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(3S,5S)-1-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propanoyl]-5-(pyrrolidine-1-carbonyl)piperidine-3-carboxylic acid
2-(2-fluorophenoxymethyl)-4-{4H,5H,6H,7H-thieno[3,2-c]pyridine-5-carbonyl}-1,3-oxazole
(3aR,5R,6S,7aS)-2-(6-fluoro-1H-1,3-benzodiazole-2-carbonyl)-octahydro-1H-isoindole-5,6-diol
5-(2,6-difluorophenoxymethyl)-N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-1,2-oxazole-3-carboxamide
1-[3-(morpholin-4-yl)propyl]-3-[1-(propan-2-yl)-1H-pyrazol-5-yl]urea
N-(4-{3-[3-(4-methylpiperazin-1-yl)-3-oxopropyl]piperidine-1-carbonyl}phenyl)acetamide
3-(pyridin-2-yl)-N-[2-(4-sulfamoylphenyl)ethyl]-1H-pyrazole-5-carboxamide
N-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}-N-(pyridin-4-ylmethyl)cyclopropanecarboxamide
methyl 2-{1-benzyl-8-[(4-acetamidophenyl)methyl]-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-3-yl}acetate
2-(dimethylamino)-2-(2-fluorophenyl)-1-[4-(4H-1,2,4-triazol-3-yl)piperidin-1-yl]ethan-1-one
{[3-(2,4-difluorophenyl)-1H-pyrazol-4-yl]methyl}[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]methylamine
N-(1-{1-[(4-methoxy-3-methylphenyl)methyl]piperidin-4-yl}-2-(3-methoxyphenyl)ethyl)-N-methylpyridine-2-carboxamide
N-[(2S)-3-methylbutan-2-yl]-1-[4-(1,3-thiazol-4-yl)phenyl]piperidin-4-amine
2-{4-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]piperazin-1-yl}-N-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-amine
3-(4-hydroxyphenyl)-N-[3-(4-methylpiperazin-1-yl)butyl]benzamide
N-(2-methyl-1-{7-[(4-methylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}propyl)furan-3-carboxamide
methyl (2R,4S)-4-hydroxy-1-[3-(4-methylphenyl)propanoyl]piperidine-2-carboxylate
N-(3-ethyl-4-methyl-1-phenyl-1H-pyrazol-5-yl)isoquinoline-5-carboxamide
8-{[4-(cyclopentyloxy)phenyl]methyl}-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
3-(3-hydroxy-3-methylbutyl)-N-{[4-(hydroxymethyl)phenyl]methyl}benzamide
2-{1-[(3-methylthiophen-2-yl)methyl]pyrrolidin-3-yl}benzoic acid
N-[(5-chloro-1-benzothiophen-3-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
4-amino-2-(2H-1,3-benzodioxol-5-yl)pyrimidine-5-carbonitrile
methyl 2-[2,4-dioxo-1-(2-phenylethyl)-8-(1,3-thiazol-2-ylmethyl)-1,3,8-triazaspiro[4.5]decan-3-yl]acetate
4-methyl-6-[4-(oxan-4-yl)piperazin-1-yl]-2-(pyridin-3-yl)pyrimidine
4-[(4-fluorophenyl)methyl]-3-{2-[4-(2-methoxyethyl)piperazin-1-yl]-2-oxoethyl}piperazin-2-one
1-[2-(piperidin-2-yl)ethyl]-N-{[4-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
2-(1-benzyl-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl)-N,N-dimethylacetamide
6-ethyl-N-methyl-N-[(5-propyl-1H-pyrazol-3-yl)methyl]pyrimidin-4-amine
2-(4-phenyl-1H-imidazol-5-yl)-4-(propan-2-yl)-1,3-thiazole
3-(4-hydroxyphenyl)-N-{3-[(4-methylphenyl)sulfanyl]propyl}-1H-pyrazole-5-carboxamide
3-[2-(4-benzylpiperidin-1-yl)-2-oxoethyl]-3-(2-methylphenyl)-1-(pyridin-3-ylmethyl)pyrrolidine-2,5-dione
1-[3-(4-methoxyphenyl)-1H-pyrazole-5-carbonyl]-3-(1-methyl-1H-imidazol-2-yl)piperidine
(1S,5R)-6-(cyclobutylmethyl)-3-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane
N-[2-(4-fluorophenyl)-2-(pyrrolidin-1-yl)ethyl]-3-[5-oxo-2-(thiophen-3-ylmethyl)pyrrolidin-2-yl]propanamide
1-[4-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]-2-(oxan-2-ylmethoxy)ethan-1-one
N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
1-{2-[2-(3-fluorophenyl)ethyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}-N-[(3S)-2-oxoazepan-3-yl]piperidine-4-carboxamide
(2S,4R)-4-amino-N,N-diethyl-1-(1-ethyl-6-methyl-2-oxo-1,2-dihydropyridine-3-carbonyl)pyrrolidine-2-carboxamide
1-benzyl-4-(5-phenyl-1,3,4-thiadiazol-2-yl)-1,4-diazepan-6-ol
(4aS,7aR)-1-[2-(3-methoxyphenoxy)acetyl]-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
8-cyclopropanecarbonyl-2-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
4-[(2S)-1-{3-fluoro-6-methylimidazo[1,2-a]pyridine-2-carbonyl}pyrrolidine-2-carbonyl]morpholine
4-(2-{[1-(5-propylpyrimidin-4-yl)piperidin-4-yl]amino}ethyl)phenol
1-(2-{[(2-ethoxypyridin-3-yl)methyl]amino}pyrimidin-4-yl)piperidin-3-ol
4-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
{[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}(methyl)[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amine
5-(2,4-difluorophenoxymethyl)-N-methyl-N-[4-(morpholin-4-yl)butyl]-1,2-oxazole-3-carboxamide
5-[3-(3-methoxyphenyl)-1H-pyrazol-5-yl]-3-(propan-2-yl)-1,2,4-oxadiazole
N-(2-{[5-(2,4-difluorophenoxymethyl)-1,2-oxazol-3-yl]formamido}ethyl)acetamide