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2-{2-[6-(benzyloxy)-4-cyclohexyl-3-oxo-1,4-diazepan-1-yl]-2-oxoethyl}-4-methyl-1,2-dihydrophthalazin-1-one
4-{6-amino-1H-pyrrolo[2,3-b]pyridin-4-yl}-3-hydroxybenzoic acid
1-[(3-fluorophenyl)methyl]-N-[2-(3-methylpyridin-2-yl)ethyl]-6-oxopiperidine-3-carboxamide
1-[1-ethyl-5-(3-fluorobenzoyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]-4-phenylpiperazine
3-({5-[1-(4-fluorophenyl)-3,5-dimethyl-1H-pyrazol-4-yl]-1H,4H-pyrazolo[3,4-d]imidazol-1-yl}methyl)pyridine
6-methyl-2-({2-oxo-2-[3-(pyrimidin-4-yl)piperidin-1-yl]ethyl}sulfanyl)-3,4-dihydropyrimidin-4-one
3-(oxolan-3-yl)-1-(2-phenylethyl)-5-(pyrrolidin-1-ylmethyl)-1H-1,2,4-triazole
2-(2-methyl-1,3-thiazol-4-yl)-N-(1-phenylpiperidin-4-yl)acetamide
4-({4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidin-1-yl}methyl)pyridine
7-methoxy-N-[3-(1-methyl-1H-1,3-benzodiazol-2-yl)propyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-[(4-amino-6-{[2-(2-oxoimidazolidin-1-yl)ethyl]amino}pyrimidin-2-yl)sulfanyl]-N,N-dimethylacetamide
1-[2-chloro-5-(1H-pyrazol-1-yl)benzoyl]-4-(2-methoxyethyl)piperazine
2-[4-({1-[(2-fluorophenyl)methyl]-2-(propane-2-sulfonyl)-1H-imidazol-5-yl}methyl)piperazin-1-yl]ethan-1-ol
N-[2-(2-methoxyphenyl)ethyl]-4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}butanamide
3-(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine-5-carbonyl)-1,2-dihydroquinoxalin-2-one
1-{4-[({1-[(3-methoxyphenyl)methyl]piperidin-3-yl}amino)methyl]thiophen-2-yl}ethan-1-one
(3aR,6aR)-2-cyclopentyl-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
methyl({[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}){[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}amine
N-[1-(methoxymethyl)cyclopentyl]-2-(2-oxopyrrolidin-1-yl)propanamide
(5S,9aS,9bS)-5-(1-ethyl-3-methyl-1H-pyrazol-4-yl)-2-(3-methoxyphenyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-(oxolan-2-ylmethyl)-1-[1-(3-phenylpropyl)piperidin-4-yl]piperidine-4-carboxamide
N-[2-(1-{5-[(phenylsulfanyl)methyl]furan-2-carbonyl}piperidin-2-yl)ethyl]acetamide
N-(1,4-dioxan-2-ylmethyl)-N,5,7-trimethylpyrido[2,3-d]pyrimidin-4-amine
1-(4-methyl-1,3-thiazole-5-carbonyl)-N-[4-(3-methylphenyl)phenyl]piperidine-4-carboxamide
N-[1-methyl-4-(2-oxo-1,3-oxazolidin-3-yl)-1H-indazol-3-yl]cyclobutanecarboxamide
(2S,4S)-1-[(5-chlorothiophen-2-yl)methyl]-N-ethyl-4-[2-(methylsulfanyl)acetamido]pyrrolidine-2-carboxamide
3-cyclopropyl-N-(pyridin-4-yl)-1H-pyrazole-5-carboxamide
{[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}[1-(1,5-dimethyl-1H-pyrazol-4-yl)ethyl]amine
N-(1-{1-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1,2,5,6-tetrahydropyridin-3-yl}propyl)-N-methylacetamide
5-[(2S)-1-({4-[2-(1H-imidazol-1-yl)ethoxy]phenyl}methyl)pyrrolidin-2-yl]-3-methyl-1,2,4-oxadiazole
4-(2,4-dioxoimidazolidin-1-yl)-N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]benzamide
1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-5-methyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-1H-pyrazole-4-carboxamide
4-chloro-N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-N-methyl-2-propanamidobenzamide
3-(1-butyl-3-methyl-1H-pyrazol-5-yl)-1-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-1-(pyridin-3-ylmethyl)urea
ethyl 4-{7-acetamido-1-[2-(pyridin-2-yl)ethyl]-1H-1,3-benzodiazole-5-amido}piperidine-1-carboxylate
N-{[2-(4-acetylpiperazin-1-yl)pyridin-3-yl]methyl}-4-methoxy-3-methylbenzamide
N-(3,3-dimethyl-2-oxobutyl)-2-[(4S,6R)-6-methyl-2-sulfanylidene-1,3-diazinan-4-yl]acetamide
1-{[3-(4-methylpiperidine-1-carbonyl)-1,2-oxazol-5-yl]methyl}piperidin-4-ol
1-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1-methyl-1H-imidazole-2-carbonyl)piperidine
N-cyclopentyl-3-{[3-(1H-1,2,3-triazol-1-yl)propyl]sulfamoyl}benzamide
1-(3-{6-amino-1H-pyrrolo[2,3-b]pyridin-4-yl}-4-(morpholin-4-yl)phenyl)ethan-1-one
4-{3-cyclopropyl-5-[5-(propan-2-yl)-1,3-oxazol-4-yl]-1H-1,2,4-triazol-1-yl}-3-methylpyridine
{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}(2-methoxyethyl)(propan-2-yl)amine
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N-methylquinoline-3-carboxamide
1-(3-chlorophenyl)-4-[1-(dimethyl-1,3-thiazole-5-carbonyl)piperidin-3-yl]piperazine
(3aR,6aS)-1-oxo-5-{[4-(pyridin-2-yl)phenyl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-2-{3-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}acetamide
2-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridine-3-carbonitrile
(3S,4R)-1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-4-(3-methylthiophen-2-yl)piperidin-3-ol