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[(3R,4R)-4-{[ethyl(methyl)amino]methyl}-1-{[2-(4-methoxyphenyl)pyrimidin-5-yl]methyl}pyrrolidin-3-yl]methanol
2-(pyridin-4-yl)-N-[2-(1,3-thiazol-4-yl)ethyl]quinoline-4-carboxamide
3-(2,3-dichlorophenyl)-2-methyl-6-(4H-1,2,4-triazol-4-yl)pyridine
2-(propan-2-yloxy)-N-[(3R,4S)-4-propyl-1-(1,3-thiazol-2-yl)pyrrolidin-3-yl]acetamide
N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}methanesulfonamide
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-N,1,3-trimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
N-(3-methylphenyl)-3-[1-(pyridine-3-carbonyl)piperidin-4-yl]propanamide
3-(5-{[2-(pyrrolidin-1-ylmethyl)piperidin-1-yl]methyl}thiophen-2-yl)prop-2-yn-1-ol
7-[(5-fluoro-3-methyl-1H-indol-2-yl)methyl]-2,7-diazaspiro[4.5]decane
1-[3-(2H-1,3-benzodioxole-5-carbonyl)piperidin-1-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
(2S,4R)-4-(3-chlorobenzamido)-N-ethyl-1-(1H-imidazol-2-ylmethyl)pyrrolidine-2-carboxamide
4-{[(3S)-1-benzylpyrrolidin-3-yl]carbamoyl}-3,5-dimethyl-1H-pyrrole-2-carboxylic acid
(1R,3S,5S)-8-[2-methyl-6-(piperidin-4-yl)pyrimidin-4-yl]-8-azabicyclo[3.2.1]octan-3-ol
1-(1-acetylpiperidin-4-yl)-4-methanesulfonyl-1,4-diazepane-6-carboxylic acid
2-ethoxy-4-({methyl[(3-methylpyridin-4-yl)methyl]amino}methyl)phenol
2-benzyl-9-[(1-ethyl-1H-pyrazol-3-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
(1S,5R)-3-acetyl-N-(5-chloro-2-methoxyphenyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
2-(4-methanesulfonylphenyl)-1-(3-phenylpropyl)-1H-imidazole
{4-[(3-methoxyphenyl)methyl]-1-[6-(1-methyl-1H-imidazol-2-yl)pyridazin-3-yl]piperidin-4-yl}methanol
2-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}-5-(pyrrolidine-1-carbonyl)pyridine
2-(4-chlorophenyl)-7-methoxy-3-[(4-methyl-1,4-diazepan-1-yl)methyl]quinoline
1-[3-(hydroxymethyl)-3-(2-methoxyethyl)piperidin-1-yl]-3-(4H-1,2,4-triazol-4-yl)propan-1-one
(5-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}furan-2-yl)methanol
2-methyl-4-(2-methylphenyl)-1-[3-(thiophen-2-yl)-1H-pyrazole-4-carbonyl]piperazine
8-(1H-imidazol-2-ylmethyl)-2-(3-methylbut-2-en-1-yl)-2,8-diazaspiro[4.5]decan-3-one
N-[2-(3-methoxyphenoxy)ethyl]-N-methyl-2-(2-oxopiperidin-1-yl)acetamide
(3S,4S)-4-cyclopropyl-1-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}pyrrolidine-3-carboxylic acid
N,2,6-trimethyl-N-[(5-methyl-1H-1,3-benzodiazol-2-yl)methyl]pyrimidine-4-carboxamide
N-{[5-(dimethylcarbamoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-2-methylimidazo[1,2-a]pyrimidine-3-carboxamide
1-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
2-[(1-{5,6-dimethylthieno[2,3-d]pyrimidin-4-yl}piperidin-4-yl)amino]-1-(furan-2-yl)ethan-1-ol
2-{benzyl[5-(2,6-dimethoxyphenyl)-1,2,4-triazin-3-yl]amino}ethan-1-ol
4-(1-benzoxepine-4-carbonyl)-2-(4-fluorophenyl)morpholine
N-[3-({[(5-chloro-2-hydroxyphenyl)methyl]amino}methyl)-5-(piperidine-1-carbonyl)phenyl]methanesulfonamide
5-cyclopropyl-1-[1-(2-methoxyphenoxy)propan-2-yl]-4-phenyl-1H-imidazole
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-2-(methoxymethyl)-1-methyl-5-(2-phenylacetamido)-1H-1,3-benzodiazole-7-carboxamide
[(2R)-1-(1-benzofuran-3-carbonyl)pyrrolidin-2-yl]methanol
(5S)-5-({[(5-acetylthiophen-3-yl)methyl](pyridin-4-ylmethyl)amino}methyl)pyrrolidin-2-one
N-[2-(cyclohex-1-en-1-yl)ethyl]-6-[3-(pyridin-3-yl)propanoyl]-6-azaspiro[2.5]octane-1-carboxamide
1-[2-(dimethylamino)-2-(5-methylfuran-2-yl)ethyl]-3-(3-methyl-1,2,4-thiadiazol-5-yl)urea
(4aS,7aR)-1-{3-[4-(dimethylamino)phenyl]propanoyl}-4-ethyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-cyclopropyl-3-[4-(4-methoxyphenyl)piperazine-1-carbonyl]-6-methyl-1-(thiophen-2-ylmethyl)-1,4-dihydropyridin-4-one
N-[(3S,4R)-4-(4-methoxyphenyl)-1-[(2-methoxyphenyl)methyl]pyrrolidin-3-yl]acetamide
6-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]-1,2,3,4-tetrahydroquinoxaline-2,3-dione
2-[methyl({5-[4-(pyrimidin-2-yl)-1,4-diazepane-1-carbonyl]pyridin-2-yl})amino]ethan-1-ol
6-(2,6-dimethoxypyridin-3-yl)-4-(4-methylpiperazin-1-yl)quinazoline
(1S,5R)-6-(2-methoxyethyl)-3-[(3-methyl-1,2-oxazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
2-({6-[3-(methylsulfanyl)phenyl]pyridazin-3-yl}amino)ethan-1-ol
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-[3-(dimethylamino)propyl]-N-methylacetamide
(4aS,7aR)-1-(3-hydroxy-2-methylbenzoyl)-4-(pyrimidin-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione