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N-benzyl-3-{1-[3-(3-methoxyphenyl)propanoyl]piperidin-4-yl}-N-methylpropanamide
5-[1-(1H-imidazol-1-ylmethyl)cyclopropyl]-3-(2-phenylethyl)-1H-1,2,4-triazole
4-({4-[2-(4-ethylpiperazin-1-yl)ethoxy]phenyl}methyl)morpholine
4-{4-[3-(2-chlorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}pyrimidin-2-amine
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-2-(1H-pyrazol-1-yl)benzamide
1-{[1-(5-chloropyridin-2-yl)-1H-pyrrol-2-yl]methyl}-4-(5-methyl-1,3,4-thiadiazol-2-yl)piperazine
2-(1-benzyl-3-oxopiperazin-2-yl)-N-[(4-phenyl-1,3-thiazol-5-yl)methyl]acetamide
5-{[2-(ethylsulfanyl)-1,3-thiazol-4-yl]methyl}-3-methyl-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazole
1-[3-(4-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]-2-methoxy-2-methylpropan-1-one
1-cyclobutanecarbonyl-4-(3-phenylbutyl)-1,4-diazepane
9-[2-(1H-pyrazol-1-yl)butanoyl]-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}isoquinoline
11-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]-7-methyl-3,7,11-triazaspiro[5.6]dodecane
N-[(3S)-2-oxoazepan-3-yl]-N-{[4-(pyridin-2-ylmethoxy)phenyl]methyl}thiophene-2-carboxamide
6-ethoxy-4-methyl-2-{4-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]piperidin-1-yl}quinazoline
1-[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
4-{[4-(2-methoxyphenoxy)piperidin-1-yl]methyl}-1,5-dimethyl-1H-pyrrole-2-carbonitrile
N-(1,4-dioxan-2-ylmethyl)-1-methyl-6-(2-phenylethyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-[4-({[3-(1H-imidazol-1-yl)propyl]amino}methyl)-2-methoxyphenoxy]-3-(morpholin-4-yl)propan-2-ol
4-[7-({methyl[2-(pyridin-2-yl)ethyl]amino}methyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl]pyrrolidin-2-one
1-{2-chloro-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-N-(2,3-dihydro-1,4-benzodioxin-6-yl)piperidin-3-amine
3-{2-[4-(5-chloropyridin-2-yl)piperazin-1-yl]-2-oxoethyl}-3-(2-fluorophenyl)-1-(2-methoxyethyl)pyrrolidine-2,5-dione
2-{2-[2-(dimethylamino)ethyl]-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}-5,6-dimethylpyridine-3-carbonitrile
1-[1-(3-aminothiophene-2-carbonyl)piperidin-4-yl]piperidin-4-ol
1-[3-(pyridin-2-ylmethoxy)piperidin-1-yl]-3-[5-(thiophen-3-yl)-1,3,4-oxadiazol-2-yl]propan-1-one
1-(1-{2-methylimidazo[1,2-a]pyridine-6-carbonyl}azetidin-3-yl)piperidine
4-[5-(3,4-difluorophenoxymethyl)-1,2-oxazole-3-carbonyl]thiomorpholine
1'-{[2-(2,3-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}spiro[indene-1,4'-piperidine]
2-amino-6-(1,3-dimethyl-1H-pyrazol-4-yl)-4-{4-[1-(dimethylamino)ethyl]phenyl}pyridine-3-carbonitrile
2-[(1-acetylpiperidin-4-yl)oxy]-5-chloro-N-(quinolin-3-ylmethyl)benzamide
7-[2,2-dimethyl-1-(thiophen-2-yl)cyclopropanecarbonyl]-2-methyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
5-cyclopropyl-N-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]-1,3,4-oxadiazol-2-amine
methyl 3-[(3S,4R)-1-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]-4-(dimethylamino)piperidin-3-yl]propanoate
1-(1,3-dihydro-2-benzofuran-5-yl)-3-{[1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]methyl}urea
N-[3-(1H-pyrazol-1-yl)phenyl]-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidine-3-carboxamide
N-[2-(2-oxopiperidin-1-yl)ethyl]-2-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
4-(2,5-dimethoxyphenyl)-2-({methyl[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]amino}methyl)phenol
methyl 3-(2-chlorobenzenesulfonamido)-5-[(cyclohexylformamido)methyl]benzoate
2-[(4-{[1-(dimethylsulfamoyl)piperidin-4-yl]oxy}phenyl)formamido]acetamide
1-[4-({3-[2-(3-methoxyphenyl)piperidine-1-carbonyl]-1,2-oxazol-5-yl}methoxy)phenyl]ethan-1-one
1-(2,3-dihydro-1H-inden-2-yl)-N-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]piperidin-3-amine
(5S,9aS,9bS)-2-[(3-chlorophenyl)methyl]-5-[(E)-2-(2-methoxyphenyl)ethenyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
2-(2,3-dimethylbenzamido)-N-[3-(morpholin-4-yl)propyl]-7-oxo-4,5,6,7-tetrahydro-1,3-benzothiazole-5-carboxamide
1-benzyl-N,N-dimethyl-5-{[(4-phenyl-1,3-thiazol-2-yl)methyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
(3aR,6aR)-2-acetyl-5-[6-(methoxymethyl)pyrimidin-4-yl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
7-chloro-3-[(ethylamino)methyl]-1-(2-phenoxyethyl)-1,2-dihydroquinolin-2-one
dimethyl({[(3S,4R)-4-(propan-2-yl)-1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}pyrrolidin-3-yl]sulfamoyl})amine
1-(2-methoxyacetyl)-N-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}piperidine-4-carboxamide
(2S)-4-methyl-2-{[3-oxo-4-(3-phenylpropyl)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-11-yl]amino}pentanamide
1-(3-{4-[(3-fluorophenyl)methyl]-3-oxopiperazin-1-yl}-3-oxopropyl)azepan-2-one