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(3R,4S)-3,4-dimethyl-1-[3-(pyridin-2-yl)-1H-pyrazole-5-carbonyl]piperidin-4-ol
1-{1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]piperidin-3-yl}-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
N-ethyl-N-[(3S,4R)-4-hydroxyoxolan-3-yl]-3-methyl-5-propyl-1-benzofuran-2-carboxamide
methyl 5-{[1-(2-fluorophenyl)propan-2-yl]amino}-3-(furan-2-amido)-1-methyl-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-phenyl-4-[2-(propylsulfanyl)acetyl]piperazin-2-one
(3S,4R)-1-[2-(azepan-1-yl)-2-oxoethyl]-4-(4-fluorophenyl)pyrrolidine-3-carboxylic acid
6-({methyl[1-(1,3-thiazol-2-yl)ethyl]amino}methyl)pyridine-2-carboxylic acid
1-(5-methoxyfuran-2-carbonyl)-N-[2-(pyridin-3-yloxy)phenyl]pyrrolidine-2-carboxamide
3-[5-(4-phenylbutyl)-1,3,4-oxadiazol-2-yl]-1-(thiomorpholin-4-yl)propan-1-one
3-({2H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}(methyl)amino)-1-(1,2,3,4-tetrahydroquinolin-1-yl)propan-1-one
6-[(dimethyl-1,3-thiazol-5-yl)methyl]-2,5-dioxo-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
(1S,2S)-2-{4-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperazin-1-yl}cyclohexan-1-ol
1-[3-(4-chloro-2-methylbenzoyl)piperidin-1-yl]-3-(2-methyl-1H-1,3-benzodiazol-1-yl)propan-1-one
1-[(2,5-dimethoxyphenyl)methyl]-3-(3-fluoro-4-methoxybenzoyl)piperidine
N-[1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-3,4,7-trimethyl-1H-indole-2-carboxamide
6-(piperazin-1-yl)-N-[(3-propyl-1,2-oxazol-5-yl)methyl]pyridine-3-carboxamide
(2R)-2-amino-4-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-(2-methylpropyl)pentanamide
2-{3-[3-(3,6-dimethylpyrazin-2-yl)phenyl]-1H-pyrazol-1-yl}ethan-1-ol
1-[4-(dimethylamino)-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-(2-methoxyethoxy)ethan-1-one
1-[1-(1-cyclopropylethyl)-3-methyl-1H-pyrazol-5-yl]-3-[3-(methylsulfanyl)propyl]urea
2-chloro-4-({3-[(3-fluorophenyl)amino]piperidin-1-yl}methyl)-6-methoxyphenol
1-{3-[4-(benzyloxy)piperidin-1-yl]-3-oxopropyl}-6-methyl-1,2-dihydropyridin-2-one
methyl (2S,4S,5R)-1,2-dimethyl-5-(2-methylphenyl)-4-[(2-methylpropyl)carbamoyl]pyrrolidine-2-carboxylate
6-{3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidine-1-carbonyl}-2,2-dimethyl-3,4-dihydro-2H-pyran-4-one
N-{5H,6H,7H-cyclopenta[b]pyridin-3-ylmethyl}-3-(1H-pyrazol-1-ylmethyl)benzamide
methyl 4-(4-{[3-(3-fluorophenoxymethyl)piperidin-1-yl]methyl}-5-methyl-1,3-oxazol-2-yl)benzoate
N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)-2-(1H-pyrazol-1-yl)butanamide
2,3-dimethyl-N-[2-methyl-5-(2-oxopyrrolidin-1-yl)phenyl]-4-oxo-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carboxamide
N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]-1-{6-methylthieno[2,3-d]pyrimidin-4-yl}piperidin-4-amine
N-[(3R,4S)-4-cyclopropyl-1-[4-methyl-6-(methylamino)pyrimidin-2-yl]pyrrolidin-3-yl]oxane-4-carboxamide
1-cyclohexyl-3-methyl-5-[2-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-1H-1,2,4-triazole
2-({1-[(2-fluorophenyl)methyl]-2-(propane-2-sulfonyl)-1H-imidazol-5-yl}methyl)-1,2-oxazinane
methyl 1-[5-(2,4-difluorophenoxymethyl)-1,2-oxazole-3-carbonyl]piperidine-4-carboxylate
N-{[4-(3-methoxyphenyl)-5-[(2-phenylethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}pyridine-2-carboxamide
7-fluoro-N-(1H-imidazol-2-ylmethyl)-N,3-dimethyl-1-benzofuran-2-carboxamide
7-(3-cyclohexyl-1H-pyrazole-4-carbonyl)-2,7-diazaspiro[4.4]nonane-1,3-dione
5-[4-(2-chlorophenyl)piperazine-1-carbonyl]-1-cyclohexyl-N-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
(1R,5R)-6-benzyl-3-[1-(difluoromethyl)-1H-pyrazole-3-carbonyl]-3,6-diazabicyclo[3.2.2]nonane
6-(4-fluorophenyl)-2-[(1S,5R)-6-methyl-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]pyridine-3-carboxylic acid
2-cyclopropyl-4-hydroxy-N-[(4-sulfamoylphenyl)methyl]pyrimidine-5-carboxamide
1-{[3-(3-fluorophenyl)oxolan-3-yl]methyl}-4-(2-methylpyridin-4-yl)-1,4-diazepane
1-(2-methyl-4-phenylpyridine-3-carbonyl)-4-(3-methylpyridin-2-yl)piperazine
(2S)-1-[4-phenyl-5-(4-phenyl-1,3-thiazol-2-yl)-1H-imidazol-1-yl]propan-2-ol
6-[2-(methylsulfanyl)acetyl]-N-(3-phenylpropyl)-6-azaspiro[2.5]octane-1-carboxamide
1-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-3-methoxypropan-1-one
3-chloro-6-{4-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]piperazin-1-yl}pyridine-2-carboxylic acid
2-[3-({methyl[2-(1H-pyrazol-4-yl)ethyl]amino}methyl)phenyl]-6-phenyl-3,4-dihydropyrimidin-4-one
N-[2-(2-methoxyphenyl)ethyl]-3-(2-phenylethyl)-4,5-dihydro-1,2-oxazole-5-carboxamide
1-(4-methylpiperazin-1-yl)-3-[1-(2-methylquinolin-4-yl)piperidin-3-yl]propan-1-one
1-(5-methyl-2-{[1-(pyridin-4-ylmethyl)piperidin-4-yl]oxy}benzoyl)azetidin-3-ol