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4-[2-(4-fluorophenyl)pyrrolidine-1-carbonyl]-3-methyl-1-propyl-1H-pyrazole
1-{7-oxo-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carbonyl}-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-{1-[4-hydroxy-4-(pyridin-2-yl)piperidin-1-yl]-1-oxobutan-2-yl}-2,3-dihydro-1H-isoindol-1-one
4-[(4-{5-[(2-methoxyethyl)sulfanyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)methyl]quinoline
2-{1-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]piperidin-4-yl}-1,3-benzoxazole
{[2-(azocane-1-carbonyl)-6-chloroimidazo[1,2-a]pyridin-3-yl]methyl}[(1-methyl-1H-pyrazol-4-yl)methyl]amine
N-(3,5-dimethoxyphenyl)-3-[1-(pyrrolidine-1-carbonyl)piperidin-3-yl]propanamide
3-({1-[(2-aminopyrimidin-5-yl)methyl]pyrrolidin-3-yl}methyl)-1-(4-fluorophenyl)urea
1-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-5-oxopyrrolidine-3-carboxylic acid
3-{[3-(1H-pyrazol-1-yl)phenyl]formamido}butanoic acid
2-[2-(benzyloxy)phenyl]-N-(4H-1,2,4-triazol-4-yl)acetamide
1-{1-[2-(2-chlorophenoxy)acetyl]piperidin-4-yl}-N,N-diethyl-1H-1,2,3-triazole-4-carboxamide
(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-6-(1,3-thiazole-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}(isoquinolin-5-ylmethyl)amine
2-{5-methyl-2-oxo-4-[2-(thiophen-3-yl)acetyl]piperazin-1-yl}benzonitrile
(2S)-1-[9-hydroxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
(2S,4R)-4-(2-ethoxyacetamido)-N-methyl-1-[(phenylcarbamoyl)methyl]pyrrolidine-2-carboxamide
1-{7-[(2,3-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}ethan-1-one
{1-[(3,5-dichloropyridin-4-yl)methyl]piperidin-4-yl}(pyridin-2-yl)methanol
2-[2-(2-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N-[1-(pyridin-3-yl)propan-2-yl]acetamide
3-[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]propanamide
N-(1-{1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-2-(2-fluorophenyl)ethyl)-N-methylthiophene-2-carboxamide
1-[2-(4-methylpentyl)morpholin-4-yl]-3-(1H-pyrazol-4-yl)propan-1-one
N-[(3S,4R)-1-(cyclopropylmethyl)-4-(4-methoxyphenyl)pyrrolidin-3-yl]acetamide
3-[(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)amino]-1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-1-one
N-[3-(1H-pyrazol-1-yl)propyl]-5-(3,4,5-trimethoxyphenyl)-1,2,4-triazin-3-amine
N-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}-4-(trifluoromethyl)pyrimidin-2-amine
N-[2-(azepane-1-carbonyl)phenyl]-2-(1H-indazol-3-yl)acetamide
1-(6-fluoro-2-oxo-1,2,3,4-tetrahydroquinolin-8-yl)-3-{1-oxaspiro[4.4]nonan-3-yl}urea
ethyl 1-(6,7-dimethoxy-3-{[(thiophen-3-ylmethyl)amino]methyl}quinolin-2-yl)piperidine-3-carboxylate
methyl 3-[4-({4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]piperidin-1-yl}methyl)-1H-pyrazol-1-yl]propanoate
9-methoxy-7-(3-methoxyphenyl)-4-[(2-methoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-[(2S)-2-[4-(4-chlorophenoxy)piperidine-1-carbonyl]pyrrolidin-1-yl]ethan-1-one
7-(2-methoxyacetamido)-1-methyl-2-(pyridin-3-yl)-N-{spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-5-ylmethyl}-1H-1,3-benzodiazole-5-carboxamide
4-[(2S)-1-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}pyrrolidine-2-carbonyl]morpholine
6-({pyrazolo[1,5-a]pyridin-3-ylmethyl}amino)-N-[3-(pyridin-2-yl)propyl]pyridine-3-carboxamide
N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-3-(4H-1,2,4-triazol-4-yl)benzamide
methyl (2S,4S)-4-(3-fluorobenzamido)-1-[(4-methoxy-2,5-dimethylphenyl)methyl]pyrrolidine-2-carboxylate
9-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-2-[(5-methylpyrazin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
N,1,4,6-tetramethyl-N-{[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
2-({[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}(methyl)amino)-2-[2-(methylsulfanyl)phenyl]acetic acid
4-[4-(1,3-dimethyl-1H-pyrazol-4-yl)pyrimidin-2-yl]-1-phenylpiperazin-2-one
N-(1-{7-[(4-fluoro-3-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)furan-3-carboxamide
1-methyl-8-{2-[methyl(phenyl)amino]acetyl}-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
3-(3-fluorophenyl)-4-{[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-2-one
N-(2H-1,3-benzodioxol-5-ylmethyl)-4-methyl-3-(2-oxoimidazolidin-1-yl)benzamide
N-{[3-methoxy-4-(oxolan-3-yloxy)phenyl]methyl}-N-(pyridin-3-ylmethyl)cyclopropanecarboxamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-[4-(methylamino)benzoyl]piperidin-3-ol
2-[2-(morpholin-4-yl)ethyl]-2,3-dihydro-1,2-benzothiazol-3-one
3-cyclopropyl-1-phenyl-5-{5-[(4H-1,2,4-triazol-3-ylsulfanyl)methyl]furan-2-yl}-1H-1,2,4-triazole