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7-chloro-1-(2-phenoxyethyl)-3-{[(pyridin-3-ylmethyl)amino]methyl}-1,2-dihydroquinolin-2-one
2-(5-{[2-(ethoxymethyl)pyrrolidin-1-yl]methyl}furan-2-yl)-1-methyl-1H-1,3-benzodiazole
1-[2-(4-methylphenoxymethyl)furan-3-carbonyl]azepan-3-amine
(diphenylmethyl)({[6-(pyrrolidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl})amine
1-(4,7-dimethylquinazolin-2-yl)-N-(2-methoxyethyl)azepan-4-amine
N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-amine
5,6-dimethyl-N-{[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]methyl}thieno[2,3-d]pyrimidin-4-amine
1-(2-hydroxyethyl)-N-methyl-N-(quinolin-5-ylmethyl)-1H-1,3-benzodiazole-5-carboxamide
2-amino-6-{4-[3-(1-methylpiperidin-3-yl)propanoyl]piperazin-1-yl}-3,4-dihydropyrimidin-4-one
(5-{1-[3-(3-ethyl-1,2,4-oxadiazol-5-yl)phenyl]-1H-imidazol-2-yl}furan-2-yl)methanol
(2S,4R)-4-amino-N-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]pyrrolidine-2-carboxamide
(3R,4R)-1-{[3-(hydroxymethyl)-4-(propan-2-yloxy)phenyl]methyl}-4-{methyl[2-(pyridin-2-yl)ethyl]amino}piperidin-3-ol
(2R)-2-amino-3-(furan-2-yl)-N-methyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]propanamide
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}-3-(morpholin-4-yl)propanamide
N-{[5-(thiophen-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-[(2,3-difluorophenyl)methyl]-3-hydroxy-3-({[(3-methyl-1H-pyrazol-5-yl)methyl]amino}methyl)piperidin-2-one
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-N-methyl-1-(1-methylpiperidin-4-yl)piperidine-3-carboxamide
3-{1-[(2-aminopyridin-3-yl)methyl]piperidin-4-yl}-N-[(3-chlorophenyl)methyl]propanamide
1-[(3,4-dimethylphenyl)methyl]-N-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]piperidine-4-carboxamide
3-[2-(4-chlorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]piperidine
2-[ethyl({[(3R,4R)-4-(hydroxymethyl)-1-(1-methyl-1H-indole-4-carbonyl)pyrrolidin-3-yl]methyl})amino]ethan-1-ol
(1r,4r)-4-{[6-(dimethylamino)pyrimidin-4-yl]amino}cyclohexan-1-ol
N-[(3-fluoro-4-methylphenyl)methyl]-1-(4-methylquinazolin-2-yl)pyrrolidine-2-carboxamide
N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
1-{1-[(2-chloro-4-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-2-(4-fluorophenyl)piperidine
N-[(2R,3R)-1'-[(2,5-difluorophenyl)methyl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(methylsulfanyl)acetamide
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-2-(2-methyl-1H-indol-3-yl)acetamide
4-methyl-6-{[(1R,5R)-6-methyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]sulfonyl}quinolin-2-ol
3-(2-butyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[3-(pyridin-3-yloxy)propyl]propanamide
1-(4-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperazin-1-yl)-3-(dimethylamino)propan-2-ol
[(4-{1-azabicyclo[3.2.1]octan-5-yloxy}phenyl)methyl][(3-methylpyridin-4-yl)methyl]amine
methyl (2S,4S)-1-[(4-chlorophenyl)methyl]-4-propanamidopyrrolidine-2-carboxylate
(1H-imidazol-2-ylmethyl)(methyl)[(3-{[1-(naphthalene-2-sulfonyl)piperidin-4-yl]oxy}phenyl)methyl]amine
methyl 3-{[methyl(oxan-2-ylmethyl)carbamoyl]amino}benzoate
5-{[2-(2-acetamidoethyl)piperidin-1-yl]methyl}-2-methoxybenzoic acid
methyl (2S,4S,5R)-5-(2,3-difluorophenyl)-1-methyl-4-[(pyridin-4-ylmethyl)carbamoyl]pyrrolidine-2-carboxylate
4-phenyl-N-{[1-(4,4,4-trifluorobutanoyl)piperidin-3-yl]methyl}benzamide
{[3-(6-methoxynaphthalen-2-yl)-1H-pyrazol-4-yl]methyl}(methyl)[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amine
N-(3-cyanophenyl)-3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidine-1-carboxamide
N-[2-(2-fluorophenyl)-2-(pyrrolidin-1-yl)ethyl]-4-(1H-pyrazol-3-yl)benzamide
N-ethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-6-[(oxan-2-ylmethyl)amino]pyridine-3-carboxamide
5,7-dimethyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]pyrido[2,3-d]pyrimidin-4-amine
2-[(3R,4S)-3-amino-4-(5-methylfuran-2-yl)pyrrolidin-1-yl]-1-[(2R,6S)-2,6-dimethylmorpholin-4-yl]ethan-1-one
5,6-dimethyl-2-[6-oxo-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-2-yl]pyridine-3-carbonitrile
N-[3-(5-cyclopropyl-1H-pyrazol-1-yl)propyl]-3-(1-methylpiperidin-2-yl)propanamide
N,2-dimethyl-6-(propan-2-yl)-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}pyrimidin-4-amine
N,N-dimethyl-2-({5-[3-(3-methylbutanoyl)piperidine-1-carbonyl]pyridin-2-yl}amino)acetamide
4-hydroxy-3-methyl-N-{[1-(2-methylpropyl)piperidin-3-yl]methyl}benzamide
6-{4-[1-(2,2-dimethylpropyl)pyrrolidin-3-yl]piperidin-1-yl}pyridine-2-carbonitrile
4-[(6-methoxypyridin-3-yl)methyl]-3-methyl-1-(2-methylpropyl)piperazin-2-one