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4-{2-[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]acetyl}-1-(2-methylphenyl)piperazin-2-one
N-(furan-2-ylmethyl)-2-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-(prop-2-yn-1-yl)benzamide
N,N-dimethyl-3-{[2-(3-methyl-1H-1,2,4-triazol-5-yl)pyrrolidin-1-yl]sulfonyl}benzamide
N-[(2-fluorophenyl)methyl]-3-{1-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]piperidin-3-yl}propanamide
2-(2-methylpropyl)-8-(1,3-thiazol-2-yl)-2,8-diazaspiro[4.5]decan-3-one
methyl (2S,4R)-4-cyclohexaneamido-1-[(4-methoxyphenyl)methyl]pyrrolidine-2-carboxylate
1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one
3-[(4-{[1-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)ethyl]amino}-6-methylpyrimidin-2-yl)amino]phenol
1-benzyl-5-(thiophen-3-yl)-1H,4H-pyrazolo[3,4-d]imidazole
N-{1-[1-(2,1,3-benzothiadiazol-5-ylmethyl)piperidin-4-yl]-2-phenylethyl}-N-methyl-2-(1H-pyrazol-1-yl)acetamide
1-{1-[(5-chlorofuran-2-yl)methyl]azetidin-3-yl}-3,5-dimethyl-1H-pyrazole
1-{1-[3-(4-fluorophenyl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}piperidin-3-ol
6-fluoro-2-{2-[3-(3-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]ethyl}-1H-1,3-benzodiazole
8-chloro-N,N-bis(1,3-oxazol-4-ylmethyl)quinoline-2-carboxamide
2-(cyclobutylmethyl)-7-[(2,3-dimethoxyphenyl)methyl]-2,7-diazaspiro[4.5]decane
(2S,4S,5R)-5-(2,3-difluorophenyl)-4-{[2-(dimethylamino)ethyl](methyl)carbamoyl}-1-methylpyrrolidine-2-carboxylic acid
(4-methyl-5-{[1-(quinoline-2-carbonyl)piperidin-4-yl]methyl}-4H-1,2,4-triazol-3-yl)methanol
(1R,5R)-6-(cyclopropylmethyl)-3-[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]-3,6-diazabicyclo[3.2.2]nonane
2,6-dihydroxy-N-[1-phenyl-3-(1H-1,2,4-triazol-1-yl)propyl]benzamide
3-[2-(2,6-difluorophenyl)ethyl]-1-(3-propyl-1H-pyrazole-4-carbonyl)piperidine
N-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-1H-pyrrolo[2,3-b]pyridin-6-amine
2-(1H-1,3-benzodiazol-1-ylmethyl)-N-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-1,3-oxazole-4-carboxamide
9-(2,4-dimethylbenzoyl)-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-methoxy-N-[(1S,3S)-3-{[4-(pyridin-4-yl)pyrimidin-2-yl]amino}cyclopentyl]propanamide
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-N-methyl-2-oxo-2H-chromene-3-carboxamide
5-[5-(furan-3-yl)-1,2,4-oxadiazol-3-yl]-6-methyl-2-(oxolane-3-carbonyl)-1,2,3,4-tetrahydro-2,7-naphthyridine
4-(2-methyl-1H-imidazol-1-yl)-1-[(1S,5R)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]butan-1-one
(4aS,8aR)-1-[2-(1H-imidazol-4-yl)ethyl]-6-(2-methyl-1,3-thiazole-4-carbonyl)-decahydro-1,6-naphthyridin-2-one
2,6-dimethyl-4-{4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine
4-[4-(2-fluorobenzoyl)piperazin-1-yl]-2-(pyridin-3-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
2-{4-[1-(furan-3-ylmethyl)-1H-imidazol-2-yl]phenoxy}ethan-1-ol
ethyl 4-({1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}amino)piperidine-1-carboxylate
2-(2H-1,3-benzodioxol-5-yl)quinoxaline
1-(3-{3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}piperidin-1-yl)propan-1-one
1-{[2-cyclohexylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-3-(methoxymethyl)piperidine
[(2R)-1-(8-fluoroquinoline-2-carbonyl)pyrrolidin-2-yl]methanol
N-[4-(3-methoxyphenyl)phenyl]-1-(3-methylbutanoyl)piperidine-3-carboxamide
5-(4-chlorophenyl)-N-methyl-N-(pyrazin-2-ylmethyl)-1,2,4-triazin-3-amine
1-{pyrazolo[1,5-a]pyridine-3-carbonyl}-4-(pyrrolidine-1-carbonyl)piperidine
2-ethyl-9-(2-hydroxynaphthalene-1-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
N-{[4-(2,3-dihydro-1H-inden-2-yloxy)phenyl]methyl}-2,5-dimethoxy-N-[(3S)-2-oxoazepan-3-yl]benzamide
N-methyl-3-(4-{4-[(3-methylpiperidin-1-yl)methyl]-1H-1,2,3-triazol-1-yl}piperidine-1-carbonyl)pyridin-2-amine
8-(3,5-dimethylbenzoyl)-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-amino-8-(4-methyl-2-oxo-2H-chromen-7-yl)-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
(3S,9aR)-2-methyl-3-(2-methylpropyl)-8-[(1-phenyl-1H-pyrazol-4-yl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
8-(3-methoxypropanoyl)-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
1-cycloheptyl-6-oxo-N-[(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]piperidine-3-carboxamide
8-[4-(difluoromethoxy)benzenesulfonyl]-2,8-diazaspiro[4.5]decan-3-one
(3R,4S)-N,N-dimethyl-1-[6-methyl-2-(morpholin-4-yl)pyrimidin-4-yl]-4-(propan-2-yl)pyrrolidin-3-amine
4-[(3-chlorophenyl)methyl]-1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1,4-diazepan-5-one