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ethyl 4-{[1-(4-methylpyridin-2-yl)propyl]amino}piperidine-1-carboxylate
3-[5-(oxan-2-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]-1-(pyrrolidin-1-yl)propan-1-one
N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-3-(4-fluorophenyl)-1H-pyrazole-5-carboxamide
2-acetamido-N-({4-[4-(2-methoxyphenyl)piperazin-1-yl]quinazolin-2-yl}methyl)acetamide
2-(3-phenylpropyl)-5-[4-(pyrimidin-2-yl)piperazine-1-carbonyl]-1,3-benzoxazole
1-(4-chlorophenyl)-N-({5-methyl-2-[3-(propane-2-sulfonamido)phenyl]-1,3-oxazol-4-yl}methyl)cyclopropane-1-carboxamide
1-{2-[3-(3-chlorobenzoyl)piperidine-1-carbonyl]phenyl}ethan-1-one
1-(2-hydroxyethyl)-5-(1H-indol-2-ylmethyl)-N-(1-phenylethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-cyclohexyl-2-(2-oxo-1,2-dihydropyridin-1-yl)-N-(pyridin-4-ylmethyl)acetamide
2-(2H-1,3-benzodioxol-5-yl)-5-(quinoxalin-5-ylmethyl)-2,3,4,5-tetrahydro-1,5-benzothiazepine
2-methoxy-5-[2-(6-methoxynaphthalen-2-yl)morpholine-4-carbonyl]phenol
3-(4,4-difluoropiperidine-1-carbonyl)-N-(oxolan-3-yl)benzene-1-sulfonamide
2-(1-{[3-(2-methylpropyl)-3H-imidazo[4,5-b]pyridin-2-yl]methyl}cyclopentyl)-1-(piperazin-1-yl)ethan-1-one
2-cyclohexyl-5-{[4-(pyridin-3-ylmethoxy)piperidin-1-yl]methyl}pyrimidine
1-[(3-methoxyphenyl)methyl]-N-[(1-methyl-1H-indol-3-yl)methyl]piperidin-3-amine
N-methyl-N-[2-(1H-pyrazol-1-yl)ethyl]-2-(1H-1,2,3,4-tetrazol-5-yl)benzamide
1-[2-chloro-5-(morpholin-4-yl)phenyl]-3-[1-(1-methyl-1H-pyrazol-4-yl)propyl]urea
3-[1-(2-{3-oxo-2-azaspiro[4.5]decan-2-yl}acetyl)piperidin-4-yl]benzonitrile
N-{[2-chloro-5-(trifluoromethyl)phenyl]methyl}-1-methylpiperidine-2-carboxamide
4-[(3-chloro-5-fluoro-4-methoxyphenyl)methyl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
1-[9-methoxy-7-(6-methoxypyridin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-3-(4-methylphenyl)propan-1-one
(2S)-2-(methoxymethyl)-N-(1-methyl-1H-1,3-benzodiazol-5-yl)pyrrolidine-1-carboxamide
1-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propan-1-one
3-(1-butyl-1H-imidazol-2-yl)-1-(4-chloro-3-methylbenzoyl)piperidine
2-[2-({4-[2-(piperidine-1-carbonyl)phenoxy]piperidin-1-yl}methyl)-1H-pyrrol-1-yl]pyrimidine
N-ethyl-N-[2-(3-methoxyphenoxy)ethyl]-2-{[1,2,4]triazolo[1,5-a]pyrimidin-6-yl}acetamide
2-(benzyloxy)-1-[(2S,6S)-6-(hydroxymethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-4-yl]ethan-1-one
4-(1-methoxypropan-2-yl)-1-[2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]piperidine
4-{6-[4-(pyridin-2-ylmethoxy)piperidin-1-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl}thiomorpholine
5-(3-acetylphenoxymethyl)-N-(2,2-dimethyloxan-4-yl)-1H-pyrazole-3-carboxamide
3-(furan-2-ylmethyl)-3-(1-hydroxybutan-2-yl)-1-(6-methylpyridin-3-yl)urea
2-(ethanesulfonyl)-7-[(2-fluoro-5-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decane
N-[(1R,3R)-3-aminocyclopentyl]-5-[(4-methylpiperidin-1-yl)methyl]furan-2-carboxamide
4-(3-{[1-(1H-pyrazole-4-carbonyl)piperidin-4-yl]oxy}benzoyl)morpholine
3-methyl-N-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}-1H-pyrazole-5-carboxamide
ethyl 1-(2-{4-[2-(2-methoxyphenyl)acetamido]-1H-pyrazol-1-yl}acetyl)piperidine-3-carboxylate
1-methyl-1-[3-(1-methyl-1H-imidazol-2-yl)propyl]-3-(1-methyl-4-phenyl-1H-pyrazol-5-yl)urea
3-(azocan-1-yl)-N-{1-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}propanamide
3,5,7-trimethyl-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]-1H-indole-2-carboxamide
3-(2-methyl-1H-indol-1-yl)-N-[2-(morpholin-4-yl)ethyl]propanamide
1-(2-fluorophenyl)-4-{1-[3-(1H-pyrazol-1-yl)benzoyl]piperidin-3-yl}piperazine
(2S,4S)-4-{[(2,6-difluorophenyl)methyl]amino}-N-(propan-2-yl)-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
4-(naphthalen-2-yloxy)-1-[(3E)-pent-3-enoyl]piperidine-4-carboxylic acid
(1R,6S)-9-methyl-N-(3-methylcinnolin-5-yl)-3,9-diazabicyclo[4.2.1]nonane-3-carboxamide
N1,N1-dimethyl-N3-[3-(4-methyl-1H-pyrazol-1-yl)propyl]piperidine-1,3-dicarboxamide
3-[(3S,7S,8aS)-1,4-dioxo-3-(propan-2-yl)-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(3-chlorophenyl)urea
[(3R,4R)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-[(6-methylpyridin-2-yl)methyl]pyrrolidin-3-yl]methanol
5-benzyl-5-{1-[1-(morpholin-4-yl)cyclohexanecarbonyl]piperidin-4-yl}imidazolidine-2,4-dione
6-[(2R,3S,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]hexan-1-ol
(3S,4S)-4-[ethyl(methyl)amino]-1-{[2-(morpholin-4-yl)quinolin-3-yl]methyl}pyrrolidin-3-ol