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(2S,4R)-4-(cyclooctylamino)-N-ethyl-1-(naphthalen-1-ylmethyl)pyrrolidine-2-carboxamide
(2S)-1-{[4-(cyclopentyloxy)phenyl]methyl}-2-(methoxymethyl)pyrrolidine
2-(1-methyl-4-{[4-(2-methylpropyl)phenyl]methyl}piperazin-2-yl)ethan-1-ol
2-[(2-fluorophenyl)methyl]-N-[2-(5-methyl-4H-1,2,4-triazol-3-yl)ethyl]-1,3-benzoxazole-6-carboxamide
3-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonane-3-carbonyl]-2H-chromen-2-one
2-(azepan-1-yl)-1-{3-[(4-fluorophenyl)methyl]-3-(hydroxymethyl)piperidin-1-yl}ethan-1-one
(3aS,6aR)-5-(2H-1,3-benzodioxol-4-ylmethyl)-3-cyclopentyl-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N-cyclopropyl-N-({4-[(4-fluorophenyl)methoxy]-3-methoxyphenyl}methyl)-2,3-dimethyl-1H-indole-7-carboxamide
N-{[3-(difluoromethoxy)phenyl]methyl}-1-ethyl-5-oxopyrrolidine-3-carboxamide
methyl 3-(2-methoxyacetamido)-5-({[2-(trifluoromethyl)phenyl]formamido}methyl)benzoate
N-{1-[1-(2H-1,3-benzodioxol-5-ylmethyl)piperidin-4-yl]-2-phenylethyl}-N,1,3-trimethyl-1H-pyrazole-5-carboxamide
methyl 3-(3-ethynylbenzoyl)-7-oxo-9-(pyridin-2-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-[(2R,3R)-3-(dimethylamino)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]-2-(4-methyl-1,2,5-oxadiazol-3-yl)ethan-1-one
5-(6-methoxy-2H-1,3-benzodioxol-5-yl)-1-(1-phenylethyl)-1H,4H-pyrazolo[3,4-d]imidazole
methyl(pyrazin-2-ylmethyl){[4-(trifluoromethyl)phenyl]methyl}amine
N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-4-carboxamide
methyl 6-[3-(3-methylphenoxymethyl)piperidin-1-yl]pyrimidine-4-carboxylate
(1s,4s)-4-hydroxy-N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]cyclohexane-1-carboxamide
3-[3-(3-methylthiophen-2-yl)phenyl]-1-(pyrrolidin-3-ylmethyl)-1H-pyrazole
2-[2-(1H-imidazol-4-yl)ethyl]-8-[3-(methylsulfanyl)propanoyl]-2,8-diazaspiro[5.5]undecan-3-one
2,5-dimethyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
N-[3-(3-chlorophenyl)phenyl]-1-(cyclopent-1-ene-1-carbonyl)piperidine-4-carboxamide
N-[(2-ethyl-5-fluoro-3-methyl-1H-indol-7-yl)methyl]-2-(1H-imidazol-1-yl)acetamide
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-4-(piperidin-1-yl)piperidine-4-carboxamide
N-cyclohexyl-4-methoxy-3-{[1-(propan-2-yl)piperidin-4-yl]oxy}benzamide
(1S,5R)-6-(4-methylpiperazine-1-carbonyl)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)-1-[2-(morpholin-4-ylmethyl)piperidin-1-yl]propan-1-one
4-fluoro-N-[(1-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}piperidin-3-yl)methyl]benzamide
1-(2-ethoxyethyl)-N-methyl-N-[(3-methylpyridin-4-yl)methyl]-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
3-(2,6-dimethylpyridin-3-yl)-1-methyl-1-[1-(pyridin-3-yl)propyl]urea
(3aR,6aR)-2-acetyl-5-[(1-phenyl-1H-pyrazol-5-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
8-methoxy-5-(1,2,3,4-tetrahydroisoquinolin-7-yl)quinoline
N-(2,1,3-benzothiadiazol-5-ylmethyl)-2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-methylacetamide
2-{3-methyl-5-[5-(thiophen-2-yl)-1H-pyrazol-4-yl]-1H-1,2,4-triazol-1-yl}pyridine
N-{[5-methyl-7-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-4-(thiophen-2-yl)butanamide
3-{2-[({6-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[2,1-b][1,3]thiazol-5-yl}methyl)amino]ethyl}-1,3-oxazolidin-2-one
[(3,4-dimethoxyphenyl)methyl]({[1-(2-methoxyethyl)piperidin-4-yl]methyl})(pyridin-4-ylmethyl)amine
5-[2-(1-methyl-1H-imidazol-2-yl)phenyl]-3-phenyl-1H-1,2,4-triazole
2-{[3-(2-amino-1,3-thiazol-4-yl)propyl]amino}-N-(3-fluoro-4-methylphenyl)acetamide
N5-(1,3-benzothiazol-2-ylmethyl)-1-(cyclohexylmethyl)-N3,N3-dimethyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
(2R,3R)-2-hydroxy-3-(morpholin-4-yl)-N-phenyl-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-carboxamide
2-{[(5-tert-butyl-1H-pyrazol-3-yl)methyl](thiophen-2-ylmethyl)amino}butan-1-ol
1-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)sulfonyl]-4-(5-methylpyridin-2-yl)piperidin-4-ol
1-{1-[(1-cyclopentyl-1H-imidazol-5-yl)methyl]piperidin-3-yl}-2-phenylethan-1-one
N-cyclopentyl-N-[(2,5-dimethoxyphenyl)methyl]pyridine-4-carboxamide
1-(2,2-dimethylpropyl)-3-hydroxy-3-({[(3-methylpyridin-2-yl)methyl]amino}methyl)piperidin-2-one
3-(5-amino-1H-1,2,4-triazol-3-yl)-1-[9-hydroxy-7-(4-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propan-1-one
2-({2-[3-(N-ethylacetamido)pyrrolidine-1-carbonyl]phenyl}amino)acetic acid
5-{2-[4-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]-2-oxoethyl}-6-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
[(1R,5S,6S)-3-azabicyclo[3.1.0]hexan-6-ylmethyl][(2-fluorophenyl)methyl]propylamine