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3-methoxy-N-(oxolan-2-ylmethyl)-N-({3-[2-(thiophen-2-yl)ethoxy]phenyl}methyl)benzamide
2-(1-cyclopentyl-3-oxopiperazin-2-yl)-N-[(3-methylphenyl)methyl]acetamide
(2S)-N2-[(2,4-dichloro-6-methylphenyl)methyl]pyrrolidine-1,2-dicarboxamide
2-[1-(3-methyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]-1,2,3,4-tetrahydroisoquinoline
5-[(2-fluorophenyl)methyl]-5-(1-{[2-(prop-2-en-1-yloxy)phenyl]methyl}piperidin-4-yl)imidazolidine-2,4-dione
3-{3-oxo-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-8-yl}propanoic acid
1-[(4-methyl-1H-imidazol-5-yl)methyl]-3-(2-phenylethyl)piperidine
N-[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
(2R)-3-phenyl-2-(4H-1,2,4-triazol-4-yl)propan-1-ol
2-[(1-cyclopentylpiperidin-4-yl)oxy]-N-[2-(diethylamino)ethyl]-5-methoxybenzamide
1-cyclopentanecarbonyl-N-[(4,6-dimethylpyridin-3-yl)methyl]piperidine-4-carboxamide
1-{5-[1-ethyl-3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]-2-methylphenyl}imidazolidin-2-one
1-(2-{2-amino-4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}-2-oxoethyl)-4-phenylpyrrolidin-2-one
4-{[2-(2-methoxyphenyl)pyrrolidin-1-yl]methyl}-5-methyl-2-[4-(methylsulfanyl)phenyl]-1,3-oxazole
(4aR,7aS)-1-methanesulfonyl-4-[3-(pyridin-4-yl)propanoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-{1-[1-(2,5-dimethylfuran-3-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-1-(2-methoxyphenyl)urea
N-(2,3-dihydro-1-benzofuran-2-ylmethyl)-N-methyl-5-propyl-1,3,4-oxadiazole-2-carboxamide
1-(3-methoxypropyl)-3-(pyridin-2-ylmethyl)-8-(pyridin-4-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[(dimethyl-1,3-thiazol-2-yl)methyl]-3-{5-[2-(4-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}propanamide
(3R,4R)-4-cyclopropyl-N-[2-(2-fluorophenyl)ethyl]-4-hydroxy-3-methylpiperidine-1-carboxamide
N-(3-chloro-2-methylphenyl)-2-[4-(pyrrolidine-1-carbonyl)morpholin-3-yl]acetamide
N-{1-[(3-methoxyphenyl)methyl]piperidin-3-yl}-2-[4-(methylsulfanyl)phenyl]acetamide
1-(2-methoxyacetyl)-3-(3-methoxypropyl)piperidine-3-carboxylic acid
2-(dimethylamino)-2-(3-fluorophenyl)-N-[2-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]acetamide
4-(4-chlorophenoxy)-1-(1,3-thiazol-4-ylmethyl)piperidine
2-{3-[2-(3-fluorophenyl)ethyl]piperidin-1-yl}-5-(piperidine-1-carbonyl)pyridine
2-methyl-2-({1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidin-3-yl}formamido)propanamide
1-(cyclopropylmethyl)-5-[(3-ethoxy-4-methoxyphenyl)methyl]-N-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-ethyl-5-methyl-N-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}-1H-pyrazole-3-carboxamide
1-(2,5-dimethylbenzoyl)-4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
1-{2-[4-(2-methylphenoxy)piperidin-1-yl]-2-oxoethyl}piperidine-4-carboxamide
2-(2,3-dimethoxy-5-methylphenyl)-5-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]pyridine
N-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1H-1,2,3-triazole-5-carboxamide
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-1-[2-(trifluoromethyl)morpholin-4-yl]ethan-1-one
methyl({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)[(2,3,6-trifluorophenyl)methyl]amine
(1S,5R)-6-methyl-3-{[5-(1-methyl-1H-1,3-benzodiazol-2-yl)furan-2-yl]methyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}cyclopentanecarboxamide
2-(furan-2-carbonyl)-6-methyl-5-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridine
2-{1-[(4-chloro-3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(3-methoxyphenyl)ethyl]acetamide
2-{4-[(6-fluoro-4-hydroxyquinolin-2-yl)methyl]piperazin-1-yl}pyridine-3-carboxamide
3-(2-methylpropyl)-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]-1,2-oxazole-5-carboxamide
4-[(2-ethyl-1H-imidazol-1-yl)methyl]-2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazole
1-[(2-fluorophenyl)methyl]-N-[1-(1H-indol-5-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
ethyl 4-[2-(7-chloro-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetamido]piperidine-1-carboxylate
N-butyl-5-{1-[2-(dimethyl-1,2-oxazol-4-yl)acetyl]pyrrolidin-2-yl}thiophene-2-carboxamide
ethyl 4-{[1-(1,3-benzothiazol-2-yl)piperidin-3-yl]amino}piperidine-1-carboxylate
4-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-N,N-dimethyl-4-oxobutanamide
4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]piperidine
2-[4-(3-hydroxypiperidin-1-yl)piperidin-1-yl]-6-(trifluoromethyl)pyridine-3-carboxamide
N-[4-(morpholin-4-yl)-1-(2,2,2-trifluoroethyl)-1H-indazol-3-yl]-1,3-thiazole-4-carboxamide