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6-[(2R,3R,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyridine-3-carbonitrile
1-[1-(2-hydroxy-5-methylbenzoyl)piperidin-3-yl]-N-(2-hydroxyethyl)-1H-1,2,3-triazole-4-carboxamide
3-[(3aS,6aS)-octahydropyrrolo[3,4-b]pyrrole-5-sulfonyl]-N-[(5-methyl-1,2-oxazol-3-yl)methyl]benzamide
dimethyl({4-[1-(6-methylpyridine-2-carbonyl)piperidin-2-yl]phenyl}methyl)amine
2-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-6-methylpyridine-3-carboxylic acid
4-{2-[4-(pyrimidin-4-yl)piperazin-1-yl]ethyl}morpholine
methyl (2S,4S,5R)-5-(3-chlorophenyl)-1-methyl-4-[(1,2-oxazol-3-ylmethyl)carbamoyl]pyrrolidine-2-carboxylate
N-[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]-N-methyl-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N-methyl-5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carboxamide
(2E)-3-(3,4-dimethoxyphenyl)-1-{4-[2-(oxolan-2-yl)-5-(trifluoromethyl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}prop-2-en-1-one
2-[4-(1H-indol-3-ylmethyl)-1-(thiophen-3-ylmethyl)piperazin-2-yl]ethan-1-ol
N-[(1R)-1-(4-methoxyphenyl)ethyl]-1,3-dimethyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-({1-[4-(1H-1,2,4-triazol-1-yl)butanoyl]pyrrolidin-3-yl}methyl)benzoic acid
9-(3-ethyl-1H-indole-2-carbonyl)-1,4-dimethyl-1,4,9-triazaspiro[5.5]undecane
1-[(3R,4R)-3-(hydroxymethyl)-4-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]-3-(2-methoxyphenyl)propan-1-one
3-({3-[2-(3-methoxyphenyl)ethyl]piperidin-1-yl}sulfonyl)pyridine
5-[4-methoxy-2-methyl-5-(propan-2-yl)phenyl]-1-methyl-1H,4H-pyrazolo[3,4-d]imidazole
2-(2,3-dihydro-1H-inden-1-yl)-N-[1-(methoxymethyl)cyclopentyl]acetamide
N-(1-methyl-1H-pyrazol-5-yl)-2-[3-(thiophen-2-yl)-1H-pyrazol-1-yl]acetamide
3-methoxy-N-(1-{7-[2-(4-methoxyphenyl)acetyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)propanamide
[(3R,4R)-4-(azepan-1-ylmethyl)-1-[(3-chloro-2,6-difluorophenyl)methyl]pyrrolidin-3-yl]methanol
N-[2-(2,4-difluorophenyl)-1-{1-[(3-methoxyphenyl)methyl]piperidin-4-yl}ethyl]-N-methylfuran-2-carboxamide
1-ethyl-4-[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]pyrrolidin-2-one
1-(4-ethoxy-2-fluorophenyl)-3-{[1-(prop-2-en-1-yl)pyrrolidin-3-yl]methyl}urea
1-(2-chlorophenyl)-5-methyl-4-(1H-pyrrole-2-carbonyl)piperazin-2-one
N,N-diethyl-1-[6-(3-methoxyphenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]pyrrolidin-3-amine
2-[2-(hydroxymethyl)pyridin-4-yl]-N,N-bis(propan-2-yl)benzamide
4-[1-(2,2-dimethylpropyl)pyrrolidin-3-yl]-1-(5-methyl-1H-pyrazole-3-carbonyl)piperidine
N-(2-methoxy-2-methylpropyl)-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-3-carboxamide
{[3-(2-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}[2-(morpholin-4-yl)-2-(pyridin-4-yl)ethyl]amine
2-(1-ethylpiperidin-4-yl)-N-{2-hydroxy-2-[2-(trifluoromethyl)phenyl]ethyl}acetamide
N-[(4-ethylphenyl)methyl]-3-{5-[2-(2-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}-N-methylpropanamide
[(dimethyl-1,2-oxazol-4-yl)methyl][1-(1H-1,2,4-triazol-1-yl)propan-2-yl]amine
5-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-1,2-dihydropyridin-2-one
N-({8-[(2,3-difluorophenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)acetamide
N-{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]ethyl}-1-(4-fluorophenyl)cyclopropane-1-carboxamide
4-[1-({5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethyl]phenol
N-[(2S,4R,6S)-2-benzyl-6-(1-tert-butyl-3,5-dimethyl-1H-pyrazol-4-yl)oxan-4-yl]acetamide
N-(2-{5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(4-fluorophenyl)-4H-1,2,4-triazol-3-yl}ethyl)-3,4-dimethoxybenzamide
2-(2H-1,3-benzodioxol-5-yl)-N-({5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl}methyl)acetamide
1-(4-methyl-1,2,5-oxadiazole-3-carbonyl)-4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine
3-phenyl-N-[2-(3-phenylpyrrolidin-1-yl)ethyl]-1H-pyrazole-4-carboxamide
N-methyl-5-oxo-1-[4-(propan-2-yl)phenyl]-N-(pyrazin-2-ylmethyl)pyrrolidine-3-carboxamide
N-{[2-(2-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-1H-pyrazole-3-carboxamide
1-cyclohexyl-N-[2-hydroxy-2-(3-hydroxyphenyl)ethyl]piperidine-4-carboxamide
N-[3-(benzyloxy)phenyl]-4-(2-methoxyethyl)piperazine-1-carboxamide
1-[4-({[(3-fluorophenyl)methyl]amino}methyl)-2-methoxyphenoxy]-3-(pyrrolidin-1-yl)propan-2-ol
methyl 6-(2,3-dihydro-1-benzofuran-5-ylmethyl)-2-[methyl(2-methylpropyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
3-{[3-(2-methylpiperidin-1-yl)azetidin-1-yl]methyl}-7-(methylsulfanyl)-1,2-dihydroquinolin-2-one
2-(dimethylamino)-N,4-dimethyl-N-(quinolin-5-ylmethyl)pyrimidine-5-carboxamide