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4-[(1-cyclopentylpiperidin-4-yl)oxy]-N-(furan-2-ylmethyl)-3-methoxybenzamide
9-(1-phenyl-1H-1,2,3-triazole-4-carbonyl)-1-oxa-9-azaspiro[5.5]undecan-5-ol
5-{1-[2-(4-oxo-3,4-dihydro-1,2,3-benzotriazin-3-yl)acetyl]pyrrolidin-2-yl}thiophene-2-carboxamide
4-{2-[(2R,3R,6R)-3-(3-hydroxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-oxoethyl}piperazin-2-one
5-methyl-N-[(3-methylphenyl)methyl]-4-[(pyridin-2-ylmethyl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
N-(1-{4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-1-oxopropan-2-yl)methanesulfonamide
1-[(3-fluorophenyl)methyl]-4-[2-(phenylsulfanyl)ethyl]piperazine
N-[2-(4-fluorophenyl)ethyl]-N-{[7-methoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-3-(3-methyl-1H-pyrazol-1-yl)propanamide
1-methyl-4-(1-{2-[4-(methylsulfanyl)phenyl]-1H-imidazol-1-yl}butan-2-yl)piperazine
4-{[3-(2-methyl-5-propylpyrimidin-4-yl)phenyl]methyl}morpholine
7-[4-(azepan-1-ylmethyl)benzoyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-[2-(3-methoxyphenyl)ethyl]-2-(3-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
{5-methyl-7-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methanamine
5-{[3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
(2R,3R)-3-{6-oxa-9-azaspiro[4.5]decan-9-yl}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
2-(4-{[(1R,5R)-6-methyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]sulfonyl}phenoxy)acetamide
(3R,4S)-4-cyclopropyl-1-[1-(4-fluorophenyl)cyclopropanecarbonyl]pyrrolidin-3-amine
N-[1-(cyclopropylmethyl)-1H-pyrazol-5-yl]-2-[3-(5-methylfuran-2-yl)-1H-indazol-1-yl]acetamide
1-[1-(2,6-dimethoxybenzoyl)piperidin-3-yl]-4-(2-fluorophenyl)piperazine
N-[(4-acetylmorpholin-2-yl)methyl]-2-[(4-chlorophenyl)sulfanyl]acetamide
{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(1H-imidazol-2-ylmethyl)methylamine
5-[1-(2,5-dimethylbenzoyl)piperidin-4-yl]-5-(pyridin-3-yl)-3-(thiophen-3-ylmethyl)imidazolidine-2,4-dione
3-fluoro-N-{[7-(thiophen-3-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}benzamide
3-methyl-4-{6-[(pyridin-3-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}benzoic acid
N-(2-{7-[(2-methylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)cyclobutanecarboxamide
3-({2-cyclopentyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}amino)propane-1,2-diol
N-(1-{7-[(2,6-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)furan-2-carboxamide
2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-N-(thiolan-3-yl)acetamide
2-(4-methyl-1,4-diazepan-1-yl)-N-[2-(4-methylbenzenesulfonyl)ethyl]acetamide
N-(1-{7-[(4-hydroxy-3-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-3-phenylpropanamide
N-({1-[2-(dimethyl-1,2-oxazol-4-yl)acetyl]piperidin-3-yl}methyl)naphthalene-1-carboxamide
3,3-dimethyl-1-({5-[(4-methyl-1H-imidazol-2-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)urea
7-methyl-2-[2-(4-oxo-1,4-dihydroquinolin-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
1-(5-ethyl-2-methylpyrimidin-4-yl)-N-[2-(2-fluorophenoxy)ethyl]piperidin-4-amine
3-methyl-1-[2-(prop-2-en-1-yloxy)phenyl]-3-[(1,2,2-trimethylpyrrolidin-3-yl)methyl]urea
2-cyclopentyl-9-(3,4-dihydro-2H-1-benzopyran-2-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
2-(2,5-dimethylphenoxy)-1-[3-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propan-1-one
8-[(2-aminopyridin-3-yl)methyl]-3-ethyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[2-(3-methoxyphenyl)phenyl]-2-methyl-5-oxo-1,4-diazepane-1-carboxamide
{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}(methyl)[(3-phenyl-1,2-oxazol-5-yl)methyl]amine
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-[(4-ethylphenyl)methyl]-N-methyl-1,3-oxazole-4-carboxamide
2-ethoxy-6-[(4-{7-methylthieno[3,2-d]pyrimidin-4-yl}piperazin-1-yl)methyl]phenol
1-[4-(hydroxymethyl)-4-(2-phenoxyethyl)piperidin-1-yl]-2-[(4S,6R)-6-methyl-2-sulfanylidene-1,3-diazinan-4-yl]ethan-1-one
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N,5-dimethyl-1-propyl-1H-pyrazole-4-carboxamide
4-benzyl-3-[1-(4-methyl-1,2,5-oxadiazole-3-carbonyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[2-(2-fluorophenyl)ethyl]-1-(7-methanesulfonyl-4-methylquinazolin-2-yl)piperidine-4-carboxamide
2-(2-methoxyethyl)-8-[3-(1H-pyrazol-1-yl)propanoyl]-2,8-diazaspiro[5.5]undecan-3-one
1-{2-phenylimidazo[1,2-a]pyridine-6-carbonyl}-4-(4H-1,2,4-triazol-4-yl)piperidine
3-{[(5-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}furan-2-yl)methyl]sulfanyl}-4H-1,2,4-triazole
7-(8-chloroquinoline-2-carbonyl)-N,N-dimethyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine