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3-[2-(4-benzyl-3-ethyl-5-oxo-1,4-diazepan-1-yl)-2-oxoethyl]imidazolidine-2,4-dione
3-(azepane-1-carbonyl)-5-[4-(3-chlorophenyl)piperazin-1-yl]-1-methyl-4,5,6,7-tetrahydro-1H-indazole
6-(2-chlorophenyl)-N-(2-methoxybutyl)-8-oxo-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
4-chloro-N-(furan-2-ylmethyl)-1-methyl-N-(pyridin-2-ylmethyl)-1H-pyrazole-3-carboxamide
4-cyano-N-[2-oxo-2-(piperazin-1-yl)ethyl]-1H-pyrrole-2-carboxamide
N-[4-(pyridin-3-yloxy)phenyl]-1-(thian-4-yl)piperidine-4-carboxamide
N-{2-azatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-5-yl}-3-(methoxymethyl)pyrrolidine-1-carboxamide
4-{2-[6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-2-oxoethyl}-1,2,3,6-tetrahydropyridazine-3,6-dione
4-[2-(dimethylamino)-2-(3-methylphenyl)acetyl]-1-(3-methoxyphenyl)piperazin-2-one
(3aS,6aS)-2-cyclobutanecarbonyl-5-[2-(4H-1,2,4-triazol-4-yl)ethyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
6-ethyl-N4,5-dimethyl-N4-(1,3-thiazol-2-ylmethyl)pyrimidine-2,4-diamine
4-[(3,4-difluorophenyl)methyl]-3-[2-(1,2-oxazolidin-2-yl)-2-oxoethyl]piperazin-2-one
7-(3-chlorophenyl)-4-[3-(4-methyl-1H-pyrazol-1-yl)propyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-(2-acetamidoethyl)acetamide
2-(2,3-dihydro-1,4-benzodioxin-6-yl)-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
7-(2-methoxyphenyl)-2-(5-methylpyrazin-2-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
3-({[(3-ethoxyphenyl)methyl](2-hydroxyethyl)amino}methyl)-4H-chromen-4-one
(3S,4R)-1-(6-chloro-2-methylquinoline-4-carbonyl)-4-methylpiperidine-3,4-diol
1-methyl-N-[(4-methylphenyl)methyl]-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-butyl-N-methyl-2-[1-(naphthalen-1-ylmethyl)-3-oxopiperazin-2-yl]acetamide
(2-methoxyethyl)({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)(oxolan-3-ylmethyl)amine
4-methoxy-3-{[1-(propan-2-yl)piperidin-4-yl]oxy}-N-[1-(pyridin-2-yl)propan-2-yl]benzamide
4,4-difluoro-N-(1H-indazol-4-yl)piperidine-1-carboxamide
1-[4-({4-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperazin-1-yl]ethan-1-one
methyl 1-methyl-5-({9-oxo-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}sulfonyl)-1H-pyrrole-2-carboxylate
2-{1-methyl-4-[(2,4,5-trimethylphenyl)methyl]piperazin-2-yl}ethan-1-ol
N-[4-({[(5-ethylpyridin-2-yl)methyl](methyl)carbamoyl}methoxy)phenyl]propanamide
N-[1-(methoxymethyl)cyclopentyl]-2-(morpholin-2-yl)acetamide
4-[2-oxo-2-(4-phenylazepan-1-yl)ethyl]-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-3-one
2-(2H-1,3-benzodioxol-5-ylmethyl)-4-(4-{[4-(trifluoromethoxy)phenyl]methyl}piperazin-1-yl)-2,3-dihydro-1H-isoindole-1,3-dione
5-(5-chloro-2-methoxyphenyl)-N,N-dimethylthiophene-2-carboxamide
7-{2-[(1-methyl-1H-indol-3-yl)sulfanyl]acetyl}-2,7-diazaspiro[4.4]nonane-1,3-dione
N-(1-{10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}piperidin-4-yl)methanesulfonamide
N-[(2-chlorophenyl)methyl]-3-{1-[3-(6-oxo-1,4,5,6-tetrahydropyridazin-3-yl)propanoyl]piperidin-3-yl}propanamide
N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]-2-(4-oxo-3,4-dihydrophthalazin-1-yl)propanamide
2-[(1R,3S)-1-hydroxy-3-methoxy-7-azaspiro[3.5]nonan-7-yl]-1,3-thiazole-4-carboxamide
5-methyl-3-(5-{[1,2,4]triazolo[1,5-a]pyrimidine-2-carbonyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl)-1,2-oxazole
1-[(2R,3S,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(methylsulfanyl)ethan-1-one
1-(4-acetyl-4-phenylpiperidin-1-yl)-2-(3-fluoro-4-hydroxyphenyl)ethan-1-one
(1R,3S)-7-[1-(methoxymethyl)cyclobutanecarbonyl]-7-azaspiro[3.5]nonane-1,3-diol
2-[(3,4-dimethoxyphenyl)methyl]-N-(2-methoxyethyl)-N-methyl-1,3-benzoxazole-6-carboxamide
1-(4-{[(5-methyl-1,2-oxazol-3-yl)methyl]amino}-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
2-(4-acetyl-1,4-diazepan-1-yl)-2-(2,3-dimethylphenyl)acetic acid
2-(cyclopropylmethyl)-7-[3-(1-methylpiperidin-3-yl)propanoyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
4-[(7-methyl-2-oxo-1,2-dihydroquinolin-3-yl)methyl]piperazine-1-carboxamide
4-[(2Z)-5-methyl-2-phenylhex-2-en-1-yl]-1,8-dioxa-4,11-diazaspiro[5.6]dodecane
N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N,4,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
N-(2-chlorophenyl)-3-(1-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-4-yl)propanamide
(2R,3R)-3-{methyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-2-{3-oxo-1-[(4-phenylphenyl)methyl]piperazin-2-yl}acetamide