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1-(2,6-difluoro-3-methylbenzoyl)-4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepane
8-(1-ethyl-1H-pyrazole-4-carbonyl)-1-oxa-8-azaspiro[4.6]undecane
2-{[3-(2-hydroxyethyl)-4-[(4-methoxy-2,3-dimethylphenyl)methyl]piperazin-1-yl]methyl}quinolin-4-ol
1-[(4-ethoxy-3-methoxyphenyl)methyl]-4-(hydroxymethyl)azepan-4-ol
N-[(5-phenyl-1H-pyrazol-3-yl)methyl]-2-(pyridin-4-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
methyl (2S)-2-{[5-(2-chloro-4-fluorophenoxymethyl)-1,2-oxazol-3-yl]formamido}-2-phenylacetate
N-(isoquinolin-5-ylmethyl)-1-(4-methoxyphenyl)-N-methylcyclopropane-1-carboxamide
1-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-{6-methylimidazo[1,2-a]pyridine-2-carbonyl}piperazine
1-methyl-4-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
[2-(4-methyl-1H-imidazol-2-yl)ethyl]({[8-methyl-2-(piperidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amine
4-[(furan-3-ylmethyl)amino]-1-(2-phenylethyl)pyrrolidin-2-one
N-{[1-(morpholin-4-yl)cyclopentyl]methyl}-3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]propanamide
N-ethyl-3-oxo-N-[2-(pyrrolidin-1-yl)ethyl]-2,3-dihydro-1H-indene-1-carboxamide
(2H-1,3-benzodioxol-5-ylmethyl)(methyl){4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}amine
3,5-dimethyl-4-({2-methyl-2,7-diazaspiro[4.5]decan-7-yl}methyl)phenol
1-cyclohexyl-N-{[2-fluoro-5-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
N-{1-[2-(dimethyl-1,2-oxazol-4-yl)acetyl]piperidin-4-yl}methanesulfonamide
(2S,4R)-N-ethyl-4-[2-(1H-imidazol-1-yl)acetamido]-1-[(6-methylpyridin-2-yl)methyl]pyrrolidine-2-carboxamide
1-(3-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-(1H-1,2,4-triazol-1-yl)ethan-1-one
(3R,5S)-N-(2-methylpropyl)-1-(naphthalen-2-ylmethyl)-5-[3-(trifluoromethyl)phenoxymethyl]piperidine-3-carboxamide
N-[(8-methoxyquinolin-5-yl)methyl]-N-methyl-6-(4H-1,2,4-triazol-4-yl)pyridine-2-carboxamide
N-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)ethyl]-6-methoxy-N-methyl-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
5-[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-4-yl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carbonitrile
5-(2H-1,3-benzodioxol-5-yl)-3-[4-(2,6-dimethylpyridin-4-yl)piperazin-1-yl]-1,2,4-triazine
methyl 4-{[4-(3-methoxybenzoyl)piperazin-1-yl]methyl}thiophene-2-carboxylate
5-{3-[(4-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}-N-[1-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]pyridin-2-amine
1-methyl-3-phenyl-8-(propane-1-sulfonyl)-1,8-diazaspiro[4.5]decan-2-one
N-({2-[4-(2-methylphenyl)piperazin-1-yl]pyridin-3-yl}methyl)propane-2-sulfonamide
N-(2-methoxyethyl)-3-[(3S,4R)-1-(propan-2-yl)-4-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-3-yl]propanamide
methyl (2S,4S)-1-methyl-4-(3-oxo-3,4-dihydro-2H-1,4-benzoxazine-6-sulfonamido)pyrrolidine-2-carboxylate
2-{4-[2-(4,6-dimethyl-1-benzofuran-3-yl)acetyl]-2-oxopiperazin-1-yl}benzonitrile
1-{2-[4-(3-methylpyridin-4-yl)-1,4-diazepane-1-carbonyl]phenyl}ethan-1-one
3-[5-(2,5-dimethylfuran-3-yl)-3-(thiophen-2-ylmethyl)-1H-1,2,4-triazol-1-yl]-1λ6-thiolane-1,1-dione
6-(2-fluoro-6-methoxyphenyl)-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}pyridine-3-carboxamide
2-[({2,4-dimethyl-5-[(4-methylpiperidin-1-yl)methyl]phenyl}methyl)(methyl)amino]-N-methylacetamide
1-[3-(1-benzyl-1H-imidazol-2-yl)piperidin-1-yl]-3-(pyridin-3-yl)propan-1-one
2-(4-acetyl-1,4-diazepan-1-yl)-2-(2,3,4-trimethoxyphenyl)acetic acid
9-(2-methoxyethyl)-1-methyl-4-[2-(methylsulfanyl)pyrimidin-4-yl]-1,4,9-triazaspiro[5.6]dodecan-10-one
N-[2-(3-fluorophenyl)ethyl]-2-[4-(4-{[2-(1H-1,2,4-triazol-1-yl)ethyl]amino}piperidin-1-yl)phenyl]acetamide
1-{1-[3-(2-methylphenyl)phenyl]piperidin-4-yl}piperidin-3-ol
1-[5-({[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]amino}methyl)-2-methoxyphenoxy]-3-(piperidin-1-yl)propan-2-ol
{[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}[(5-ethylpyridin-2-yl)methyl]methylamine
4-{4-[2-(2,2-dimethyloxan-4-yl)-1H-imidazol-1-yl]piperidine-1-carbonyl}morpholine
1-benzyl-3-methyl-8-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-methyl-2-(2-phenyl-1H-imidazol-1-yl)-N-[2-(1H-pyrazol-4-yl)ethyl]acetamide
1-(2,4-dimethoxybenzoyl)-N-(4-methoxyphenyl)piperidin-3-amine
(2E)-1-{3-[4-(hydroxymethyl)piperidin-1-yl]piperidin-1-yl}-3-(pyridin-3-yl)prop-2-en-1-one
1-{1'-[2-(methylsulfanyl)pyrimidin-4-yl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}ethan-1-one
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-1-[4-(4H-1,2,4-triazol-4-yl)piperidin-1-yl]ethan-1-one
1-cyclopropyl-4-[4-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]pyrrolidin-2-one