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{[2-(azocane-1-carbonyl)-6-chloroimidazo[1,2-a]pyridin-3-yl]methyl}[3-(2-methyl-1H-imidazol-1-yl)propyl]amine
1-ethyl-N-{3-[(3-methoxyphenyl)carbamoyl]phenyl}piperidine-2-carboxamide
2-[2-(pyridin-2-yl)ethyl]-9-(pyrimidin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-(1,3-benzothiazol-6-yl)-3-[3-(trimethyl-1H-pyrazol-1-yl)propyl]urea
1-(4-acetyl-1,4-diazepan-1-yl)-2-(dimethylamino)-2-(3-fluorophenyl)ethan-1-one
2-{5-[2-(1H-1,3-benzodiazol-1-yl)ethyl]-1-(2-phenylethyl)-1H-1,2,4-triazol-3-yl}acetamide
methyl 3-[(2H-1,3-benzodioxol-5-ylformamido)methyl]-5-cyclohexaneamidobenzoate
1-(3-chlorophenyl)-4-[(2R)-2-hydroxy-3-methylbutanoyl]piperazin-2-one
[(2-fluoro-5-methylphenyl)methyl](methyl)[(1-methylpiperidin-2-yl)methyl]amine
1-({4-methyl-5-[1-(3,3,3-trifluoropropyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)piperidin-4-ol
2-[(2,4-difluorophenyl)methyl]-1H,2H-pyrrolo[1,2-d][1,2,4]triazin-1-one
N-[cyclopropyl(4-methylpyridin-2-yl)methyl]-2-methyl-1,3-benzothiazole-6-carboxamide
5-(hydroxymethyl)-2-methyl-4-{[2-methyl-4-(2-methylphenyl)piperazin-1-yl]methyl}pyridin-3-ol
N-(2-{7-[(2-hydroxy-5-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-methylpropanamide
3-{5-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
5-[1-(1-propylpiperidin-4-yl)pyrrolidin-2-yl]-N-(1H-pyrazol-3-yl)thiophene-2-carboxamide
3-ethyl-5-[1-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)pyrrolidin-2-yl]-1,2,4-oxadiazole
5-{2-methylimidazo[1,2-a]pyrimidin-3-yl}-3-(thiophen-3-ylmethyl)-1,2,4-oxadiazole
1-(2-benzyl-1,3-thiazole-4-carbonyl)azetidine-2-carboxylic acid
1-(4-{[4-(3-ethynylbenzoyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}piperazin-1-yl)ethan-1-one
4-{6-[(2-methoxyethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}benzoic acid
4-[2-(5-methylfuran-2-yl)phenyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
1-({3-[(3,4-dimethoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-4-(2-methoxyethyl)piperazine
1-(4-{7-chloro-3-[(cyclopentylamino)methyl]quinolin-2-yl}piperazin-1-yl)ethan-1-one
methyl 5-(cyclopentylamino)-1-(2-methylpropyl)-3-(2-phenylacetamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
3-(azocan-1-yl)-N-[2-(pyridin-2-yl)ethyl]propanamide
3-{1-[2-(2H-1,2,3-benzotriazol-2-yl)acetyl]piperidin-3-yl}-1-(4-methylpiperazin-1-yl)propan-1-one
8-(1-benzofuran-2-ylmethyl)-1-(2-methylpropyl)-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(furan-2-yl)-N,7-dimethyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-[(3,5-dimethoxyphenyl)methyl]-5-methyl-4-{[3-(morpholin-4-yl)propyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
4-[4-({4-[2-(1H-imidazol-1-yl)ethyl]piperazin-1-yl}methyl)phenyl]-2-methylbutan-2-ol
2-amino-4-(oxolan-3-yl)-6-(2,3,4-trimethoxyphenyl)pyridine-3-carbonitrile
N-{[2-(2,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-N-[(trimethyl-1H-pyrazol-4-yl)methyl]cyclopropanamine
methyl (1R,3R,3aR,6aS)-3-(2,2-dimethylpropyl)-1-(2-methoxy-2-oxoethyl)-5-methyl-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
N-benzyl-N-(cyclopropylmethyl)-2-[2,5-dioxo-3-phenyl-1-(pyridin-4-ylmethyl)pyrrolidin-3-yl]acetamide
1-(4-chlorophenyl)-5-methyl-4-[2-(2-methylphenoxy)acetyl]piperazin-2-one
N-[(2-methoxyphenyl)methyl]-5-methyl-N-(prop-2-en-1-yl)-1-propyl-1H-pyrazole-4-carboxamide
N-({1-[(2-cyanophenyl)methyl]pyrrolidin-3-yl}methyl)-2-methyl-2-(methylamino)propanamide
[(3R,4S)-4-[(4-methylpiperazin-1-yl)methyl]-1-{[3-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl]methanol
2-(2-methyl-1,3-thiazol-4-yl)-N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}acetamide
methyl (2S)-3-(4-hydroxyphenyl)-2-({9-oxo-1-azatricyclo[6.3.1.04,12]dodeca-4(12),5,7,10-tetraen-10-yl}formamido)propanoate
4-[5-chloro-2-(piperidine-1-carbonyl)phenoxy]-1-[(3,5-difluorophenyl)methyl]piperidine
2-methyl-8-[3-(trimethyl-1H-pyrazol-1-yl)propanoyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
4-hydroxy-1-(isoquinoline-5-carbonyl)piperidine-4-carboxylic acid
2-(3-methylbutyl)-8-[2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
3-[2-(1H-imidazol-1-yl)propyl]-1-{4-[(1-methylpiperidin-4-yl)oxy]phenyl}urea
(3aR,7aS)-5-methyl-2-(4-methyl-1H-imidazole-5-carbonyl)-2,3,3a,4,7,7a-hexahydro-1H-isoindole
8-[(2,3-difluorophenyl)methyl]-3-[(4-methoxyphenyl)methyl]-1-(3-methoxypropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(6R)-6-[4-(4-benzyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]-1,3-diazinane-2,4-dione
2-cyclopentyl-N-[1-(4-methylpyridin-2-yl)propyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine