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methyl 3-[(3-ethoxyphenyl)methyl]-9-[3-(1-methyl-1H-pyrazol-4-yl)propoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
6-(aminomethyl)-2-(2-{[(2R)-2-(methoxymethyl)pyrrolidin-1-yl]methyl}phenyl)-3,4-dihydropyrimidin-4-one
3-(2,1,3-benzothiadiazol-4-yl)-1-[2-(morpholin-4-yl)-2-(pyridin-4-yl)ethyl]urea
[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl][(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]amine
5-{3-oxo-3-[4-(pyrimidin-2-yl)piperazin-1-yl]propyl}-5-[(4-phenylphenyl)methyl]pyrrolidin-2-one
2-{4-[(2,3-difluorophenyl)methyl]-1-(thiophen-3-ylmethyl)piperazin-2-yl}ethan-1-ol
3-methyl-7-[2-(2-methylphenoxy)acetyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
(2S,4R)-N-ethyl-4-[4-(2-propanamidopropan-2-yl)-1H-1,2,3-triazol-1-yl]pyrrolidine-2-carboxamide
1-[5-(2,6-dimethylphenoxymethyl)-1,2-oxazole-3-carbonyl]-4-(2,4-dimethylphenyl)piperazine
6-{[(3,4-dihydro-2H-1-benzopyran-6-ylmethyl)amino]methyl}-1,4-oxazepan-6-ol
4-[3-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)propanoyl]-1-phenylpiperazin-2-one
5-(3,6-dimethyl-1-benzofuran-2-carbonyl)-N,N-dimethyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-3-carboxamide
3-{[6,6-dimethyl-1-(4-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]carbamoyl}pyridin-1-ium-1-olate
2-(3-methoxypropyl)-8-[3-(1H-1,2,4-triazol-1-yl)propanoyl]-2,8-diazaspiro[4.5]decan-3-one
(1S,9R)-11-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
N-[(1,5-dimethyl-1H-pyrazol-3-yl)methyl]-2-[1-(2,2-diphenylethyl)-3-oxopiperazin-2-yl]acetamide
1-methyl-3-(2-methylpropyl)-N-[2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)ethyl]-1H-pyrazole-5-carboxamide
N-[(3R,5S)-1-[(2-aminopyridin-3-yl)methyl]-5-(ethylcarbamoyl)pyrrolidin-3-yl]-4-methyl-1H-imidazole-2-carboxamide
{2-[4-(2-methoxyphenyl)-3-oxopiperazin-1-yl]-2-oxoethyl}urea
N-methyl-N-{2-[4-(4-methylpiperazine-1-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}-3-(trifluoromethyl)benzene-1-sulfonamide
8-(2,1,3-benzoxadiazole-5-carbonyl)-2-[2-(dimethylamino)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
2-[methyl(2-phenylethyl)amino]-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-2,3-dihydro-1H-indene-2-carboxamide
N-{[2-(dimethylamino)pyridin-3-yl]methyl}-4-(thiophen-2-yl)butanamide
N,N-diethyl-1-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}piperidine-3-carboxamide
2-(2-chlorophenoxy)-1-[(3R,4R)-3-(hydroxymethyl)-4-{[4-(hydroxymethyl)piperidin-1-yl]methyl}pyrrolidin-1-yl]ethan-1-one
3-{[2-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-{1-[({2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}carbamoyl)methyl]-1H-pyrazol-4-yl}-3-phenoxypropanamide
3-[1-(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)piperidin-4-yl]-1,3-oxazolidin-2-one
(2R,6R)-11-methoxy-4-(oxan-4-yl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
N-[1-(1-{[3-(ethoxymethyl)-4-methoxyphenyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]-2,2-dimethylpropanamide
4-(4-chloro-3-methylbenzoyl)-1-(2-methylphenyl)piperazin-2-one
3-{[(2S)-2-benzyl-3-oxopiperazin-1-yl]methyl}-6-methyl-1,2-dihydroquinolin-2-one
3-phenyl-1-[4-(quinolin-4-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]propan-1-ol
N-{[1-(4-fluorophenyl)-3,5-dimethyl-1H-pyrazol-4-yl]methyl}-3-(1-methylpiperidin-2-yl)propanamide
(3aR,6aR)-2-(2-chlorobenzoyl)-5-methanesulfonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-(4-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}-1,4-diazepan-1-yl)-1,3-benzothiazole
2-(carbamoylamino)-N-[(3R,4S)-4-cyclopropyl-1-(2-methoxyethyl)pyrrolidin-3-yl]acetamide
3-{1-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1-[4-(pyridin-2-ylmethoxy)phenyl]urea
1-(5-{6-amino-1H-pyrrolo[2,3-b]pyridin-4-yl}-1H-1,3-benzodiazol-2-yl)ethan-1-ol
methyl({[3-(4-phenylphenyl)-1H-pyrazol-4-yl]methyl})(pyrazin-2-ylmethyl)amine
(2Z)-3-(3-fluorophenyl)-N-{3-[4-(4-methylpiperazine-1-carbonyl)-1H-1,2,3-triazol-1-yl]propyl}prop-2-enamide
4-[(4-fluorophenyl)methyl]-1-[1-(2-methoxyethyl)pyrrolidine-3-carbonyl]piperidine
1-(2-oxo-2-{3-phenyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl}ethyl)-1,2-dihydropyridin-2-one
1-[3-(1H-pyrazol-5-yl)piperidin-1-yl]-2-(2,2,6,6-tetramethylpiperidin-4-yl)ethan-1-one
9-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-5-methoxy-1-oxa-9-azaspiro[5.5]undecane
5-acetyl-N-[1-(2-methoxyphenyl)propan-2-yl]-N-methyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
1,5-dimethyl (2R)-2-[(4-{[2-(dimethylamino)ethyl]amino}-5-methylthieno[2,3-d]pyrimidin-6-yl)formamido]pentanedioate
1-(2-chlorophenyl)-3-{1-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
N-cyclopropyl-5-(phenoxymethyl)-N-(pyridin-3-ylmethyl)-1H-pyrazole-3-carboxamide
methyl (2R,4S)-4-hydroxy-1-[(4-hydroxyquinolin-2-yl)methyl]piperidine-2-carboxylate