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2-{5-[(2-phenyl-1,3-thiazol-4-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}pyridine
methyl 3-[(2-fluoro-4-methoxyphenyl)methyl]-7-oxo-9-[2-(2-oxopyrrolidin-1-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
methyl 5-[(3,3-dimethylcyclohexyl)amino]-3-(2-methoxyacetamido)-1-methyl-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N,7-dimethyl-4-oxo-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-4H-chromene-2-carboxamide
1-(4-{[3-(dimethylamino)-2-methylpropyl]amino}-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
5-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
(4aS,8aR)-1-(3-methoxypropyl)-6-[3-(1,2-oxazolidin-2-yl)propanoyl]-decahydro-1,6-naphthyridin-2-one
3-methoxy-1-{4-[3-(4-methylpiperazine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}propan-1-one
1-(isoquinolin-1-yl)-4-(5-methylpyridin-2-yl)piperidin-4-ol
2-(methylsulfanyl)-N-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]pyrimidine-5-carboxamide
(2E)-1-[3-(4-methoxy-3,5-dimethylbenzoyl)piperidin-1-yl]-3-(pyridin-3-yl)prop-2-en-1-one
3-(1-methyl-1H-imidazol-2-yl)-6-[3-(1H-pyrazol-5-yl)phenyl]pyridazine
4-({1-[(2R)-2-aminopropanoyl]piperidin-4-yl}oxy)-3-chloro-N-cyclopentylbenzamide
1-(3,5-dimethyl-1-{1-[3-(propan-2-yl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]propan-2-yl}-1H-pyrazol-4-yl)ethan-1-one
N-methyl-4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}-N-[2-(oxan-2-yl)ethyl]butanamide
N-[4-({[2-(4,6-dimethylpyrimidin-2-yl)ethyl]carbamoyl}methyl)phenyl]butanamide
8-{[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-[(1,5-dimethyl-3-oxo-2-phenyl-2,3-dihydro-1H-pyrazol-4-yl)methyl]piperazine-2-carboxylic acid
6-methyl-N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-2-(pyridin-3-yl)pyrimidin-4-amine
3-methyl-1-{5-[2-(methylsulfanyl)phenoxymethyl]-1,2-oxazole-3-carbonyl}piperidine
6-(6-ethyl-2-methylquinoline-4-carbonyl)-N-phenyl-6-azaspiro[2.5]octane-1-carboxamide
1-(quinoxaline-6-carbonyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-{5-[1-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)ethyl]-1,2,4-oxadiazol-3-yl}pyridine
6-{1-[(2-chloro-6-fluorophenyl)methyl]-1H-1,2,4-triazol-5-yl}-4-methyl-3,4-dihydro-2H-1,4-benzoxazin-3-one
4-methoxy-N-(1-{1-[3-(methylsulfanyl)propyl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
4-[(2S,4R)-1-[(4-ethylphenyl)methyl]-4-[(1-methyl-1H-imidazol-2-yl)sulfanyl]pyrrolidine-2-carbonyl]morpholine
(3S)-4-{[2-cyclopropylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-1,3-dimethylpiperazin-2-one
2-(4-{[2-(furan-2-yl)pyrimidin-5-yl]methyl}piperazin-1-yl)-4-methoxypyrimidine
N-methyl-N-propyl-5-[(quinolin-6-yloxy)methyl]-1,2-oxazole-3-carboxamide
1-{1-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]cyclopentyl}pyrrolidine
ethyl 3-[(2-fluorophenyl)methyl]-1-{[5-(3-hydroxy-3-methylbut-1-yn-1-yl)thiophen-2-yl]methyl}piperidine-3-carboxylate
9-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}-6-oxa-9-azaspiro[4.5]decane
3-cyclopropyl-5-[3-(1H-pyrazol-4-yl)phenyl]-1H-1,2,4-triazole
N-[(2R,3R)-1'-(1H-imidazol-4-ylmethyl)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(methylsulfanyl)acetamide
4-({5-[3-(2-chlorophenyl)-5-methyl-1,2-oxazol-4-yl]-1,2,4-oxadiazol-3-yl}methyl)-1-methylpiperidine
N-[2-(2-chlorophenoxy)ethyl]-5-(methoxymethyl)thiophene-2-carboxamide
2-(ethylamino)-N-[1-(1-methyl-1H-imidazol-2-yl)butyl]pyrimidine-5-carboxamide
1-[(3-cyclopropyl-1H-1,2,4-triazol-5-yl)methyl]-4-phenylpyrrolidin-2-one
methyl N-(2-{8-benzyl-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}-2-oxoethyl)carbamate
3-(methanesulfonylmethyl)-N-[3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]piperidine-1-carboxamide
2-(4-{[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}piperazin-1-yl)ethan-1-ol
methyl 2-[1-(2-methoxyethyl)-8-[3-(5-methylfuran-2-yl)butyl]-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-3-yl]acetate
1-cyclopropyl-4-{[2-(2,3-dichloro-4-methylphenyl)-1H-imidazol-1-yl]methyl}pyrrolidin-2-one
2-(4-methylpiperazin-1-yl)-2-[2-(methylsulfanyl)phenyl]acetic acid
7-[(3-methylphenyl)methyl]-2-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]-2,7-diazaspiro[4.5]decane
4-[(3,5-dimethoxyphenyl)methyl]-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-(1,4-diazepane-1-sulfonyl)-N-[3-(methylsulfanyl)propyl]benzamide
N-[2-(1-hydroxycyclopentyl)ethyl]-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
4-(piperidin-1-ylmethyl)-N-[3-(1H-1,2,3-triazol-1-yl)propyl]benzamide
1-(1-{2-[4-(hydroxymethyl)phenyl]acetyl}piperidin-3-yl)-3-phenylpropan-1-one