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2-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]acetyl}-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
2-[(2E)-but-2-en-1-yl]-5-{octahydropyrrolo[1,2-a]piperazine-2-carbonyl}-1,3,4-oxadiazole
(2S,4R)-N-ethyl-4-[(naphthalen-1-ylmethyl)amino]-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
(2S,6S)-1-{imidazo[1,2-a]pyrimidin-6-ylmethyl}-4-methyl-2,6-bis(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine
N-{[2-(morpholin-4-yl)-1,3-thiazol-4-yl]methyl}-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
2-[4-(3-cyano-6-methylpyridin-2-yl)-1H-pyrazol-1-yl]-N-(1-propyl-1H-1,2,3-triazol-4-yl)acetamide
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(2-methyl-1,3-thiazole-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-{[5-chloro-7-(pyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(prop-2-en-1-yloxy)benzamide
N-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-3-(piperidine-1-carbonyl)benzene-1-sulfonamide
3-phenyl-1-{[6-(pyrrolidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}piperidine
methyl 3-[2-(3,4-difluorophenyl)acetyl]-7-oxo-9-(pyridin-2-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
methyl 1-(2-methylpropyl)-5-{[(6-methylpyridin-2-yl)methyl]amino}-3-(2-phenylacetamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
7-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-4-[(4-phenyl-1,3-thiazol-2-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-(2-hydroxyethyl)-2-[(3-methoxyphenyl)amino]-N-(1,3-thiazol-2-ylmethyl)butanamide
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-2-(5-methyl-3-oxo-2,3-dihydro-1H-pyrazol-4-yl)acetamide
N-cyclopentyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)pyrrolidine-2-carboxamide
methyl 3-methyl-4-({4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazine-1-carbonyl}amino)benzoate
[(2-chloro-6-fluorophenyl)methyl](methyl)({4-methyl-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)amine
4-(5-chloro-2-methylphenyl)-3-[2-(phenylamino)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
2-(1-cyclopentyl-4-{[2-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)ethan-1-ol
2-(4-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-2-yl)pyridine
6-[4-(piperidine-1-carbonyl)piperidin-1-yl]pyridine-2-carboxylic acid
5-[4-(morpholin-4-yl)piperidine-1-carbonyl]-N-(pyridin-4-ylmethyl)pyridin-2-amine
4-{[2-(2-aminoethyl)quinazolin-4-yl]amino}-1-(2-methoxyethyl)pyrrolidin-2-one
N-(1-benzylpyrrolidin-3-yl)-1-[4-(furan-2-yl)pyrimidin-2-yl]-5-(methoxymethyl)-1H-pyrazole-4-carboxamide
7-cyclopentyl-2-{2-[methyl(phenyl)amino]acetyl}-2,7-diazaspiro[4.5]decan-6-one
1-(2-fluoro-4-methoxyphenyl)-2-{imidazo[1,2-a]pyridine-2-carbonyl}-1H,2H,3H,4H,9H-pyrido[3,4-b]indole
N-(1H-indazol-4-yl)-4-(2-oxo-1,3-oxazolidin-3-yl)piperidine-1-carboxamide
3-(1,2,3,4-tetrahydroisoquinolin-5-yl)phenol
N-{[1-(dimethylamino)cyclohexyl]methyl}-5-(5-methylfuran-2-yl)-1,2,4-triazin-3-amine
3-(azetidine-1-carbonyl)-N-methyl-N-[2-(2-methylpiperidin-1-yl)ethyl]benzene-1-sulfonamide
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-3,6-dimethyl-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-N-methyl-1H-1,2,3-benzotriazole-5-carboxamide
ethyl 4-{2-[3-oxo-1-(pyridin-2-ylmethyl)piperazin-2-yl]acetamido}piperidine-1-carboxylate
{[6-({1-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]hex-5-en-2-yl}oxy)pyridin-3-yl]methyl}dimethylamine
N-[2-(3-chlorophenyl)ethyl]-3-(1-methylpiperidin-2-yl)propanamide
3-(5-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)propanoic acid
1-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidin-1-yl]-2-[methyl(pyridin-3-ylmethyl)amino]ethan-1-one
{[3-(2H-1,3-benzodioxol-5-yl)-1-phenyl-1H-pyrazol-4-yl]methyl}(methyl)[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amine
1-(2-fluoro-4-methanesulfonylphenyl)-4-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperazine
(4aR,7aS)-1-cyclobutanecarbonyl-4-(2,3-dihydro-1-benzofuran-5-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-cyclobutyl-5-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
3-{[(1-{1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperidin-4-yl)oxy]methyl}pyridine
3-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]pyridin-2-ol
N,N-diethyl-1-{[1-(3-phenylpropanoyl)piperidin-3-yl]methyl}-1H-1,2,3-triazole-4-carboxamide
(1-{2-[4-({[(4-chlorophenyl)methyl]amino}methyl)-3-methyl-1H-pyrazol-1-yl]ethyl}pyrrolidin-3-yl)methanol
[(1-methyl-1H-imidazol-2-yl)methyl](oxolan-2-ylmethyl)(thiophen-3-ylmethyl)amine
4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-[(1R)-1-(3-methoxyphenyl)ethyl]benzamide
2-cyclopropyl-5-[4-(1-hydroxy-3-phenylpropyl)piperidine-1-carbonyl]-3,4-dihydropyrimidin-4-one
4-[(3-chlorophenyl)methyl]-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol