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1-{2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-3-(1H-pyrazol-3-yl)piperidine
N-(1-hydroxybutan-2-yl)-3-(methylsulfanyl)-N-(pyridin-2-ylmethyl)propanamide
4-(3-{8-fluoro-1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}phenyl)-4H-1,2,4-triazole
3-{3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyridine
N-[1-(4-methylpyridin-2-yl)propyl]-2-(pyridin-4-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
1-butyl-3-(5-methylfuran-2-yl)-5-(oxolan-3-yl)-1H-1,2,4-triazole
2-{[2-fluoro-6-(trifluoromethyl)phenyl]methyl}-5-(4-methylpiperazin-1-yl)-2,3-dihydropyridazin-3-one
4,4,4-trifluoro-1-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]butan-1-one
(2R)-2-phenyl-2-({5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethan-1-ol
5-[(2-methoxyethyl)(methyl)amino]-1-methyl-N-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
(3R,4S)-1-[(3-cyclohexyl-1,2-oxazol-5-yl)methyl]-3,4-dimethylpiperidin-4-ol
1-cycloheptyl-4-({[2-(2-hydroxyethoxy)phenyl]methyl}amino)pyrrolidin-2-one
2-acetamido-N-[(2-methoxyphenyl)methyl]-N-(pyridin-3-ylmethyl)acetamide
3-(3,4-dimethyl-1H-pyrazol-5-yl)-N-[(trimethyl-1H-imidazol-2-yl)methyl]propanamide
3-{5-[1-(4-chlorophenyl)cyclobutyl]-1,3,4-oxadiazol-2-yl}-N-methyl-N-(1H-pyrazol-5-ylmethyl)propanamide
4-methoxy-6-[3-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]pyrimidin-2-amine
3-(4-hydroxyphenyl)-N-[(5-{[(3-methylphenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)methyl]-2-phenylpropanamide
1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-3-(pyrrolidin-1-yl)piperidine
5-ethyl-5-(1-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-3-carbonyl}piperidin-4-yl)imidazolidine-2,4-dione
1-{4-[2-oxo-2-(piperidin-1-yl)ethyl]piperazin-1-yl}-4-(1H-pyrazol-4-yl)butan-1-one
1-[2-(2,3-dimethoxy-5-methylphenyl)pyrimidin-4-yl]piperidin-4-ol
1-[(1S,3R)-1-(2-aminoethoxy)-3-hydroxy-7-azaspiro[3.5]nonan-7-yl]-4-(1H-imidazol-1-yl)butan-1-one
N-(pyridin-3-ylmethyl)-3-(1-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-4-yl)propanamide
(2S,4R)-4-amino-N-(propan-2-yl)-1-[3-(1H-pyrazol-1-yl)benzoyl]pyrrolidine-2-carboxamide
1-{5-[(4-ethylpiperazin-1-yl)methyl]-2-methoxyphenoxy}-3-[methyl(propan-2-yl)amino]propan-2-ol
N-[2-(methoxymethyl)-1-methyl-7-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1H-1,3-benzodiazol-5-yl]-2-phenylacetamide
N-[2-(2-fluorophenyl)ethyl]-3-(morpholine-4-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
4-({2-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}methyl)benzonitrile
3-phenyl-1-{1-[2-(pyrrolidin-1-yl)benzoyl]piperidin-4-yl}propan-1-ol
N-(4-{[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}phenyl)morpholine-2-carboxamide
5-[2-(4-fluorophenyl)pyrrolidine-1-carbonyl]-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
(1S,5R)-6-benzyl-3-({4-oxo-4H-pyrido[1,2-a]pyrimidin-2-yl}methyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1,3-dimethyl-5-{1-methyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-1H-pyrazole
3-hydroxy-N-(1-methylpiperidin-4-yl)-N-(2-phenylethyl)benzamide
3-(1-{[1-(cyclohexylmethyl)-2-methanesulfonyl-1H-imidazol-5-yl]methyl}piperidin-2-yl)propan-1-ol
3-({2-[2-(pyrrolidin-1-yl)ethyl]piperidin-1-yl}sulfonyl)benzonitrile
1-(cyclohex-3-en-1-ylmethyl)-N-[3-(1,3-thiazol-4-yl)phenyl]piperidine-4-carboxamide
6-(propan-2-yloxy)-N4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}pyrimidine-2,4-diamine
(1S,6R)-3-[(2,2-difluoro-2H-1,3-benzodioxol-4-yl)methyl]-3,9-diazabicyclo[4.2.1]nonane
1-[(3R,4S)-3-amino-4-(5-methylfuran-2-yl)pyrrolidin-1-yl]-2-ethoxyethan-1-one
1-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}-2-(2-methoxyethoxy)ethan-1-one
2-(5-acetylthiophen-3-yl)-N-{[3-(trifluoromethoxy)phenyl]methyl}acetamide
N-{2-[2-(5-amino-1H-1,2,3,4-tetrazol-1-yl)acetyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}oxolane-2-carboxamide
ethyl 4-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperazine-1-carboxylate
N-methyl-N-(2-phenoxyethyl)-1-{[3-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
2-cyclopentyl-8-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}-2,8-diazaspiro[5.5]undecan-3-one
4-(benzyloxy)-1-{[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidine
2-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}thiophen-3-amine
1-[3-(2H-1,3-benzodioxol-5-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-(1H-pyrazol-1-yl)ethan-1-one
[(2S)-1-[(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]pyrrolidin-2-yl]methanol