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4-[5-chloro-2-(piperidine-1-carbonyl)phenoxy]-1-[3-(1H-pyrazol-1-yl)propyl]piperidine
1-(3-ethoxypropanoyl)-4-(2-methoxyphenoxy)piperidine-4-carboxylic acid
[2-(4-methoxyphenyl)ethyl][(1-methylpiperidin-4-yl)methyl](4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)amine
1-[(3R,4R)-3-hydroxy-4-methyl-3-(propan-2-yl)pyrrolidin-1-yl]-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
propyl 4-(4-ethyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidine-1-carboxylate
methyl 1-[(4-{[(3,4-dimethoxyphenyl)methyl](methyl)amino}quinazolin-2-yl)methyl]piperidine-2-carboxylate
3-[(3S,7S,8aS)-1,4-dioxo-3-(propan-2-yl)-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(2,4-dichlorophenyl)urea
N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-2-(pyridin-3-yl)pyrimidine-5-carboxamide
8-[(3-chloro-4-hydroxyphenyl)methyl]-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-(4-{[5-(methoxymethyl)furan-2-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)-2-phenylethan-1-ol
N-methyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}-3-(trimethyl-1H-pyrazol-1-yl)propanamide
1-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carbonyl]-1H,2H,3H,4H,6H,10bH-pyrimido[2,1-a]isoindol-6-one
3-chloro-N-{2-[3-({methyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)phenoxy]propyl}benzamide
3-(2H-1,3-benzodioxole-5-carbonyl)-1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]piperidine
7-(2-cyclopentyl-2-phenylacetyl)-2-methyl-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
(2S,4R)-N-methyl-4-(4-{[methyl(phenylcarbamoyl)amino]methyl}-1H-1,2,3-triazol-1-yl)pyrrolidine-2-carboxamide
2-methyl-3-(2-{[4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-yl]amino}ethyl)-1H-indole-5-carbonitrile
(3R,4S)-4-phenyl-1-[5-(piperidine-1-carbonyl)pyridin-2-yl]pyrrolidin-3-amine
3-(furan-2-ylmethyl)-3-(3-methylbutan-2-yl)-1-[3-(4H-1,2,4-triazol-4-yl)phenyl]urea
5-fluoro-2-(1-{[3-(2-phenylethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-2-yl)-1H-1,3-benzodiazole
2-{2-[4-(pyridin-3-yl)-4H-1,2,4-triazol-3-yl]ethyl}phenol
N-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}-2-oxo-1,2-dihydroquinoline-4-carboxamide
4-(1H-imidazol-1-ylmethyl)-2-(4-methoxynaphthalen-1-yl)-5-methyl-1,3-oxazole
4-{[(3R,4R)-4-(azepan-1-yl)-3-hydroxypiperidin-1-yl]methyl}-1,5-dimethyl-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
8-acetyl-2-[(2-ethyl-1,3-thiazol-4-yl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-(adamantan-1-yl)-4-hydroxy-N-(2-hydroxybutyl)pyrimidine-5-carboxamide
2-(1-ethyl-8-{[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]methyl}-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-3-yl)acetamide
[(5-chlorothiophen-2-yl)methyl](2-methoxyethyl)({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)amine
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N'-(2-ethoxyphenyl)propanediamide
8-(1-cyclopropyl-5-oxopyrrolidine-3-carbonyl)-2-(3-methoxypropyl)-2,8-diazaspiro[4.5]decan-3-one
N-{1-[2-(3-chlorophenyl)ethyl]-5-oxopyrrolidin-3-yl}acetamide
[3-(prop-2-en-1-yl)-1-(pyridine-3-carbonyl)piperidin-3-yl]methanol
N-[(4,6-dimethylpyridin-2-yl)methyl]-N-methyl-2-(1-methylpiperidin-2-yl)acetamide
2-{2-[(pyridin-3-ylmethyl)amino]pyrimidin-4-yl}pyridine-4-carboxylic acid
1-[1-(2-methylbenzoyl)piperidin-3-yl]-4-[3-(trifluoromethyl)phenyl]piperazine
5-(2-chloro-4-fluorophenoxymethyl)-N-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-1,2-oxazole-3-carboxamide
dimethyl({[4-(1H-1,2,4-triazole-5-carbonyl)-1,4-oxazepan-6-yl]methyl})amine
N-{4-[3-(3,4-dimethyl-1H-pyrazol-5-yl)propanamido]-2-methylphenyl}-2,2-dimethylpropanamide
2-[3-(2-{[(3,4-difluorophenyl)methyl]carbamoyl}ethyl)piperidin-1-yl]pyridine-3-carboxamide
2-{4-[4-(cyclopropylcarbamoyl)piperidin-1-yl]piperidin-1-yl}pyridine-3-carboxamide
3-(2-phenylpropyl)-8-(1H-pyrrole-2-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
5-[3-(2-chlorophenyl)pyrrolidine-1-carbonyl]-3-[(4-methoxyphenyl)methyl]-1,2-oxazole
N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-N-(pyridin-2-ylmethyl)-5-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
methyl (2S)-2-[(2,6-dimethylquinolin-4-yl)formamido]-3-(1H-imidazol-4-yl)propanoate
5-propyl-5-{1-[4-(1H-1,2,4-triazol-1-yl)butanoyl]piperidin-4-yl}imidazolidine-2,4-dione
N-[4-(2-fluorophenoxy)phenyl]-1-[(4-methoxyphenyl)methyl]piperidine-4-carboxamide
(4R)-N,3-dimethyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-1,3-thiazolidine-4-carboxamide
7-[4-(2-phenylethyl)piperazine-1-carbonyl]-1,3-diazepane-2,4-dione
5-[2-methyl-4-(2-methylphenyl)piperazine-1-carbonyl]-2-(methylsulfanyl)pyrimidine
2-[4-(2,1,3-benzothiadiazol-5-ylmethyl)-1-[(3,5-dimethoxyphenyl)methyl]piperazin-2-yl]ethan-1-ol