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N-[(2R,3R)-1'-[3-(4-methylphenyl)propanoyl]-2-(pyridin-2-ylmethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetamide
3-({2-amino-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridin-5-yl}methyl)-3-hydroxy-1-(2-phenylethyl)piperidin-2-one
1-(2-phenylethyl)-8-(3-phenylpropyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N,5-dimethyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
4-{3-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]phenyl}morpholine
{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)(oxolan-2-ylmethyl)amine
5-methanesulfonyl-2-methyl-N-[(4-methyl-1,4-oxazepan-6-yl)methyl]pyrimidin-4-amine
2-benzyl-8-[3-(2-methyl-1H-imidazol-1-yl)propanoyl]-2,8-diazaspiro[4.5]decan-3-one
1-[benzyl(methyl)amino]-3-[4-({[2-(pyridin-2-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
2-[3-(3-fluorophenyl)-1-methyl-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-{[2-(trifluoromethyl)phenyl]methyl}acetamide
(2S,4S)-N-{2-azatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-5-yl}-1-(9H-fluoren-2-ylmethyl)-4-(pyrimidin-2-ylsulfanyl)pyrrolidine-2-carboxamide
N-methyl-N-(2-phenyl-1-{1-[(2E)-3-(pyridin-2-yl)prop-2-enoyl]piperidin-4-yl}ethyl)thiophene-2-carboxamide
3-[5-(butoxymethyl)-1,2,4-oxadiazol-3-yl]-6-methylpyridazine
3-[(3S,7S,8aS)-3-ethyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(4-ethylphenyl)urea
2-methoxy-N-[(2R,3R)-2-methoxy-1'-[2-(1H-1,2,4-triazol-1-yl)acetyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]benzamide
4-(2,4-dioxoimidazolidin-1-yl)-N-methyl-N-[1-(pyridin-3-yl)propyl]benzamide
1-{1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-5-fluoro-2-[(2-methoxyphenyl)methyl]-1H-1,3-benzodiazole
1-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}-4-(pyridin-2-ylmethyl)-1,4-diazepane
N-{[5-(2-acetylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-4-(4-methylpiperazin-1-yl)benzamide
3-(2-oxo-2-{2-oxo-3-phenyl-1,8-diazaspiro[4.5]decan-8-yl}ethyl)imidazolidine-2,4-dione
{[3-(1-benzofuran-2-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]methylamine
2-ethyl-4-(4-ethyl-2-methyl-1,3-thiazole-5-carbonyl)-1-(propan-2-yl)piperazine
{[6-chloro-2-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}[(1,5-dimethyl-1H-pyrazol-3-yl)methyl]amine
(3aS,7aR)-5-methyl-2-{[2-(thiophen-2-yl)pyrimidin-5-yl]methyl}-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
3-amino-1-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}pyrrolidine-3-carboxylic acid
(furan-2-ylmethyl)({[2-(4-methoxynaphthalen-1-yl)-5-methyl-1,3-oxazol-4-yl]methyl})(prop-2-yn-1-yl)amine
1-(2-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}-2-oxoethyl)-1,2-dihydropyridin-2-one
N-{[5-(2-acetylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-5-propyl-1,2-oxazole-3-carboxamide
2-(4-chloro-1-methyl-1H-pyrrole-2-carbonyl)-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
4-[2-(5-methylfuran-2-yl)propyl]-1-[2-(1H-pyrazol-1-yl)ethyl]-1H-1,2,3-triazole
2-({5-cyclopropyl-4-[2-(trifluoromethyl)phenyl]-4H-1,2,4-triazol-3-yl}sulfanyl)acetic acid
1-(2,2-dimethylpropyl)-3-hydroxy-3-{1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-ylmethyl}piperidin-2-one
7-(5-chloro-2-methoxyphenyl)-4-[(4-ethoxyphenyl)methyl]-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-[1-(2H-1,3-benzodioxol-5-yl)-3-[hydroxy(phenyl)methyl]-1H-1,2,4-triazol-5-yl]propanamide
1-benzyl-8-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[4-(1H-1,3-benzodiazol-2-yl)phenyl]-1-(furan-3-ylmethyl)piperidine-4-carboxamide
6-[1-(2-chlorophenyl)ethyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
4-hydroxy-N-(2-methoxyethyl)-2-phenyl-N-(pyridin-4-ylmethyl)pyrimidine-5-carboxamide
4-(furan-2-carbonyl)-7-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
6-(2-butyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-5H-[1,3]thiazolo[3,2-a]pyrimidin-5-one
3-[2-(hydroxymethyl)-1H-1,3-benzodiazol-1-yl]-1-(2-phenylpyrrolidin-1-yl)propan-1-one
[2-(1H-1,3-benzodiazol-2-yl)ethyl](1-phenoxypropan-2-yl)amine
N-[1-(4-methanesulfonylphenyl)propyl]imidazo[2,1-b][1,3]thiazole-6-carboxamide
N-[1-(pyrrolidine-1-carbonyl)piperidin-4-yl]-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
2-(2,5-dioxoimidazolidin-1-yl)-N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}acetamide
N-{[8-(naphthalen-2-ylmethyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}furan-2-carboxamide
1-(4-methanesulfonylphenyl)-3-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}urea
(4aS,7aR)-1-(1-methyl-5-phenyl-1H-pyrrole-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[3-(aminomethyl)pyrrolidin-1-yl]-2-{[(3,5-dimethylphenyl)methyl]sulfanyl}ethan-1-one
2-[(2,6-dimethylpyrimidin-4-yl)formamido]-N-(5-fluoro-2-methylphenyl)propanamide