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N-[2-(quinolin-8-yloxy)ethyl]-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)propanamide
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-[(3-methyl-1H-pyrazol-5-yl)methyl]piperidine-4-carboxamide
N-{[7-(5-acetylthiophen-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}cyclohex-1-ene-1-carboxamide
N-[4-(morpholin-4-ylmethyl)phenyl]-2-phenylpyrrolidine-1-carboxamide
N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propanamide
2-(3-methylphenoxy)-1-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}ethan-1-one
2-{[3-cyclopropyl-1-(3-methylpyridin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-4-methyl-1,2-dihydrophthalazin-1-one
4-[(2,4-dimethoxyphenyl)methyl]-9-methoxy-7-(quinolin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-methyl-1-{1-[5-(naphthalen-2-yl)-1,2,4-triazin-3-yl]piperidin-4-yl}butan-1-ol
2-{2-[(prop-2-en-1-yl)amino]benzoyl}-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
2-{1-[(2-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)acetamide
2-[9-(3-fluorobenzoyl)-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl]acetamide
8-(1-methyl-1H-indole-3-carbonyl)-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-2-(piperidin-1-yl)acetamide
3-(1-{[4-(benzyloxy)phenyl]methyl}piperidin-3-yl)-1-(pyrrolidin-1-yl)propan-1-one
methyl 2-{1-[5-(2-chloro-4-methoxyphenoxymethyl)-1,2-oxazol-3-yl]-N-methylformamido}acetate
3-[(1S,9aR)-octahydro-1H-quinolizin-1-yl]-N-{[2-(dimethylamino)-1,3-thiazol-4-yl]methyl}propanamide
1-[4-({[3-(1H-pyrazol-1-yl)propyl]amino}methyl)phenoxy]-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
{1-[1-(2-methylpropyl)-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-yl]piperidin-4-yl}methanol
6-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-5,6-dihydro-1,6-naphthyridin-5-one
1-{4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
N-{[4-(hydroxymethyl)phenyl]methyl}-2-(phenylamino)pyrimidine-5-carboxamide
ethyl 4-({3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}methyl)-1H-pyrazole-3-carboxylate
3-[(3R,4S)-1-[(2,3-difluoro-6-methoxyphenyl)methyl]-4-(morpholin-4-yl)piperidin-3-yl]propan-1-ol
14-(4-chloro-1-methyl-1H-indazol-3-yl)-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
N-[(3R,4S)-4-cyclopropyl-1-(2-hydroxyethyl)pyrrolidin-3-yl]-4,5-dimethylthiophene-2-carboxamide
1-{2-[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1H-1,3-benzodiazole
7-chloro-2-(1H-pyrazol-4-yl)quinoxaline
1-[2-({[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}amino)ethyl]imidazolidin-2-one
N-{[3-fluoro-5-(trifluoromethyl)phenyl]methyl}-3-methyl-1-propyl-1H-pyrazole-4-carboxamide
4-{5-[4-(difluoromethoxy)benzoyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-2-yl}-1H-pyrazole
(1H-indol-7-ylmethyl)(oxolan-2-ylmethyl)(thiophen-3-ylmethyl)amine
N-[5-(2-methoxyacetamido)-2-methylphenyl]-3-(1H-pyrazol-3-yl)piperidine-1-carboxamide
3-(furan-2-yl)-1-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidin-1-yl]propan-1-one
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-pentylacetamide
2-{4-[4-(2-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-1H-indole
N-benzyl-4-(1H-pyrazol-4-yl)-N-(1,3-thiazol-2-ylmethyl)butanamide
5-(2-{4-[(2-fluorophenyl)methyl]-1,4-diazepan-1-yl}-2-oxoethyl)imidazolidine-2,4-dione
2-[3-(1H-imidazol-1-ylmethyl)piperidin-1-yl]-5-methyl-4-(1-methyl-1H-pyrazol-4-yl)pyrimidine
N-{[2-(3-methoxyphenyl)-1,3-thiazol-5-yl]methyl}-2-(methylamino)acetamide
N-{4-[(5-methyl-4H-1,2,4-triazol-3-yl)methyl]phenyl}-1,1-dioxo-1λ6-thiomorpholine-4-carboxamide
N-(1-{2-[3-(4-methoxyphenoxymethyl)piperidin-1-yl]-2-oxoethyl}-1H-pyrazol-4-yl)-2-(2-methoxyphenyl)acetamide
2-(cyclopentylmethyl)-6-methyl-4-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]-N,N-bis(prop-2-en-1-yl)-1,4-dihydropyridine-3-carboxamide
N-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-6-phenylimidazo[2,1-b][1,3]thiazole-3-carboxamide
1-({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-4-(thiophene-2-carbonyl)piperazine
6-ethyl-N-[2-(4-fluorophenyl)ethyl]-2-oxo-1,2-dihydropyridine-4-carboxamide
N3-methyl-N5-[(3-methylphenyl)methyl]-N3-(2-methylpropyl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
2-{9-[(3,5-difluorophenyl)methyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}acetic acid
N-[2-(trimethyl-1H-pyrazol-1-yl)ethyl]-1H-1,3-benzodiazole-2-carboxamide