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6,7-dimethoxy-2-[1-(4-methyl-1,3-oxazole-5-carbonyl)piperidin-3-yl]-1,2,3,4-tetrahydroisoquinoline
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[1-(pyrimidin-2-yl)piperidin-3-yl]propanamide
N-[2-(1-{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-2-yl)ethyl]acetamide
3-({[2-(4-methoxy-2,5-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)amino)propane-1,2-diol
5-[2-(6-methoxynaphthalen-2-yl)morpholine-4-carbonyl]pyridin-2-amine
3-{[3-(dimethyl-1,2-oxazol-4-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]sulfonyl}pyridine
8-chloro-2-({[(5-methylpyrazin-2-yl)methyl]amino}methyl)quinolin-4-ol
1-(4-cyclopentylpyrimidin-2-yl)-4-hydroxypiperidine-4-carboxylic acid
1-{2-[(4-chlorophenyl)methyl]benzoyl}-N,N-dimethylazepan-4-amine
N-[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]-1-phenylpiperidin-4-amine
1-[1-(2,3-dimethoxybenzoyl)piperidin-3-yl]-N-(2-methylpropyl)-1H-1,2,3-triazole-4-carboxamide
2-methoxy-N-[1-methyl-2-(pyridin-3-yl)-5-{4H,5H,6H,7H-thieno[3,2-c]pyridine-5-carbonyl}-1H-1,3-benzodiazol-7-yl]acetamide
8-{2-[benzyl(methyl)amino]acetyl}-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
(1S,9S)-11-{[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
3-(piperazine-1-sulfonyl)-N-[1-(1,3-thiazol-2-yl)ethyl]benzamide
2-amino-1-{5-methanesulfonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-methylpropan-1-one
1-(4-{3-[benzyl(methyl)amino]piperidin-1-yl}piperidin-1-yl)ethan-1-one
N-[(2R,3R)-2-methoxy-1'-(1H-pyrazol-3-ylmethyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(thiophen-2-yl)acetamide
3-[(2-methoxyethyl)sulfamoyl]-5-(3-methoxyphenyl)benzoic acid
1-(5-{3-[2-(2,4-difluorophenyl)ethyl]piperidine-1-carbonyl}-1H-pyrazol-3-yl)ethan-1-one
N-(4-fluoro-2-methylphenyl)-3-(1-{[3-(methylsulfanyl)phenyl]methyl}piperidin-3-yl)propanamide
N-methyl-4-[(1-oxo-1,2-dihydroisoquinolin-2-yl)methyl]benzamide
4-[1-(2-methylbutyl)piperidin-3-yl]-5-(2-methylphenyl)-2-(pyridin-4-yl)pyrimidine
6-ethyl-3-[2-(1-methylpiperidin-2-yl)ethyl]-3,4-dihydroquinazolin-4-one
1-tert-butyl-N-(1-cyclohexyl-3-methyl-1H-pyrazol-5-yl)-5-oxopyrrolidine-3-carboxamide
3-(isoquinoline-3-carbonyl)-9-methoxy-7-oxo-N-(thiophen-2-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
1-[(3,4-dimethylphenyl)methyl]-3-(1-methyl-1H-1,2,3-triazol-4-yl)urea
N-(oxolan-3-yl)-5-[(5,6,7,8-tetrahydronaphthalen-2-yloxy)methyl]-1,2-oxazole-3-carboxamide
5-[3-(5-methylfuran-2-yl)-1H-pyrazol-5-yl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
[3-(1H-imidazol-1-yl)propyl][(2E)-2-methylpent-2-en-1-yl](pyridin-3-ylmethyl)amine
4,4,4-trifluoro-1-[4-(2-methylpyridin-4-yl)-1,4-diazepan-1-yl]butan-1-one
1-(benzyloxy)-8-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]-1,8-diazaspiro[4.5]decan-2-one
N-methyl-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetamide
7-[(2,3-dimethoxyphenyl)methyl]-2-[2-(1H-pyrazol-4-yl)ethyl]-2,7-diazaspiro[4.5]decan-6-one
ethyl 3-[(2E)-3-phenylprop-2-en-1-yl]-1-[2-(1H-1,2,3,4-tetrazol-1-yl)acetyl]piperidine-3-carboxylate
6-chloro-2-{[(2S)-4-methyl-2-phenylpiperazin-1-yl]methyl}quinoline
1-{1'-[1-(propan-2-yl)-1H-pyrrole-2-carbonyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}propan-1-one
(4aS,8aR)-6-[(5-chlorothiophen-2-yl)methyl]-1-[2-(1H-imidazol-4-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
N-{3-methyl-1-[(3-methylphenyl)methyl]-1H-pyrazol-5-yl}-5-propyl-1,2-oxazole-3-carboxamide
N-[1-(cyclohexylmethyl)piperidin-3-yl]-1-methyl-4-oxo-1,4-dihydroquinoline-3-carboxamide
9-[4-(3,5-dimethyl-1H-pyrazol-1-yl)butanoyl]-1,4,9-triazaspiro[5.5]undecan-5-one
1-[2-(pyridin-2-yl)ethyl]-5-({spiro[indene-1,4'-piperidine]-1'-yl}carbonyl)piperidin-2-one
propyl N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)carbamate
{3-[(3-chlorophenyl)methyl]-1-{[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}piperidin-3-yl}methanol
4-{[4-(1-benzofuran-2-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-1-(prop-2-en-1-yl)-1H-pyrazole
1-(cyclohex-3-en-1-ylmethyl)-4-(pyridin-3-yl)piperazine
N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-5-propyl-1,2-oxazole-3-carboxamide
2-[(2,6-dichlorophenyl)methyl]-5-(2-ethyl-2,5-dihydro-1H-pyrrole-1-carbonyl)pyrimidin-4-ol
9-(2-methoxyacetyl)-2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
(4aR,8aS)-6-cyclopentyl-1-[(3-fluorophenyl)methyl]-decahydro-1,6-naphthyridin-2-one