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1-[(4aS,8aR)-4a-(hydroxymethyl)-decahydro-1,6-naphthyridin-6-yl]-2-(4-phenylpiperidin-1-yl)ethan-1-one
1-({3-[(2-methylphenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-2-(propan-2-yl)-1H-1,3-benzodiazole
4-{3-[(2R,6S)-2,6-dimethylmorpholin-4-yl]propanoyl}-1-(4-methylphenyl)piperazin-2-one
{[3-(1-benzofuran-2-yl)-1H-pyrazol-4-yl]methyl}[2-(thiophen-2-yl)ethyl]amine
(1-{2-[2-(2-butyl-1H-imidazol-4-yl)-1H-imidazol-1-yl]ethyl}piperidin-2-yl)methanol
N-[2-(pyrrolidin-1-yl)phenyl]-5-(pyrrolidin-2-yl)thiophene-2-carboxamide
N-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-4-(pyridin-3-yl)pyrimidin-2-amine
1-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-(5-methyl-1H-1,2,4-triazol-3-yl)propan-1-one
4-({[(5-cyclopropyl-1H-pyrazol-3-yl)methyl](methyl)amino}methyl)-N-(1-methyl-1H-pyrazol-4-yl)benzamide
1-{[4-methoxy-3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl}-4-(pyridin-3-yl)piperazine
1-[(5-acetylthiophen-3-yl)methyl]-N-[4-(1,3-thiazol-4-yl)phenyl]piperidine-3-carboxamide
N-(2-fluorophenyl)-3-[(4-oxo-4H-chromen-3-yl)formamido]propanamide
2-[4-(2,5-dimethoxyphenyl)-4H-1,2,4-triazol-3-yl]ethan-1-amine
(3S,5S)-1-[(3-methylphenyl)methyl]-5-[(pyridin-3-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
N-cyclobutyl-1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
(2S,4S)-4-amino-1-[(4,5-dichlorothiophen-2-yl)sulfonyl]-N-methylpyrrolidine-2-carboxamide
9-[2-(1-methyl-1H-imidazol-2-yl)ethyl]-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
1-benzoyl-N-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]piperidin-4-amine
1-methyl-3-{2-oxo-2-[4-(pyridin-3-yloxy)piperidin-1-yl]ethyl}-3-(4-phenylphenyl)pyrrolidine-2,5-dione
methyl 3-({[5-(3-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}carbamoyl)benzoate
{[3-(1-benzofuran-2-yl)-1H-pyrazol-4-yl]methyl}(1,4-dioxan-2-ylmethyl)methylamine
4-[5-cyclopropyl-3-(2-phenylethyl)-1H-1,2,4-triazol-1-yl]-2-methylpyridine
5-[6-methyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]-1,2,3,4-tetrahydroisoquinoline
N-[3-methoxy-5-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-3-(2-methylpiperidin-1-yl)azetidine-1-carboxamide
3-[2-(2-methylphenyl)ethyl]-1-(1,3-thiazol-2-yl)piperidine
{6-[4-(3-phenylpropyl)-1,4-diazepane-1-carbonyl]pyridin-2-yl}methanol
1-(4-acetyl-6-hydroxy-1,4-diazepan-1-yl)-2-(3,4-dichlorophenyl)ethan-1-one
1-{[2-(4-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-3-ol
methyl 4-{[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]methyl}-1H-pyrazole-3-carboxylate
[(2-methoxypyrimidin-5-yl)methyl](methyl)(quinolin-5-ylmethyl)amine
ethyl 3-[(2-fluorophenyl)methyl]-1-[4-(2-oxopyrrolidin-1-yl)butanoyl]piperidine-3-carboxylate
N-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]-2-(morpholin-4-yl)-2-(pyridin-3-yl)acetamide
2-[2-(butan-2-yl)phenoxy]-1-[4-(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
1-{4-[4-(2-aminopropan-2-yl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}-3-(ethylsulfanyl)propan-1-one
2-[(3-methoxyphenyl)methyl]-8-[2-(propan-2-yloxy)acetyl]-2,8-diazaspiro[4.5]decan-3-one
(1S,5R)-3-[4-(benzyloxy)butanoyl]-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[(3-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}phenyl)methyl]-1H-pyrazole
methyl 5-[3-(2-hydroxyphenyl)-1H-pyrazole-5-carbonyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
1-methyl-9-(4-oxo-1,4-dihydroquinoline-2-carbonyl)-1,4,9-triazaspiro[5.5]undecan-5-one
3-[(4aR,7aS)-4-cyclopentanecarbonyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid
2-benzyl-9-(cyclopentylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-N'-(2-methylphenyl)propanediamide
(3S,9aR)-3-benzyl-8-[(2,5-dimethylphenyl)methyl]-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
8-[3-(5,6-dimethyl-1H-1,3-benzodiazol-2-yl)propanoyl]-2-methyl-2,8-diazaspiro[4.5]decan-3-one
N-(2-fluoropyridin-3-yl)-3-hydroxy-1-oxa-8-azaspiro[4.5]decane-8-carboxamide
N-[(3R,4S)-4-cyclopropyl-1-(pyrazine-2-carbonyl)pyrrolidin-3-yl]-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-3-carboxamide
2-({4-[4-(5-methylpyrimidin-2-yl)phenyl]-1H-pyrrolo[2,3-b]pyridin-6-yl}amino)ethan-1-ol
ethyl 1-(pyridin-4-ylmethyl)-5-[2-(1,3-thiazol-4-yl)acetyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-(3-cyclopentylpropyl)-2-(4-ethylpiperazin-1-yl)-2,3-dihydro-1H-indene-2-carboxamide
N-[(2-methoxyphenyl)methyl]-2-(morpholin-3-yl)-N-(pyridin-4-ylmethyl)acetamide