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2-({[(3R,4R)-1-[3-(difluoromethoxy)benzoyl]-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
1,3-dimethyl-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
N-(1-benzylpyrrolidin-3-yl)-3-[1-(pyrazin-2-yl)piperidin-4-yl]propanamide
5-{4-[(4-phenyl-4H-1,2,4-triazol-3-yl)methyl]piperidine-1-carbonyl}pyridine-2-carbonitrile
2-[3-(2-methylpropyl)-5-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidin-5-yl]-1H-1,2,4-triazol-1-yl]pyridine
2-{[2-(2H-1,3-benzodioxol-5-yl)-8-methoxy-2,3,4,5-tetrahydro-1,5-benzothiazepin-5-yl]methyl}phenol
2-methoxy-1-{1'-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}ethan-1-one
3-[(2,1,3-benzoxadiazol-4-ylmethyl)(methyl)amino]-N-methylbutanamide
5-{2-[5-(2-chloro-6-fluoro-3-methylphenyl)-4-phenyl-1H-imidazol-1-yl]ethyl}-1H-1,2,3,4-tetrazole
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-3-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)propanamide
1-{1-[5-(1H-imidazol-1-ylmethyl)pyridin-2-yl]piperidin-4-yl}piperidin-4-ol
1-[2-(morpholin-4-ylmethyl)phenyl]-3-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}urea
3-(2-phenylpropyl)-8-[2-(1H-1,2,4-triazol-1-yl)acetyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-(dimethylamino)-N-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}-2-(3-methylphenyl)acetamide
8-[4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzoyl]-1-oxa-8-azaspiro[4.5]decane
4-{3-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrol-5-yl]-3-oxopropyl}-N-methylbenzene-1-sulfonamide
N-[2-(2-fluorophenyl)-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]ethyl]-N,2-dimethylfuran-3-carboxamide
methyl 5-[(1-benzothiophen-2-ylmethyl)amino]-3-acetamido-1-(oxolan-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N,N-dimethyl-2-[(1S,5R)-3-[(1-methyl-1H-indol-2-yl)methyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
5-[(4-benzylpiperidin-1-yl)methyl]-N-methyl-N-(oxolan-2-ylmethyl)-1,2-oxazole-3-carboxamide
3-({[2-(2-ethoxyphenoxy)ethyl](methyl)amino}methyl)-4H-chromen-4-one
2-[3-(4-chlorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]pyridine-3-carbonitrile
N-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-3-(4-methyl-1,3-thiazol-5-yl)propanamide
6-(4-fluorophenyl)-N-methylimidazo[2,1-b][1,3]thiazole-3-carboxamide
1-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazin-1-yl}-2-(1-propylpiperidin-4-yl)ethan-1-one
1-{[5-methyl-2-(thiophen-3-yl)-1,3-oxazol-4-yl]methyl}-3-(3-methylphenoxymethyl)piperidine
2-(2-methoxy-5-methylphenyl)-2-[4-(pyridin-2-ylmethoxy)piperidin-1-yl]acetic acid
phenyl (7S,9aR)-8-methyl-7-(2-methylpropyl)-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate
1-{2-cyclopropyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}-4-(1H-pyrazol-1-ylmethyl)piperidine
N-methyl-2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)-N-[(4-methyl-1,3-thiazol-2-yl)methyl]acetamide
2-{2-[2-(4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]ethyl}-1,3-benzothiazole
1-benzyl-N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-1H-pyrazole-4-carboxamide
(4aR,8aS)-6-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-1-{[4-(trifluoromethyl)phenyl]methyl}-decahydro-1,6-naphthyridin-2-one
1-[3-(3-fluorophenoxymethyl)piperidin-1-yl]-2-methoxyethan-1-one
N-[1-(3,5-difluorophenyl)cyclopropyl]-1-(2-methoxyacetyl)piperidine-4-carboxamide
3-(5-methylfuran-2-yl)-N-[2-(2-oxoimidazolidin-1-yl)ethyl]-1H-pyrazole-5-carboxamide
2-[(2R)-2-aminopropanoyl]-N-methyl-N-(1,3-thiazol-2-ylmethyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
(3aS,6aR)-3-[3-(4-methoxyphenyl)propyl]-5-(pyrrolidine-1-sulfonyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
(1S,5R)-3-benzyl-6-{[2-(morpholin-4-yl)pyrimidin-5-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane
N-[(2,4-dimethoxyphenyl)methyl]-3-{1-[(4-hydroxyphenyl)methyl]piperidin-3-yl}propanamide
1-ethyl-N-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]-3-methylpiperidine-3-carboxamide
1-(2,6-difluoro-3-methoxybenzoyl)-4-[1-(pyrrolidin-1-yl)ethyl]piperidine
ethyl 1-{2-[1-(2-methoxyethyl)-3-(3-methoxyphenyl)-2,5-dioxopyrrolidin-3-yl]acetyl}piperidine-3-carboxylate
N-ethyl-5-(2-fluorophenoxymethyl)-N-[(5-methylfuran-2-yl)methyl]-1H-pyrazole-3-carboxamide
(1S,5R)-3-[2-(3-chloro-4-hydroxyphenyl)acetyl]-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(2-ethylphenyl)-2-{methyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}acetic acid
3-[5-(2H-1,3-benzodioxol-5-ylmethyl)-1,3,4-oxadiazol-2-yl]-N-[2-(4-methoxyphenyl)ethyl]propanamide
methyl({2-[4-(thiomorpholine-4-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}){[3-(trifluoromethyl)phenyl]methyl}amine
N-{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]ethyl}-5-methyl-1-propyl-1H-pyrazole-4-carboxamide
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carboxamide