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(1R,5S,8S)-3-({4-[2-(1H-imidazol-1-yl)ethoxy]phenyl}methyl)-8-methoxy-3-azabicyclo[3.2.1]octane
N-[2-(dimethylamino)ethyl]-3-{[1-(1-ethylpiperidine-2-carbonyl)piperidin-4-yl]oxy}-N-methylbenzamide
N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(pyridin-3-ylmethyl)cyclohex-1-ene-1-carboxamide
8-[(3-chloro-4,5-dimethoxyphenyl)methyl]-1-oxa-8-azaspiro[4.6]undecane
3-[3-(dimethylamino)propyl]-5-[1-(2-methylbenzoyl)piperidin-4-yl]-5-[(2-methylphenyl)methyl]imidazolidine-2,4-dione
1-(4-methyl-1H-pyrrole-2-carbonyl)-3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
(3R,4R)-1-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]-4-cyclopropyl-3-methylpiperidin-4-ol
6-{2-[(5-methylpyrazin-2-yl)methyl]-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}pyridine-3-carboxylic acid
2-[(4-chlorophenyl)methyl]-8-[(6-methylpyridin-2-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
{1-[(1-{[3,5-dimethyl-2-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-3-yl)methyl]-1H-1,2,3-triazol-4-yl}methanamine
4-{5-[2-(3-chloro-1,2-oxazol-5-yl)ethyl]-3-methyl-1H-1,2,4-triazol-1-yl}-1-methyl-1,2-dihydroquinolin-2-one
1-(3-benzoylpiperidin-1-yl)-3-(3-chloro-1,2-oxazol-5-yl)propan-1-one
(3S)-3-amino-3-{[2-(3-phenylpropoxy)phenyl]carbamoyl}propanoic acid
4-methoxy-N-(1-phenylcyclopropyl)-3-{[1-(propan-2-yl)piperidin-4-yl]oxy}benzamide
9-cycloheptyl-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
N-butyl-2-methyl-N-(pyridin-4-ylmethyl)-2,8-diazaspiro[4.5]decane-3-carboxamide
4-{[2-(2-methoxyethyl)-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl]methyl}benzamide
1-[2-(4-chloro-2-methylphenoxy)ethyl]-4-(piperidine-3-carbonyl)piperazine
7-(3-chlorophenyl)-4-(piperidin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
5-[5-fluoro-4-(morpholin-4-yl)pyrimidin-2-yl]thiophene-2-carboxylic acid
methyl(3-methylbut-2-en-1-yl)[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]amine
1-(4-methyl-1,2,5-oxadiazol-3-yl)-4-{[3-(4-phenylphenyl)-1H-pyrazol-4-yl]methyl}piperazine
3-(3-hydroxy-1,2-oxazol-5-yl)-1-{2-[2-(4-hydroxyphenyl)ethyl]piperidin-1-yl}propan-1-one
(4aR,8aS)-6-{[3-(benzyloxy)phenyl]methyl}-1-{[3-(trifluoromethyl)phenyl]methyl}-decahydro-1,6-naphthyridin-2-one
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-N-methyl-2-(pyridin-4-yl)pyrimidine-5-carboxamide
1-(5-{[(5-chloropyridin-3-yl)oxy]methyl}-1,2-oxazole-3-carbonyl)-4-(thiophen-2-ylmethyl)-1,4-diazepane
(3S,4S)-1-[3-(1H-imidazol-2-yl)benzoyl]-4-propylpyrrolidine-3-carboxylic acid
2-(1H-imidazol-2-yl)-N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}benzamide
N-({3,5-dimethoxy-4-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]-2,2-diphenylacetamide
2-hydroxy-2-methyl-N-({5-methyl-2-[2-(3-phenoxypropanamido)phenyl]-1,3-oxazol-4-yl}methyl)propanamide
N-[1-(furan-2-carbonyl)piperidin-3-yl]-2,4-dimethylpyrimidine-5-carboxamide
5-({4-[4-(2-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)quinoline
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-(5-chlorothiophene-2-carbonyl)pyrrolidine-3-carboxylic acid
(1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}-4-(3-phenylpropyl)piperidin-4-yl)methanol
[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl][1-(1H-1,2,4-triazol-1-yl)propan-2-yl]amine
1-[(4aR,8aR)-4a-hydroxy-7-(1H-imidazol-2-ylmethyl)-decahydro-2,7-naphthyridin-2-yl]-2-methoxyethan-1-one
5-({2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidin-1-yl}methyl)-2-(thiophen-2-yl)pyrimidine
3-[(2-methoxyphenyl)methyl]-5-(4H-1,2,4-triazol-4-ylmethyl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazole
N-methyl-2-(2-oxo-1,2-dihydropyridin-1-yl)-N-[2-(1H-pyrazol-1-yl)ethyl]acetamide
6-[(2-methylpyrrolidin-1-yl)methyl]-2-oxo-N-(quinolin-3-ylmethyl)-1,2-dihydropyridine-3-carboxamide
(3R,4R)-1-[(4-chloro-3-fluorophenyl)methyl]-4-cyclopropyl-3-methylpiperidin-4-ol
ethyl 1-ethyl-5-(1H-indole-6-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
3-[(2-butyl-1H-imidazol-4-yl)methyl]-5-methyl-5-(piperidin-4-yl)imidazolidine-2,4-dione
methyl 4-{[3-(2-hydroxyethyl)-4-(thiophen-2-ylmethyl)piperazin-1-yl]methyl}benzoate
N-methyl-4-(pyridin-2-yl)-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}pyrimidin-2-amine
methyl(1,2-oxazol-5-ylmethyl){[5-(2-phenylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}amine
1-[1'-(5-fluoro-2-methylbenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
N-[1-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-3,5-dimethyl-1H-indole-2-carboxamide
1-[(2,3-dimethoxyphenyl)methyl]-3-{[ethyl(methyl)amino]methyl}-3-hydroxypiperidin-2-one
[(4-cyclopropyl-5-{1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methyl]dimethylamine