N-methylspiro[2.2]pentane-1-carboxamide
(2R,3R,6R)-3-(4-methoxyphenyl)-5-(quinoxalin-2-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-(2-{4-[1-(4-chlorophenyl)cyclopropanecarbonyl]piperazin-1-yl}ethyl)-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
N-(3-fluorophenyl)-1-[(1-phenyl-1H-pyrazol-4-yl)methyl]piperidin-3-amine
4-(3-chloropyridin-2-yl)-1-[(3-methoxyphenyl)methyl]piperazin-2-one
1-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}-2-(4-methyl-1,4-diazepan-1-yl)ethan-1-one
1-cyclohexanecarbonyl-N-(2-methanesulfonylethyl)pyrrolidine-2-carboxamide
N-(5-methyl-1,3,4-thiadiazol-2-yl)-2-[3-(methylsulfanyl)propanoyl]-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
8-{[4-(methylsulfanyl)phenyl]methyl}-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
N-[2-methyl-1-(7-{[3-(trifluoromethyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)propyl]furan-3-carboxamide
7-[4-(1-butyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-3-methyl-3,4-dihydroquinazolin-4-one
5-{[benzyl(methyl)amino]methyl}-N-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-1,2-oxazole-3-carboxamide
5-ethyl-3-[2-(4-methoxyphenyl)ethyl]-5-(1-{[4-(methylsulfanyl)phenyl]methyl}piperidin-4-yl)imidazolidine-2,4-dione
2-[2-(dimethylamino)ethyl]-9-(5-ethyl-1H-pyrrole-2-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
7-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]-1-oxa-7-azaspiro[3.5]nonane
8-(4-amino-5-methylpyrimidin-2-yl)-2-cyclopropanecarbonyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-2-(pyrrolidin-1-yl)benzamide
2-(dimethylamino)-8-[(8-fluoro-4-hydroxyquinolin-2-yl)methyl]-1,3,8-triazaspiro[4.5]dec-1-en-4-one
3-[2-(4-fluorophenyl)ethyl]-1-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperidine
3-(2H-1,3-benzodioxol-5-yl)-N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]propanamide
({6-chloro-2-methylimidazo[1,2-a]pyridin-3-yl}methyl)[(2-fluorophenyl)methyl](2-methoxyethyl)amine
1-[(3-chlorophenyl)methyl]-4-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}piperazine
2-(3-aminoazepane-1-carbonyl)-5-methoxy-4H-pyran-4-one
2-[methyl({4-methyl-5-[1-(oxan-4-yl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)amino]ethan-1-ol
(2R,3S,6R)-3-phenyl-5-(pyridin-4-ylmethyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
[(5-{1-[(2-fluoro-5-methoxyphenyl)methyl]piperidin-3-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]dimethylamine
N-[(2R,3R)-2-methoxy-1'-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(methylsulfanyl)acetamide
3-[4-(3-acetylphenyl)phenyl]-1-ethyl-1-(oxan-4-yl)urea
7-(2-hydroxy-5-methoxybenzoyl)-2-(pyridin-4-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-(1-benzylpiperidin-4-yl)-1-[(3R,4S)-4-hydroxy-3,4-dimethylpiperidin-1-yl]ethan-1-one
2-chloro-4-({[(1-ethyl-1H-imidazol-2-yl)methyl](methyl)carbamoyl}amino)-N,N-dimethylbenzamide
({2,4-dimethyl-5-[(4-methylpiperazin-1-yl)methyl]phenyl}methyl)(methyl)(oxan-2-ylmethyl)amine
1-(2-cyclopropylphenyl)-3-[(1-propyl-1H-pyrazol-4-yl)methyl]urea
4-[2,2-dimethyl-3-(morpholin-4-yl)propyl]-2-[(3-fluorophenyl)methyl]morpholine
1-methyl-N-(1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-3-yl)piperidine-4-carboxamide
5-methoxy-2-[3-(pyridin-2-ylmethoxy)piperidine-1-carbonyl]-4H-pyran-4-one
3-({ethyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amino}methyl)-6-methoxy-1,2-dihydroquinolin-2-one
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
4-{[(butan-2-yl)(pyridin-4-ylmethyl)amino]methyl}-2-chlorophenol
2-methoxy-1-[1'-(3,3,3-trifluoro-2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
2-[(3R,4S)-3-(3-hydroxypropyl)-4-(4-methylpiperazin-1-yl)piperidine-1-carbonyl]-6-methoxyphenol
4-[4-(4-ethyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]-4-oxo-N-(1,3,4-thiadiazol-2-yl)butanamide
7-(2-methylphenyl)-4-(oxane-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol